IL155163A0 - Metabotropic glutamate receptor antagonists - Google Patents
Metabotropic glutamate receptor antagonistsInfo
- Publication number
- IL155163A0 IL155163A0 IL15516301A IL15516301A IL155163A0 IL 155163 A0 IL155163 A0 IL 155163A0 IL 15516301 A IL15516301 A IL 15516301A IL 15516301 A IL15516301 A IL 15516301A IL 155163 A0 IL155163 A0 IL 155163A0
- Authority
- IL
- Israel
- Prior art keywords
- receptor antagonists
- glutamate receptor
- metabotropic glutamate
- metabotropic
- antagonists
- Prior art date
Links
- 102000016193 Metabotropic glutamate receptors Human genes 0.000 title 1
- 108010010914 Metabotropic glutamate receptors Proteins 0.000 title 1
- 239000003825 glutamate receptor antagonist Substances 0.000 title 1
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- C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
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- C07D215/18—Halogen atoms or nitro radicals
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00203419 | 2000-10-02 | ||
| PCT/EP2001/011135 WO2002028837A1 (en) | 2000-10-02 | 2001-09-25 | Metabotropic glutamate receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL155163A0 true IL155163A0 (en) | 2003-10-31 |
Family
ID=8172097
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL15516301A IL155163A0 (en) | 2000-10-02 | 2001-09-25 | Metabotropic glutamate receptor antagonists |
| IL155163A IL155163A (en) | 2000-10-02 | 2003-03-31 | History of quinoline as antagonists of the metabotropic glutamate receptor, the process for their preparation and the pharmaceutical preparations containing them |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL155163A IL155163A (en) | 2000-10-02 | 2003-03-31 | History of quinoline as antagonists of the metabotropic glutamate receptor, the process for their preparation and the pharmaceutical preparations containing them |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US7115630B2 (de) |
| EP (1) | EP1332133B1 (de) |
| JP (1) | JP2004510764A (de) |
| KR (1) | KR100818965B1 (de) |
| CN (1) | CN1703403A (de) |
| AR (1) | AR035065A1 (de) |
| AT (1) | ATE400558T1 (de) |
| AU (2) | AU9384701A (de) |
| BG (1) | BG107672A (de) |
| BR (1) | BR0114253A (de) |
| CA (1) | CA2421782A1 (de) |
| CZ (1) | CZ20031145A3 (de) |
| DE (1) | DE60134762D1 (de) |
| EA (1) | EA007464B1 (de) |
| EE (1) | EE05195B1 (de) |
| ES (1) | ES2309095T3 (de) |
| HR (1) | HRP20030229A2 (de) |
| HU (1) | HUP0302167A3 (de) |
| IL (2) | IL155163A0 (de) |
| MX (1) | MXPA03002907A (de) |
| MY (1) | MY147730A (de) |
| NO (1) | NO325079B1 (de) |
| NZ (1) | NZ524945A (de) |
| PL (1) | PL360677A1 (de) |
| SK (1) | SK5212003A3 (de) |
| UA (1) | UA76726C2 (de) |
| WO (1) | WO2002028837A1 (de) |
| ZA (1) | ZA200302515B (de) |
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| US5475007A (en) * | 1993-05-28 | 1995-12-12 | The Regents Of The University Of California | 1,2,3,4-tetrahydroquinoline-2,3,4-trione-3 or 4-oximes and the use thereof |
| JPH0733743A (ja) * | 1993-07-22 | 1995-02-03 | Kyorin Pharmaceut Co Ltd | 2−アリール−4−キノリノール誘導体 |
| JPH08295690A (ja) * | 1995-04-26 | 1996-11-12 | Tokuyama Corp | クロメン化合物 |
