DK0638317T3 - Farmaceutisk præparat, der indeholder glucosidase- og/eller amylasehæmmere og lipasehæmmer - Google Patents

Farmaceutisk præparat, der indeholder glucosidase- og/eller amylasehæmmere og lipasehæmmer

Info

Publication number
DK0638317T3
DK0638317T3 DK94111436T DK94111436T DK0638317T3 DK 0638317 T3 DK0638317 T3 DK 0638317T3 DK 94111436 T DK94111436 T DK 94111436T DK 94111436 T DK94111436 T DK 94111436T DK 0638317 T3 DK0638317 T3 DK 0638317T3
Authority
DK
Denmark
Prior art keywords
inhibitors
pharmaceutical preparation
preparation containing
amylase
lipase
Prior art date
Application number
DK94111436T
Other languages
English (en)
Inventor
Klaus-Dieter Bremer
Pavel Sawlewicz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of DK0638317T3 publication Critical patent/DK0638317T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
DK94111436T 1993-08-05 1994-07-22 Farmaceutisk præparat, der indeholder glucosidase- og/eller amylasehæmmere og lipasehæmmer DK0638317T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH233993 1993-08-05

Publications (1)

Publication Number Publication Date
DK0638317T3 true DK0638317T3 (da) 2000-06-26

Family

ID=4231504

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94111436T DK0638317T3 (da) 1993-08-05 1994-07-22 Farmaceutisk præparat, der indeholder glucosidase- og/eller amylasehæmmere og lipasehæmmer

Country Status (24)

Country Link
US (1) US5643874A (da)
EP (1) EP0638317B1 (da)
JP (1) JP2780932B2 (da)
KR (1) KR100342285B1 (da)
CN (1) CN1076196C (da)
AT (1) ATE190503T1 (da)
AU (1) AU684793B2 (da)
BR (1) BR9403170A (da)
CA (1) CA2128044C (da)
CZ (1) CZ286202B6 (da)
DE (1) DE59409200D1 (da)
DK (1) DK0638317T3 (da)
ES (1) ES2144019T3 (da)
GR (1) GR3033643T3 (da)
HU (1) HU222346B1 (da)
IL (1) IL110510A (da)
NO (1) NO313490B1 (da)
NZ (1) NZ264142A (da)
PL (1) PL175997B1 (da)
PT (1) PT638317E (da)
RU (1) RU2141844C1 (da)
SA (1) SA94150156B1 (da)
TW (1) TW381025B (da)
ZA (1) ZA945673B (da)

