DE69838651D1 - Erythromycinderivate - Google Patents

Erythromycinderivate

Info

Publication number
DE69838651D1
DE69838651D1 DE69838651T DE69838651T DE69838651D1 DE 69838651 D1 DE69838651 D1 DE 69838651D1 DE 69838651 T DE69838651 T DE 69838651T DE 69838651 T DE69838651 T DE 69838651T DE 69838651 D1 DE69838651 D1 DE 69838651D1
Authority
DE
Germany
Prior art keywords
erythromycin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69838651T
Other languages
English (en)
Other versions
DE69838651T2 (de
DE69838651T9 (de
Inventor
Yong-Jin Wu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of DE69838651D1 publication Critical patent/DE69838651D1/de
Publication of DE69838651T2 publication Critical patent/DE69838651T2/de
Application granted granted Critical
Publication of DE69838651T9 publication Critical patent/DE69838651T9/de
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
DE69838651T 1998-01-02 1998-12-21 Erythromycin-Derivate Expired - Fee Related DE69838651T9 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7035898P 1998-01-02 1998-01-02
US70358P 1998-01-02

Publications (3)

Publication Number Publication Date
DE69838651D1 true DE69838651D1 (de) 2007-12-13
DE69838651T2 DE69838651T2 (de) 2008-03-06
DE69838651T9 DE69838651T9 (de) 2008-06-12

Family

ID=22094819

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69838651T Expired - Fee Related DE69838651T9 (de) 1998-01-02 1998-12-21 Erythromycin-Derivate

Country Status (36)

Country Link
US (1) US6825171B2 (de)
EP (2) EP1044208A1 (de)
JP (1) JP2002500231A (de)
KR (1) KR20010033822A (de)
CN (1) CN1285841A (de)
AP (1) AP1060A (de)
AR (5) AR012764A1 (de)
AT (1) ATE377018T1 (de)
AU (1) AU759019B2 (de)
BG (1) BG104640A (de)
BR (1) BR9812992A (de)
CA (1) CA2317131C (de)
CO (1) CO4970773A1 (de)
CZ (1) CZ20002456A3 (de)
DE (1) DE69838651T9 (de)
DZ (1) DZ2699A1 (de)
EA (1) EA200000600A1 (de)
ES (1) ES2294641T3 (de)
GT (1) GT199800207A (de)
HR (1) HRP20000444A2 (de)
HU (1) HUP0100566A3 (de)
IL (1) IL136721A0 (de)
IS (1) IS5527A (de)
MA (1) MA26588A1 (de)
NO (1) NO20003346L (de)
NZ (1) NZ504987A (de)
OA (1) OA11440A (de)
PA (1) PA8465901A1 (de)
PE (1) PE20000119A1 (de)
PL (1) PL341647A1 (de)
SK (1) SK9772000A3 (de)
TN (1) TNSN98236A1 (de)
UY (2) UY25331A1 (de)
WO (1) WO1999035157A1 (de)
YU (1) YU40900A (de)
ZA (1) ZA9811940B (de)