| JP2000511532A (ja) * | 1996-05-20 | 2000-09-05 | メルク エンド カンパニー インコーポレーテッド | 性腺刺激ホルモン放出ホルモンのアンタゴニスト |
| WO1999003822A1 (en) * | 1997-07-18 | 1999-01-28 | Georgetown University | Bicyclic metabotropic glutamate receptor ligands |
| WO1999026927A2 (en) | 1997-11-21 | 1999-06-03 | Nps Pharmaceuticals, Inc. | Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
| ATE289602T1 (de) * | 1998-08-27 | 2005-03-15 | Pfizer Prod Inc | Quinolin-2-on-derivate verwendbar als antikrebsmittel |
| JP2000169450A (ja) * | 1998-09-30 | 2000-06-20 | Kyorin Pharmaceut Co Ltd | 6―アリ―ルキノリンカルボン酸誘導体とその付加塩及びそれらの製造方法 |
| BR9916827A (pt) | 1998-12-23 | 2001-10-16 | Janssen Pharmaceutica Nv | Derivados de quinolina 1,2-anelados |
| DE19859750A1 (de) * | 1998-12-23 | 2000-06-29 | Henkel Kgaa | Mittel zum Färben von keratinhaltigen Fasern |
| KR20010102073A (ko) * | 1999-02-11 | 2001-11-15 | 실버스타인 아써 에이. | 항암제로 유용한 헤테로아릴-치환된 퀴놀린-2-온 유도체 |
| CA2402096A1 (en) * | 2000-03-07 | 2001-09-13 | Takeda Chemical Industries, Ltd. | Vasoactive agents |
| IL155163A0 (en) * | 2000-10-02 | 2003-10-31 | Janssen Pharmaceutica Nv | Metabotropic glutamate receptor antagonists |
-
2001
- 2001-09-25 IL IL15516301A patent/IL155163A0/xx unknown
- 2001-09-25 SK SK521-2003A patent/SK5212003A3/sk unknown
- 2001-09-25 ES ES01974298T patent/ES2309095T3/es not_active Expired - Lifetime
- 2001-09-25 DE DE60134762T patent/DE60134762D1/de not_active Expired - Lifetime
- 2001-09-25 UA UA2003032796A patent/UA76726C2/uk unknown
- 2001-09-25 HR HR20030229A patent/HRP20030229A2/hr not_active Application Discontinuation
- 2001-09-25 EP EP01974298A patent/EP1332133B1/de not_active Expired - Lifetime
- 2001-09-25 BR BR0114253-4A patent/BR0114253A/pt not_active IP Right Cessation
- 2001-09-25 WO PCT/EP2001/011135 patent/WO2002028837A1/en not_active Ceased
- 2001-09-25 US US10/381,987 patent/US7115630B2/en not_active Expired - Fee Related
- 2001-09-25 NZ NZ524945A patent/NZ524945A/en not_active IP Right Cessation
- 2001-09-25 AT AT01974298T patent/ATE400558T1/de not_active IP Right Cessation
- 2001-09-25 KR KR1020037002014A patent/KR100818965B1/ko not_active Expired - Fee Related
- 2001-09-25 AU AU9384701A patent/AU9384701A/xx active Pending
- 2001-09-25 JP JP2002532423A patent/JP2004510764A/ja active Pending
- 2001-09-25 EA EA200300428A patent/EA007464B1/ru not_active IP Right Cessation
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- 2001-09-25 CN CNA018167179A patent/CN1703403A/zh active Pending
- 2001-09-25 CZ CZ20031145A patent/CZ20031145A3/cs unknown
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- 2001-09-25 CA CA002421782A patent/CA2421782A1/en not_active Abandoned
- 2001-09-25 AU AU2001293847A patent/AU2001293847B2/en not_active Ceased
- 2001-09-25 PL PL36067701A patent/PL360677A1/xx not_active IP Right Cessation
- 2001-09-27 MY MYPI20014515A patent/MY147730A/en unknown
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- 2003-03-31 IL IL155163A patent/IL155163A/en not_active IP Right Cessation
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2005
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