ATE259823T1 - Tricyclische erythromycinderivate - Google Patents

Tricyclische erythromycinderivate

Info

Publication number
ATE259823T1
ATE259823T1 AT96936579T AT96936579T ATE259823T1 AT E259823 T1 ATE259823 T1 AT E259823T1 AT 96936579 T AT96936579 T AT 96936579T AT 96936579 T AT96936579 T AT 96936579T AT E259823 T1 ATE259823 T1 AT E259823T1
Authority
AT
Austria
Prior art keywords
compounds
erythromycin derivatives
tricyclic
tricyclic erythromycin
antibacterial
Prior art date
Application number
AT96936579T
Other languages
English (en)
Inventor
Yat Sun Or
Ly Tam Phan
Daniel T Chu
Kenneth P Spina
Robert Hallas
Richard L Elliott
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Application granted granted Critical
Publication of ATE259823T1 publication Critical patent/ATE259823T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT96936579T 1995-11-08 1996-10-17 Tricyclische erythromycinderivate ATE259823T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55524695A 1995-11-08 1995-11-08
PCT/US1996/016585 WO1997017356A1 (en) 1995-11-08 1996-10-17 Tricyclic erythromycin derivatives

Publications (1)

Publication Number Publication Date
ATE259823T1 true ATE259823T1 (de) 2004-03-15

Family

ID=24216555

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96936579T ATE259823T1 (de) 1995-11-08 1996-10-17 Tricyclische erythromycinderivate

Country Status (12)

Country Link
EP (1) EP0876388B1 (de)
JP (1) JP2000500133A (de)
KR (1) KR19990067492A (de)
AT (1) ATE259823T1 (de)
AU (1) AU7447096A (de)
DE (1) DE69631609T2 (de)
DK (1) DK0876388T3 (de)
ES (1) ES2218604T3 (de)
IL (1) IL123551A0 (de)
MX (1) MX9803692A (de)
PT (1) PT876388E (de)
WO (1) WO1997017356A1 (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6274715B1 (en) * 1995-11-08 2001-08-14 Abbott Laboratories Tricyclic erythromycin derivatives
ATE296831T1 (de) * 1996-09-04 2005-06-15 Abbott Lab 6-0-substituierte ketoliden mit antibakteriellen wirkung
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
US5922683A (en) * 1997-05-29 1999-07-13 Abbott Laboratories Multicyclic erythromycin derivatives
DK0984975T3 (da) * 1997-05-29 2003-08-11 Abbott Lab Multicykliske erythromycinderivater
ZA987689B (en) * 1997-09-02 1999-02-24 Abbott Lab 3-descladinose 6-O substituted erythromycin derivatives
US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
IL134608A0 (en) * 1997-09-30 2001-04-30 Abbott Lab 3'-n- modified 6-o-substituted erythromycin ketolide derivatives having antibacterial activity
US6124269A (en) * 1997-10-29 2000-09-26 Abbott Laboratories 2-Halo-6-O-substituted ketolide derivatives
US6046171A (en) * 1997-10-29 2000-04-04 Abbott Laboratories 6,11-bridged erythromycin derivatives
CO4990972A1 (es) * 1997-10-29 2000-12-26 Abbott Lab Derivados de eritromicina en puente 6,11
PA8461401A1 (es) 1997-10-29 2000-05-24 Pfizer Prod Inc Derivados de eritromicina triciclicos
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
PT952157E (pt) 1998-04-24 2003-11-28 Pfizer Prod Inc Derivados 9a, 11b-desidro de 9-oxima-3-ceto-6-o-metileritromicina
AU3439899A (en) 1998-06-03 1999-12-20 Pfizer Products Inc. Tricyclic 3-keto derivatives of 6-o-methylerythromycin
FR2780977B1 (fr) * 1998-07-09 2000-09-01 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
JP4573925B2 (ja) * 1998-07-09 2010-11-04 アベンティス・ファーマ・ソシエテ・アノニム 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
WO2003024986A1 (en) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. 6-o-carbamate-11,12-lacto-ketolide antimicrobials
CA2469304A1 (en) 2001-12-05 2003-06-19 Ortho-Mcneil Pharmaceutical, Inc. 6-o acyl ketolide antibacterials
WO2003102010A1 (en) * 2002-05-31 2003-12-11 Janssen Pharmaceutica N.V. 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents
ES2331867B1 (es) 2008-07-17 2010-10-27 Entrechem, S.L. Sintesis enzimatica de derivados enantiomericamente enriquecidos de trans-ciclopentano- 1,2-diaminas.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2104889T3 (es) * 1990-11-28 1997-10-16 Taisho Pharmaceutical Co Ltd Derivado de 6-o-metileritromicina a.
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
DE69301916T2 (de) * 1992-04-22 1996-08-08 Taisho Pharmaceutical Co., Ltd., Tokio/Tokyo 5-0-desosaminylerythronolid a derivate

Also Published As

Publication number Publication date
MX9803692A (es) 1998-09-30
EP0876388B1 (de) 2004-02-18
EP0876388A1 (de) 1998-11-11
WO1997017356A1 (en) 1997-05-15
AU7447096A (en) 1997-05-29
IL123551A0 (en) 1998-10-30
PT876388E (pt) 2004-07-30
DE69631609T2 (de) 2005-01-05
DE69631609D1 (en) 2004-03-25
JP2000500133A (ja) 2000-01-11
KR19990067492A (ko) 1999-08-25
DK0876388T3 (da) 2004-06-07
ES2218604T3 (es) 2004-11-16

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