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EP1137654A1 (de) 1998-12-10 2001-10-04 Pfizer Products Inc. Carbamat- und carbazat-ketolide antibiotika
EP1298138B1 (de) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamat und Carbazat Ketolid Antibiotika
EP1749832A3 (de) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamat und Carbazat Ketolid Antibiotika
EP1754700A3 (de) 1999-01-27 2007-05-09 Kosan Biosciences, Inc. synthese von oligoketiden
SK10172001A3 (sk) 1999-01-27 2002-06-04 Pfizer Products Inc. Ketolidové antibiotiká
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6458771B1 (en) 1999-04-16 2002-10-01 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
MXPA01010524A (es) 1999-04-16 2002-03-14 Kosan Biosciences Inc Agentes macrolidos anti-infecciosos.
US6939861B2 (en) 1999-04-16 2005-09-06 Kosan Biosciences, Inc. Amido macrolides
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US6514944B2 (en) 1999-04-16 2003-02-04 Kosan Biosciences, Inc. Macrolide antiinfective agents
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ID27331A (id) * 1999-09-29 2001-03-29 Pfizer Prod Inc Pembuatan antibiotik-antibiotik ketolida karbamat
EP1114826A3 (de) * 1999-12-29 2001-10-31 Pfizer Products Inc. Antibakterielle und prokinetische Makroliden
US6562795B2 (en) 2000-02-18 2003-05-13 Kosan Biosciences, Inc. Motilide compounds
US20020115621A1 (en) 2000-08-07 2002-08-22 Wei-Gu Su Macrolide antibiotics
US6472372B1 (en) 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
US6756359B2 (en) 2001-07-03 2004-06-29 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
CA2460947A1 (en) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. 6-o-carbamate-11,12-lacto-ketolide antimicrobials
BR0214748A (pt) 2001-12-05 2004-11-23 Ortho Mcneil Pharm Inc Derivados 6-oacil-cetolidas de eritromicina, úteis como antibacterianos
AU2003234650A1 (en) 2002-05-31 2003-12-19 Janssen Pharmaceutica N.V. 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents
JP2006524706A (ja) 2003-04-25 2006-11-02 カイロン コーポレイション 新規なケトライド誘導体
PT1836211E (pt) 2004-12-21 2010-04-08 Pfizer Prod Inc Macrólidos
CN101568343A (zh) 2006-06-12 2009-10-28 雷蒙特亚特特拉维夫大学有限公司 用于治疗癌症的方法
BR112015015075A2 (pt) 2012-12-24 2019-01-15 Univ Ramot agentes para tratar doenças genéticas resultantes de mutações sem sentido e métodos para identificar as mesmas.

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Also Published As

Publication number Publication date
AR020016A2 (es) 2002-03-27
AR012764A1 (es) 2000-11-08
AR019788A2 (es) 2002-03-13
AP9801421A0 (en) 1998-12-31
CZ20002456A3 (cs) 2001-09-12
GT199800207A (es) 2000-06-22
WO1999035157A1 (en) 1999-07-15
SK9772000A3 (en) 2002-09-10
ATE377018T1 (de) 2007-11-15
CA2317131A1 (en) 1999-07-15
PL341647A1 (en) 2001-04-23
EA200000600A1 (ru) 2001-02-26
HRP20000444A2 (en) 2001-04-30
DZ2699A1 (fr) 2003-03-29
ZA9811940B (en) 2000-06-30
YU40900A (sh) 2003-01-31
NO20003346D0 (no) 2000-06-27
AP1060A (en) 2002-04-23
HUP0100566A3 (en) 2003-07-28
EP1642901B1 (de) 2007-10-31
AR019789A2 (es) 2002-03-13
UY25331A1 (es) 2000-12-29
IL136721A0 (en) 2001-06-14
TNSN98236A1 (fr) 2005-03-15
BG104640A (en) 2001-09-28
CA2317131C (en) 2004-11-02
AU1501599A (en) 1999-07-26
DE69838651T2 (de) 2008-03-06
CN1285841A (zh) 2001-02-28
KR20010033822A (ko) 2001-04-25
PE20000119A1 (es) 2000-02-17
CO4970773A1 (es) 2000-11-07
HUP0100566A2 (hu) 2001-07-30
ES2294641T3 (es) 2008-04-01
AR019790A2 (es) 2002-03-13
NZ504987A (en) 2002-11-26
EP1044208A1 (de) 2000-10-18
AU759019B2 (en) 2003-04-03
NO20003346L (no) 2000-08-29
JP2002500231A (ja) 2002-01-08
MA26588A1 (fr) 2004-12-20
UY25587A1 (es) 1999-09-27
DE69838651T9 (de) 2008-06-12
WO1999035157B1 (en) 1999-10-14
PA8465901A1 (es) 2000-09-29
EP1642901A1 (de) 2006-04-05
BR9812992A (pt) 2000-10-17
IS5527A (is) 2000-06-09
US6825171B2 (en) 2004-11-30
US20040067897A1 (en) 2004-04-08
OA11440A (en) 2004-04-28

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8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee