EE9400070A - Bioloogiliselt aktiivsed eburnameniini derivaadid, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess - Google Patents
Bioloogiliselt aktiivsed eburnameniini derivaadid, neid sisaldavad farmatseutilised segud ja nende valmistamise protsessInfo
- Publication number
- EE9400070A EE9400070A EE9400070A EE9400070A EE9400070A EE 9400070 A EE9400070 A EE 9400070A EE 9400070 A EE9400070 A EE 9400070A EE 9400070 A EE9400070 A EE 9400070A EE 9400070 A EE9400070 A EE 9400070A
- Authority
- EE
- Estonia
- Prior art keywords
- preparation
- pharmaceutical compositions
- biologically active
- compositions containing
- eburnamenine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D461/00—Heterocyclic compounds containing indolo [3,2,1-d,e] pyrido [3,2,1,j] [1,5]-naphthyridine ring systems, e.g. vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU9201911A HU209678B (en) | 1992-06-09 | 1992-06-09 | Process for producing biologically active eburnamenin-14-carbonyl-amino derivatives and pharmaceutical compositions containing them |
Publications (1)
Publication Number | Publication Date |
---|---|
EE9400070A true EE9400070A (et) | 1995-12-15 |
Family
ID=10982021
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EE9400070A EE9400070A (et) | 1992-06-09 | 1994-06-29 | Bioloogiliselt aktiivsed eburnameniini derivaadid, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess |
Country Status (18)
Country | Link |
---|---|
US (1) | US5510345A (et) |
EP (1) | EP0644885A1 (et) |
JP (1) | JPH07507793A (et) |
KR (1) | KR950701924A (et) |
AU (1) | AU4352493A (et) |
CA (1) | CA2136547A1 (et) |
CZ (1) | CZ307994A3 (et) |
EE (1) | EE9400070A (et) |
FI (1) | FI945780A (et) |
GR (1) | GR1001597B (et) |
HR (1) | HRP930957A2 (et) |
HU (1) | HU209678B (et) |
IL (1) | IL105942A0 (et) |
LT (1) | LT3118B (et) |
NZ (1) | NZ253308A (et) |
SI (1) | SI9300309A (et) |
WO (1) | WO1993025550A1 (et) |
ZA (1) | ZA934037B (et) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2005286648A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors |
CA2580787A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes |
MX2007003327A (es) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Derivados heterociclicos, y su uso como mediadores de estearoil-coa desaturasa. |
EP2269610A3 (en) | 2004-09-20 | 2011-03-09 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
TW200626138A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
CN101083992A (zh) | 2004-09-20 | 2007-12-05 | 泽农医药公司 | 抑制人硬脂酰CoA去饱和酶的哒嗪衍生物 |
AR051092A1 (es) | 2004-09-20 | 2006-12-20 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como inhibidores de la estearoil-coa |
WO2006034474A2 (en) * | 2004-09-23 | 2006-03-30 | Reddy Us Therapeutics, Inc. | Novel pyridine compounds, process for their preparation and compositions containing them |
CA2618646A1 (en) | 2005-06-03 | 2007-11-15 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
EP2276750A2 (en) * | 2008-03-27 | 2011-01-26 | Auckland Uniservices Limited | Substituted pyrimidines and triazines and their use in cancer therapy |
CN101928286A (zh) * | 2009-06-18 | 2010-12-29 | 谢开智 | 长春胺衍生物及制备方法 |
PT2968316T (pt) | 2013-03-13 | 2019-10-29 | Forma Therapeutics Inc | Derivados de 2-hidroxi-1-{4-[(4-fenilfenil)carbonil]piperazin-1-il}etano-1-ona e compostos relacionados como inibidores da sintase de ácidos gordos (fasn) para o tratamento do cancro |
US10774064B2 (en) | 2016-06-02 | 2020-09-15 | Cadent Therapeutics, Inc. | Potassium channel modulators |
SI3571193T1 (sl) | 2017-01-23 | 2022-04-29 | Cadent Therapeutics, Inc. | Modulatorji kalijevega kanalčka |
JP2022508945A (ja) | 2018-10-22 | 2022-01-19 | カデント セラピューティクス,インコーポレーテッド | カリウムチャネルモジュレーターの結晶形態 |
CN113382633A (zh) | 2018-10-29 | 2021-09-10 | 福马治疗股份有限公司 | (4-(2-氟-4-(1-甲基-1H-苯并[d]咪唑-5-基)苯甲酰基)哌嗪-1-基)(1-羟基环丙基)甲酮的固体形式 |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2176516B1 (et) * | 1972-03-22 | 1975-03-14 | Synthelabo | |
HU171663B (hu) * | 1975-09-01 | 1978-02-28 | Richter Gedeon Vegyeszet | Sposob poluchenija novykh proizvodnykh 14-skobka-zamehhennogo metil-skobka zakryta-vinkana |
US4547505A (en) * | 1983-03-25 | 1985-10-15 | Degussa Aktiengesellschaft | N-Phenyl-N-'-cycloalkylalkanoylpiperazine useful as analgetics and process for its production |
WO1987001706A2 (en) | 1985-09-12 | 1987-03-26 | The Upjohn Company | C20 through c26 amino steroids |
US5099019A (en) * | 1985-09-12 | 1992-03-24 | Upjohn Company | Amines useful in producing pharmaceutically active CNS compounds |
WO1987007895A1 (en) | 1986-06-23 | 1987-12-30 | The Upjohn Company | Androstane-type and cortical aminoesters |
JPH02502824A (ja) | 1987-04-03 | 1990-09-06 | ジ・アップジョン・カンパニー | アミノ‐9,10‐セコステロイド類 |
CA1338012C (en) | 1987-04-27 | 1996-01-30 | John Michael Mccall | Pharmaceutically active amines |
FR2644789B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 19-nor, 3-ceto comportant une chaine en 17 aminosubstituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
FR2644788B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 3-ceto comportant une chaine en 17 amino-substituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
FR2644787B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 21 aminosubstitues, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
CA2071000A1 (en) | 1990-01-26 | 1991-07-27 | John M. Mccall | 5-oxygenated-2,4,6-triaminopyrimidines |
-
1992
- 1992-06-09 HU HU9201911A patent/HU209678B/hu not_active IP Right Cessation
-
1993
- 1993-06-02 LT LTIP599A patent/LT3118B/lt not_active IP Right Cessation
- 1993-06-08 CA CA002136547A patent/CA2136547A1/en not_active Abandoned
- 1993-06-08 WO PCT/HU1993/000036 patent/WO1993025550A1/en not_active Application Discontinuation
- 1993-06-08 NZ NZ253308A patent/NZ253308A/en unknown
- 1993-06-08 AU AU43524/93A patent/AU4352493A/en not_active Abandoned
- 1993-06-08 EP EP93913456A patent/EP0644885A1/en not_active Withdrawn
- 1993-06-08 GR GR930100233A patent/GR1001597B/el unknown
- 1993-06-08 US US08/351,447 patent/US5510345A/en not_active Expired - Fee Related
- 1993-06-08 HR HR930957A patent/HRP930957A2/xx not_active Application Discontinuation
- 1993-06-08 IL IL105942A patent/IL105942A0/xx unknown
- 1993-06-08 CZ CZ943079A patent/CZ307994A3/cs unknown
- 1993-06-08 ZA ZA934037A patent/ZA934037B/xx unknown
- 1993-06-08 JP JP6501317A patent/JPH07507793A/ja active Pending
- 1993-06-09 SI SI9300309A patent/SI9300309A/sl unknown
-
1994
- 1994-06-29 EE EE9400070A patent/EE9400070A/et unknown
- 1994-12-08 FI FI945780A patent/FI945780A/fi not_active Application Discontinuation
- 1994-12-09 KR KR1019940704495A patent/KR950701924A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
ZA934037B (en) | 1994-01-06 |
HUT64540A (en) | 1994-01-28 |
US5510345A (en) | 1996-04-23 |
CA2136547A1 (en) | 1993-12-23 |
JPH07507793A (ja) | 1995-08-31 |
CZ307994A3 (en) | 1995-07-12 |
AU4352493A (en) | 1994-01-04 |
GR1001597B (el) | 1994-06-30 |
SI9300309A (sl) | 1993-12-31 |
LTIP599A (en) | 1994-07-15 |
HU209678B (en) | 1994-10-28 |
IL105942A0 (en) | 1993-10-20 |
FI945780A0 (fi) | 1994-12-08 |