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US6267952B1 (en) * 1998-01-09 2001-07-31 Geltex Pharmaceuticals, Inc. Lipase inhibiting polymers
DE19802700A1 (de) * 1998-01-24 1999-07-29 Bayer Ag Verfahren zur Herstellung einer im Mund schnell zerfallenden Arzneiform, die als Wirkstoff Acarbose enthält
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EP1143999B1 (en) * 1999-01-22 2004-07-21 Hunza di Pistolesi Elvira & C. S.a.S. Lipoprotein complexes and compositions containing them
AR025587A1 (es) 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones en dispersion que contienen inhibidores de lipasa
US6235305B1 (en) * 1999-10-29 2001-05-22 2Pro Chemical Essentially nonabsorbable lipase inhibitor derivatives, pharmaceutical compositions and methods of use therefor
US6342519B2 (en) * 1999-10-29 2002-01-29 2 Pro Chemical Oxetanone derivatives
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US6348492B1 (en) * 1999-10-29 2002-02-19 2Pro Chemical Oxetanone derivatives
KR100349334B1 (ko) * 1999-12-08 2002-08-21 박관화 아카비오신 글루코실 시몬진 및 그것의 제조방법.
US7713546B1 (en) 2001-04-03 2010-05-11 Soft Gel Technologies, Inc. Corosolic acid formulation and its application for weight-loss management and blood sugar balance
ES2240516T3 (es) * 2000-07-28 2005-10-16 F. Hoffmann-La Roche Ag Nuevo uso de los inhibidores de lipasa.
PL204443B1 (pl) * 2000-07-28 2010-01-29 Hoffmann La Roche Kompozycja farmaceutyczna zawierająca inhibitor lipazy, sposób wytwarzania kompozycji farmaceutycznej, zestaw do leczenia otyłości, zastosowanie kompozycji farmaceutycznej oraz zastosowanie orlistatu i substancji wiążącej kwasy żółciowe
US6849609B2 (en) * 2001-04-10 2005-02-01 James U. Morrison Method and composition for controlled release acarbose formulations
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US7649002B2 (en) 2004-02-04 2010-01-19 Pfizer Inc (3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
US20060185357A1 (en) * 2004-05-07 2006-08-24 Kovacevich Ian D Independently drawing and tensioning lines with bi-directional rotary device having two spools
EP1744772B1 (en) 2004-05-10 2017-08-16 University of Copenhagen Flaxseeds for body weight management
US20060029567A1 (en) 2004-08-04 2006-02-09 Bki Holding Corporation Material for odor control
AP2007003979A0 (en) * 2004-11-23 2007-06-30 Warner Lambert Co 7-(2h-pyrazol-3-yl)-3,5-dihyroxy-heptanoic acid derivatives as hmg co-a reductase inhibitors for thetreatment of lipidemia
US8283312B2 (en) * 2005-02-04 2012-10-09 The Research Foundation Of State University Of New York Compositions and methods for modulating body weight and treating obesity-related disorders
US20060229261A1 (en) * 2005-04-12 2006-10-12 John Devane Acarbose methods and formulations for treating chronic constipation
US20070009615A1 (en) * 2005-04-29 2007-01-11 Litao Zhong Compositions and methods for controlling glucose uptake
US20090208584A1 (en) * 2005-06-09 2009-08-20 Tomohiro Yoshinari Solid preparation
WO2007015162A1 (en) * 2005-08-04 2007-02-08 Pfizer Limited Piperidinoyl-pyrrolidine and piperidinoyl-piperidine compounds
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US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
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AR063275A1 (es) * 2006-10-12 2009-01-14 Epix Delaware Inc Compuestos de carboxamida, una composicion farmaceutica que los comprende y su uso en la preparacion de un medicamento para el tratamiento de enfermedades mediadas por la activacion de ccr2.
CN101583593A (zh) 2006-11-13 2009-11-18 辉瑞产品公司 二芳基、二吡啶基和芳基-吡啶基衍生物及其用途
AU2007323193A1 (en) * 2006-11-20 2008-05-29 Glenmark Pharmaceuticals S.A. Acetylene derivatives as Stearoyl CoA Desaturase inhibitors
JP5498168B2 (ja) 2006-12-01 2014-05-21 ブリストル−マイヤーズ スクイブ カンパニー アテローム性動脈硬化および循環器疾患の治療のためのｃｅｔｐ阻害剤としてのｎ−（（３−ベンジル）−２，２−（ビス−フェニル）−プロパン−１−アミン誘導体
SI2002825T1 (sl) * 2007-06-14 2013-10-30 Krka Farmacevtski sestavki, ki obsegajo orlistat
EP2625968A1 (en) * 2007-09-12 2013-08-14 Københavns Universitet Composition and methods for increasing the suppression of hunger and reducing the digestibility of non-fat energy satiety
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JP5752359B2 (ja) * 2010-02-25 2015-07-22 富士フイルム株式会社 体重増加抑制組成物及びこれを含む食品
JP2013528172A (ja) 2010-05-21 2013-07-08 ファイザー・インク ２−フェニルベンゾイルアミド
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JP2016510306A (ja) * 2012-05-08 2016-04-07 セリックスビオ プライヴェート リミテッド 高血糖の治療のための組成物及び方法
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Also Published As

Publication number Publication date
BR9403170A (pt) 1995-04-18
HU9402249D0 (en) 1994-09-28
SA94150156B1 (ar) 2005-05-15
ZA945673B (en) 1995-02-07
CN1076196C (zh) 2001-12-19
NO942900L (no) 1995-02-06
KR100342285B1 (ko) 2002-10-25
IL110510A (en) 1999-03-12
HUT68300A (en) 1995-06-28
RU94028653A (ru) 1996-09-10
PT638317E (pt) 2000-07-31
HU222346B1 (hu) 2003-06-28
JP2780932B2 (ja) 1998-07-30
NO942900D0 (da) 1994-08-04
US5643874A (en) 1997-07-01
ATE190503T1 (de) 2000-04-15
PL175997B1 (pl) 1999-03-31
KR950005319A (ko) 1995-03-20
EP0638317B1 (de) 2000-03-15
AU6883994A (en) 1995-02-16
NO313490B1 (no) 2002-10-14
JPH0753409A (ja) 1995-02-28
IL110510A0 (en) 1994-11-11
ES2144019T3 (es) 2000-06-01
RU2141844C1 (ru) 1999-11-27
CA2128044A1 (en) 1995-02-06
DE59409200D1 (de) 2000-04-20
CZ286202B6 (cs) 2000-02-16
TW381025B (en) 2000-02-01
CZ182594A3 (en) 1995-02-15
CN1106701A (zh) 1995-08-16
NZ264142A (en) 1996-11-26
PL304557A1 (en) 1995-02-06
GR3033643T3 (en) 2000-10-31
EP0638317A1 (de) 1995-02-15
AU684793B2 (en) 1998-01-08
CA2128044C (en) 2007-02-20

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