DE60134762D1 - Metabotropische glutamatrezeptor-antagonisten - Google Patents
Metabotropische glutamatrezeptor-antagonistenInfo
- Publication number
- DE60134762D1 DE60134762D1 DE60134762T DE60134762T DE60134762D1 DE 60134762 D1 DE60134762 D1 DE 60134762D1 DE 60134762 T DE60134762 T DE 60134762T DE 60134762 T DE60134762 T DE 60134762T DE 60134762 D1 DE60134762 D1 DE 60134762D1
- Authority
- DE
- Germany
- Prior art keywords
- receptor antagonists
- glutamate receptor
- metabotropic glutamate
- metabotropic
- antagonists
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 102000016193 Metabotropic glutamate receptors Human genes 0.000 title 1
- 108010010914 Metabotropic glutamate receptors Proteins 0.000 title 1
- 239000003825 glutamate receptor antagonist Substances 0.000 title 1
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
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- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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EP00203419 | 2000-10-02 | ||
PCT/EP2001/011135 WO2002028837A1 (en) | 2000-10-02 | 2001-09-25 | Metabotropic glutamate receptor antagonists |
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DE60134762T Expired - Lifetime DE60134762D1 (de) | 2000-10-02 | 2001-09-25 | Metabotropische glutamatrezeptor-antagonisten |
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EP (1) | EP1332133B1 (de) |
JP (1) | JP2004510764A (de) |
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JPH0733743A (ja) * | 1993-07-22 | 1995-02-03 | Kyorin Pharmaceut Co Ltd | 2−アリール−4−キノリノール誘導体 |
JPH08295690A (ja) * | 1995-04-26 | 1996-11-12 | Tokuyama Corp | クロメン化合物 |
WO1997044339A1 (en) * | 1996-05-20 | 1997-11-27 | Merck & Co., Inc. | Antagonists of gonadotropin releasing hormone |
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DE69923849T2 (de) * | 1998-08-27 | 2006-01-12 | Pfizer Products Inc., Groton | Quinolin-2-on-derivate verwendbar als antikrebsmittel |
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BR0114253A (pt) * | 2000-10-02 | 2003-07-01 | Janssen Pharmaceutica Nv | Antagonistas de receptor de glutamato metabotrópico |
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2001
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- 2001-09-25 CN CNA018167179A patent/CN1703403A/zh active Pending
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- 2001-09-25 AU AU2001293847A patent/AU2001293847B2/en not_active Ceased
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- 2001-09-25 HU HU0302167A patent/HUP0302167A3/hu unknown
- 2001-09-25 ES ES01974298T patent/ES2309095T3/es not_active Expired - Lifetime
- 2001-09-25 KR KR1020037002014A patent/KR100818965B1/ko not_active IP Right Cessation
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- 2001-09-25 JP JP2002532423A patent/JP2004510764A/ja active Pending
- 2001-09-25 US US10/381,987 patent/US7115630B2/en not_active Expired - Fee Related
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