PT876388E - Derivados de eritromicina triciclica - Google Patents

Derivados de eritromicina triciclica

Info

Publication number
PT876388E
PT876388E PT96936579T PT96936579T PT876388E PT 876388 E PT876388 E PT 876388E PT 96936579 T PT96936579 T PT 96936579T PT 96936579 T PT96936579 T PT 96936579T PT 876388 E PT876388 E PT 876388E
Authority
PT
Portugal
Prior art keywords
trycyclic
compounds
erythromycin derivatives
antibacterial
erythromycin
Prior art date
Application number
PT96936579T
Other languages
English (en)
Inventor
Kenneth P Spina
Robert Hallas
Richard L Edelson
Daniel T Chu
Yat Sun Or
Ly Tam Phan
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of PT876388E publication Critical patent/PT876388E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
PT96936579T 1995-11-08 1996-10-17 Derivados de eritromicina triciclica PT876388E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55524695A 1995-11-08 1995-11-08

Publications (1)

Publication Number Publication Date
PT876388E true PT876388E (pt) 2004-07-30

Family

ID=24216555

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96936579T PT876388E (pt) 1995-11-08 1996-10-17 Derivados de eritromicina triciclica

Country Status (12)

Country Link
EP (1) EP0876388B1 (pt)
JP (1) JP2000500133A (pt)
KR (1) KR19990067492A (pt)
AT (1) ATE259823T1 (pt)
AU (1) AU7447096A (pt)
DE (1) DE69631609T2 (pt)
DK (1) DK0876388T3 (pt)
ES (1) ES2218604T3 (pt)
IL (1) IL123551A0 (pt)
MX (1) MX9803692A (pt)
PT (1) PT876388E (pt)
WO (1) WO1997017356A1 (pt)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6274715B1 (en) * 1995-11-08 2001-08-14 Abbott Laboratories Tricyclic erythromycin derivatives
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
ATE299508T1 (de) * 1996-09-04 2005-07-15 Abbott Lab 6-o-substituierte ketoliden mit antibakteriellen wirkung
US5922683A (en) * 1997-05-29 1999-07-13 Abbott Laboratories Multicyclic erythromycin derivatives
DK0984975T3 (da) * 1997-05-29 2003-08-11 Abbott Lab Multicykliske erythromycinderivater
ZA987689B (en) * 1997-09-02 1999-02-24 Abbott Lab 3-descladinose 6-O substituted erythromycin derivatives
US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
KR20010030807A (ko) * 1997-09-30 2001-04-16 스티븐 에프. 웨인스톡 항균 활성을 갖는 3'-n-변형된, 6-o-치환된에리트로마이신 케톨리드 유도체
AR015986A1 (es) * 1997-10-29 2001-05-30 Abbott Lab Derivados de eritromicina puenteados en 6,11, composiciones farmaceuticas que los contienen, su uso para la manufactura de un medicamento y procedimientospara su preparacion
US6124269A (en) * 1997-10-29 2000-09-26 Abbott Laboratories 2-Halo-6-O-substituted ketolide derivatives
US6046171A (en) * 1997-10-29 2000-04-04 Abbott Laboratories 6,11-bridged erythromycin derivatives
PA8461401A1 (es) 1997-10-29 2000-05-24 Pfizer Prod Inc Derivados de eritromicina triciclicos
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
ATE243219T1 (de) * 1998-04-24 2003-07-15 Pfizer Prod Inc 9a, 11b-dehydro derivative von 9-oxime-3-keto-6-0-methylerythromycin
WO1999062920A1 (en) * 1998-06-03 1999-12-09 Pfizer Products Inc. Tricyclic 3-keto derivatives of 6-o-methylerythromycin
FR2780977B1 (fr) * 1998-07-09 2000-09-01 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
JP4573925B2 (ja) 1998-07-09 2010-11-04 アベンティス・ファーマ・ソシエテ・アノニム 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
JP2005503416A (ja) 2001-09-17 2005-02-03 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド 6−o−カルバメート−11,12−ラクト−ケトライド抗菌剤
CA2469304A1 (en) 2001-12-05 2003-06-19 Ortho-Mcneil Pharmaceutical, Inc. 6-o acyl ketolide antibacterials
CN1671726A (zh) * 2002-05-31 2005-09-21 詹森药业有限公司 3-脱克拉定糖基-6-o-氨基甲酰基和6-o-烷氧基羰基大环内酯抗菌药
ES2331867B1 (es) 2008-07-17 2010-10-27 Entrechem, S.L. Sintesis enzimatica de derivados enantiomericamente enriquecidos de trans-ciclopentano- 1,2-diaminas.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69127457T2 (de) * 1990-11-28 1998-01-22 Taisho Pharmaceutical Co Ltd 6-0-methylerythromycin a-derivat
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
WO1993021200A1 (fr) * 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. Derive de 5-o-desosaminylerythronolide a

Also Published As

Publication number Publication date
DE69631609T2 (de) 2005-01-05
IL123551A0 (en) 1998-10-30
ATE259823T1 (de) 2004-03-15
KR19990067492A (ko) 1999-08-25
JP2000500133A (ja) 2000-01-11
DE69631609D1 (en) 2004-03-25
ES2218604T3 (es) 2004-11-16
EP0876388A1 (en) 1998-11-11
MX9803692A (es) 1998-09-30
WO1997017356A1 (en) 1997-05-15
DK0876388T3 (da) 2004-06-07
EP0876388B1 (en) 2004-02-18
AU7447096A (en) 1997-05-29

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