HU9201911D0 (en) | 1992-09-28 |
EP0644885A1 (en) | 1995-03-29 |
LT3118B (en) | 1994-12-27 |
WO1993025550A1 (en) | 1993-12-23 |
NZ253308A (en) | 1995-11-27 |
HRP930957A2 (en) | 1995-02-28 |
KR950701924A (ko) | 1995-05-17 |
FI945780A (fi) | 1994-12-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EE9500080A (et) | Erütromütsiini derivaadid, nende valmistamismeetod ja neid sisaldav farmatseutiline kompositsioon | |
EE9700333A (et) | Substitueeritud 4-fenüülaminotiasoolid, nende valmistamise meetod ja neid sisaldavad farmakoloogilised kompositsioonid | |
EE9400455A (et) | Peptiidi derivaadid, nende valmistamise protsess, neid sisaldavad ravimpreparaadid ja nende kasutamine | |
EE03609B1 (et) | Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid | |
EE03002B1 (et) | 1,3-oksatiolaannukleosiidi analoogid, neid sisaldavad ravimpreparaadid ja nende valmistamise meetod | |
FI942913A0 (fi) | Isatiinijohdannaiset, menetelmät niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset | |
EE03111B1 (et) | Glükokortikosteroidi epimeerid, nende valmistamise protsessid ja neid sisaldavad ravimpreparaadid | |
EE9400070A (et) | Bioloogiliselt aktiivsed eburnameniini derivaadid, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess | |
EE9800426A (et) | Asendatud 2,4-tiasolidiindiooni derivaadid, nende valmistamismeetodid ja neid sisaldavad farmatseutilised kompositsioonid | |
FI951789A0 (fi) | Uusia taksaanijohdannaisia, niiden valmistus ja niitä sisältävät farmaseuttiset koostumukset | |
IL104356A0 (en) | Benzofuranyl-and thiophenylmethylthio-alkanecarboxylic acid derivatives,their preparation and pharmaceutical compositions containing them | |
FI945781A0 (fi) | Uudet pregnaanirungon sisältävät steroidit, niitä sisältävät farmaseuttiset koostumukset ja menetelmä niiden valmistamiseksi | |
IL97501A0 (en) | 4-pyridone derivatives,their preparation and pharmaceutical compositions containing them | |
FI960316A (fi) | Oksatiolaanit, menetelmä niiden valmistamiseksi ja niitä sisältävät farmaseuttiset koostumukset | |
EE9400148A (et) | Tienotiasiini derivaadid, nende valmistamise meetod ja neid sisaldavad farmatseutilised preparaadid | |
IL106549A0 (en) | Heterocyclic derivatives,their preparation and pharmaceutical compositions containing them | |
FI951561A0 (fi) | Uudet 17 -substituoidut 4-androstaanijohdannaiset, niitä sisältävät farmaseuttiset koostumukset ja menetelmä niiden valmistamiseksi | |
AU8917891A (en) | Poly-aminopyrrolecarboxamido derivatives, processes for their preparation and pharmaceutical compositions containing them | |
IL105370A0 (en) | Propenoyl-imidazole derivatives,their preparation and pharmaceutical compositions containing them | |
IL104347A0 (en) | Substituted benzimidazole derivatives,their preparation and pharmaceutical compositions containing them | |
EE04347B1 (et) | 8-asabitsüklo[3.2.1]oktaan-3-metaanamiini derivaadid, neid sisaldav ravim ja farmatseutiline kompositsioon | |
FI942675A0 (fi) | Uudet substituoidut oksatsinoisokinoliinijohdannaiset, niitä sisältävät farmaseuttiset koostumukset sekä menetelmä niiden valmistamiseksi | |
IL104840A0 (en) | Sulphonylbenzyl-substituted imidazolylpropenoic acid derivatives,their preparation and pharmaceutical compositions containing them | |
IL104892A0 (en) | Substituted phenylquinazoline derivatives,their preparation and pharmaceutical compositions containing them | |
FI972129A (fi) | 6-metoksi-1H-bentsotriatsoli-5-karboksamidijohdannaisia, menetelmä niiden valmistamiseksi ja niitä sisältäviä lääkekoostumuksia |