DE1951273A1 - 5-Aminomethyloxazolidin-2-on-Derivate,Verfahren zu ihrer Herstellung und ihre Verwendung als Wirkstoffkomponente von Arzneimitteln - Google Patents

5-Aminomethyloxazolidin-2-on-Derivate,Verfahren zu ihrer Herstellung und ihre Verwendung als Wirkstoffkomponente von Arzneimitteln

Info

Publication number
DE1951273A1
DE1951273A1 DE19691951273 DE1951273A DE1951273A1 DE 1951273 A1 DE1951273 A1 DE 1951273A1 DE 19691951273 DE19691951273 DE 19691951273 DE 1951273 A DE1951273 A DE 1951273A DE 1951273 A1 DE1951273 A1 DE 1951273A1
Authority
DE
Germany
Prior art keywords
hcl
group
aminomethyloxazolidin
derivatives
derivatives according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19691951273
Other languages
German (de)
English (en)
Inventor
Colette Douzon
Claude Fauran
Claude Gouret
Guy Raynaud
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Delalande SA filed Critical Delalande SA
Publication of DE1951273A1 publication Critical patent/DE1951273A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE19691951273 1968-10-22 1969-10-10 5-Aminomethyloxazolidin-2-on-Derivate,Verfahren zu ihrer Herstellung und ihre Verwendung als Wirkstoffkomponente von Arzneimitteln Pending DE1951273A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49963/68A GB1222708A (en) 1968-10-22 1968-10-22 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation

Publications (1)

Publication Number Publication Date
DE1951273A1 true DE1951273A1 (de) 1970-05-06

Family

ID=10454141

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19691951273 Pending DE1951273A1 (de) 1968-10-22 1969-10-10 5-Aminomethyloxazolidin-2-on-Derivate,Verfahren zu ihrer Herstellung und ihre Verwendung als Wirkstoffkomponente von Arzneimitteln

Country Status (9)

Country Link
US (1) US3687965A (enExample)
BE (1) BE740092A (enExample)
CH (1) CH498853A (enExample)
DE (1) DE1951273A1 (enExample)
ES (1) ES372342A1 (enExample)
FR (1) FR2021204B1 (enExample)
GB (1) GB1222708A (enExample)
LU (1) LU59620A1 (enExample)
NL (1) NL6915339A (enExample)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2630107A1 (de) * 1975-07-04 1977-01-27 Nippon Chemiphar Co 5-benzyl-2-oxazolidon-derivate und verfahren zu ihrer herstellung
DE2538424A1 (de) * 1975-08-29 1977-03-03 Nordmark Werke Gmbh Neue oxazolidinone, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
EP0300272A1 (de) * 1987-07-18 1989-01-25 MERCK PATENT GmbH Oxazolidinone
EP0623615A1 (de) * 1993-05-01 1994-11-09 MERCK PATENT GmbH Adhäsionsrezeptor -Antagonisten

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4048164A (en) * 1971-06-18 1977-09-13 Delalande S.A. N'-substituted derivatives of 4'-(N-piperazinylmethyl)spiro dibenzocycloheptadi- (or tri-) ene-5,2'-dioxolane(1',3')
LU80081A1 (fr) * 1977-08-26 1979-05-15 Delalande Sa Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique
FR2435473A2 (fr) * 1978-08-17 1980-04-04 Delalande Sa Nouvelles n-aryle oxazolidinones, oxazolidinethiones et pyrrolidinones, leur procede de preparation et leur application en therapeutique
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
FR2458547B2 (fr) * 1978-06-09 1986-05-16 Delalande Sa Nouvelles n-aryle azolones, leur procede de preparation et leur application en therapeutique
FR2500450A1 (fr) * 1981-02-25 1982-08-27 Delalande Sa Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
US4405794A (en) * 1981-12-18 1983-09-20 The Dow Chemical Company Preparation of 2-oxazolidinone and ethyleneurea
US4535792A (en) * 1982-02-17 1985-08-20 Hauni-Werke Korber & Co. Kg. Apparatus for treating perforated webs of tipping paper or the like
US4461773A (en) * 1982-09-15 1984-07-24 E. I. Dupont De Nemours And Company P-Oxooxazolidinylbenzene compounds as antibacterial agents
US4500717A (en) * 1983-03-28 1985-02-19 The Dow Chemical Company Process for preparation of 2-oxazolidinones
US4705799A (en) * 1983-06-07 1987-11-10 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
ES533097A0 (es) * 1983-06-07 1985-08-01 Du Pont Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno.
JPS6183170A (ja) * 1984-09-28 1986-04-26 Nippon Chemiphar Co Ltd 新規な１，３−オキサゾリジン−２−オン誘導体およびその製造法
CA1260948A (en) 1984-12-05 1989-09-26 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents
US4921869A (en) * 1987-10-09 1990-05-01 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5036093A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5039690A (en) * 1987-10-09 1991-08-13 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A (en) * 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4985429A (en) * 1987-10-09 1991-01-15 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
CA1320730C (en) * 1987-10-16 1993-07-27 The Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4942183A (en) * 1987-10-16 1990-07-17 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A (en) * 1987-10-21 1990-12-11 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
ATE95176T1 (de) * 1987-10-21 1993-10-15 Du Pont Merck Pharma Aminomethyl-oxo-oxazolidinyl-ethenylbenzenderivate, nuetzlich als antibakterielles mittel.
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5043443A (en) * 1988-07-29 1991-08-27 Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives
US5883093A (en) * 1995-09-12 1999-03-16 Pharmacia & Upjohn Company Phenyloxazolidinone antimicrobials
CA2318969A1 (en) 1998-01-23 1999-07-29 Mikhail F. Gordeev Oxazolidinone combinatorial libraries, compositions and methods of preparation
DE60212959T2 (de) * 2001-04-07 2007-02-15 Astrazeneca Ab Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika
WO2003035648A1 (en) * 2001-10-25 2003-05-01 Astrazeneca Ab Aryl substituted oxazolidinones with antibacterial activity
TW200302095A (en) * 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
NZ535592A (en) * 2002-02-28 2006-07-28 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1545951A1 (de) * 1965-07-24 1970-05-14 Henkel & Cie Gmbh Verfahren zur Herstellung von substituierten Oxazolidonen

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2630107A1 (de) * 1975-07-04 1977-01-27 Nippon Chemiphar Co 5-benzyl-2-oxazolidon-derivate und verfahren zu ihrer herstellung
DE2538424A1 (de) * 1975-08-29 1977-03-03 Nordmark Werke Gmbh Neue oxazolidinone, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
EP0300272A1 (de) * 1987-07-18 1989-01-25 MERCK PATENT GmbH Oxazolidinone
US4970217A (en) * 1987-07-18 1990-11-13 Merck Patent Gesellschaft Mit Beschrankter Haftung Oxazolidinones
EP0623615A1 (de) * 1993-05-01 1994-11-09 MERCK PATENT GmbH Adhäsionsrezeptor -Antagonisten

Also Published As

Publication number Publication date
FR2021204B1 (enExample) 1973-06-08
FR2021204A1 (enExample) 1970-07-17
US3687965A (en) 1972-08-29
GB1222708A (en) 1971-02-17
NL6915339A (enExample) 1970-04-24
ES372342A1 (es) 1972-01-16
CH498853A (fr) 1970-11-15
LU59620A1 (enExample) 1970-04-10
BE740092A (enExample) 1970-04-10

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Legal Events

Date Code Title Description
SH Request for examination between 03.10.1968 and 22.04.1971