GB1222708A - Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation - Google Patents

Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation

Info

Publication number
GB1222708A
GB1222708A GB49963/68A GB4996368A GB1222708A GB 1222708 A GB1222708 A GB 1222708A GB 49963/68 A GB49963/68 A GB 49963/68A GB 4996368 A GB4996368 A GB 4996368A GB 1222708 A GB1222708 A GB 1222708A
Authority
GB
United Kingdom
Prior art keywords
radical
oxazolidinones
novel
substituted
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB49963/68A
Other languages
English (en)
Inventor
Claude Fauran
Claude Gouret
Guy Raynaud
Colette Douzoh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Delalande SA filed Critical Delalande SA
Priority to GB49963/68A priority Critical patent/GB1222708A/en
Priority to US863354A priority patent/US3687965A/en
Priority to ES372342A priority patent/ES372342A1/es
Priority to CH1528169A priority patent/CH498853A/fr
Priority to FR696934659A priority patent/FR2021204B1/fr
Priority to BE740092D priority patent/BE740092A/xx
Priority to NL6915339A priority patent/NL6915339A/xx
Priority to LU59620D priority patent/LU59620A1/xx
Priority to DE19691951273 priority patent/DE1951273A1/de
Publication of GB1222708A publication Critical patent/GB1222708A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB49963/68A 1968-10-22 1968-10-22 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation Expired GB1222708A (en)

Priority Applications (9)

Application Number Priority Date Filing Date Title
GB49963/68A GB1222708A (en) 1968-10-22 1968-10-22 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
US863354A US3687965A (en) 1968-10-22 1969-10-02 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
ES372342A ES372342A1 (es) 1968-10-22 1969-10-09 Procedimiento de preparacion de derivados de aminometil-5 oxazolidinona-2.
CH1528169A CH498853A (fr) 1968-10-22 1969-10-10 Procédé de préparation de nouveaux dérivés de l'aminométhyl-5 oxazolidinone-2
FR696934659A FR2021204B1 (enExample) 1968-10-22 1969-10-10
BE740092D BE740092A (enExample) 1968-10-22 1969-10-10
NL6915339A NL6915339A (enExample) 1968-10-22 1969-10-10
LU59620D LU59620A1 (enExample) 1968-10-22 1969-10-10
DE19691951273 DE1951273A1 (de) 1968-10-22 1969-10-10 5-Aminomethyloxazolidin-2-on-Derivate,Verfahren zu ihrer Herstellung und ihre Verwendung als Wirkstoffkomponente von Arzneimitteln

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB49963/68A GB1222708A (en) 1968-10-22 1968-10-22 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation

Publications (1)

Publication Number Publication Date
GB1222708A true GB1222708A (en) 1971-02-17

Family

ID=10454141

Family Applications (1)

Application Number Title Priority Date Filing Date
GB49963/68A Expired GB1222708A (en) 1968-10-22 1968-10-22 Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation

Country Status (9)

Country Link
US (1) US3687965A (enExample)
BE (1) BE740092A (enExample)
CH (1) CH498853A (enExample)
DE (1) DE1951273A1 (enExample)
ES (1) ES372342A1 (enExample)
FR (1) FR2021204B1 (enExample)
GB (1) GB1222708A (enExample)
LU (1) LU59620A1 (enExample)
NL (1) NL6915339A (enExample)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2118470A (en) * 1982-02-17 1983-11-02 Hauni Werke Koerber & Co Kg Apparatus for treating perforated webs of tipping paper or the like
US4705799A (en) * 1983-06-07 1987-11-10 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4985429A (en) * 1987-10-09 1991-01-15 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A (en) * 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4048164A (en) * 1971-06-18 1977-09-13 Delalande S.A. N'-substituted derivatives of 4'-(N-piperazinylmethyl)spiro dibenzocycloheptadi- (or tri-) ene-5,2'-dioxolane(1',3')
FR2315925A1 (fr) * 1975-07-04 1977-01-28 Nippon Chemiphar Co Nouveaux derives de 5-benzyle-2-oxazolidone, leur procede de preparation et leur application en therapeutique
DE2538424C2 (de) * 1975-08-29 1983-01-05 Nordmark-Werke Gmbh, 2000 Hamburg 4-substituierte 5-Phenyl-oxazolidon-(2)- Verbindungen und ein diese enthaltendes pharmazeutisches Präparat
LU80081A1 (fr) * 1977-08-26 1979-05-15 Delalande Sa Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique
FR2435473A2 (fr) * 1978-08-17 1980-04-04 Delalande Sa Nouvelles n-aryle oxazolidinones, oxazolidinethiones et pyrrolidinones, leur procede de preparation et leur application en therapeutique
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
FR2458547B2 (fr) * 1978-06-09 1986-05-16 Delalande Sa Nouvelles n-aryle azolones, leur procede de preparation et leur application en therapeutique
FR2500450A1 (fr) * 1981-02-25 1982-08-27 Delalande Sa Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
US4405794A (en) * 1981-12-18 1983-09-20 The Dow Chemical Company Preparation of 2-oxazolidinone and ethyleneurea
US4461773A (en) * 1982-09-15 1984-07-24 E. I. Dupont De Nemours And Company P-Oxooxazolidinylbenzene compounds as antibacterial agents
US4500717A (en) * 1983-03-28 1985-02-19 The Dow Chemical Company Process for preparation of 2-oxazolidinones
ES533097A0 (es) * 1983-06-07 1985-08-01 Du Pont Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno.
JPS6183170A (ja) * 1984-09-28 1986-04-26 Nippon Chemiphar Co Ltd 新規な１，３−オキサゾリジン−２−オン誘導体およびその製造法
CA1260948A (en) 1984-12-05 1989-09-26 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents
DE3723797A1 (de) * 1987-07-18 1989-01-26 Merck Patent Gmbh Oxazolidinone
US4921869A (en) * 1987-10-09 1990-05-01 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5036093A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5039690A (en) * 1987-10-09 1991-08-13 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
CA1320730C (en) * 1987-10-16 1993-07-27 The Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4942183A (en) * 1987-10-16 1990-07-17 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A (en) * 1987-10-21 1990-12-11 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
ATE95176T1 (de) * 1987-10-21 1993-10-15 Du Pont Merck Pharma Aminomethyl-oxo-oxazolidinyl-ethenylbenzenderivate, nuetzlich als antibakterielles mittel.
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5043443A (en) * 1988-07-29 1991-08-27 Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives
ATE181735T1 (de) * 1993-05-01 1999-07-15 Merck Patent Gmbh Substituierte 1-phenyl-oxazolidin-2-on derivate, deren herstellung und deren verwendung als adhäsionsrezeptor-antagonisten
US5883093A (en) * 1995-09-12 1999-03-16 Pharmacia & Upjohn Company Phenyloxazolidinone antimicrobials
CA2318969A1 (en) 1998-01-23 1999-07-29 Mikhail F. Gordeev Oxazolidinone combinatorial libraries, compositions and methods of preparation
DE60212959T2 (de) * 2001-04-07 2007-02-15 Astrazeneca Ab Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika
WO2003035648A1 (en) * 2001-10-25 2003-05-01 Astrazeneca Ab Aryl substituted oxazolidinones with antibacterial activity
TW200302095A (en) * 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
NZ535592A (en) * 2002-02-28 2006-07-28 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1545951A1 (de) * 1965-07-24 1970-05-14 Henkel & Cie Gmbh Verfahren zur Herstellung von substituierten Oxazolidonen

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2118470A (en) * 1982-02-17 1983-11-02 Hauni Werke Koerber & Co Kg Apparatus for treating perforated webs of tipping paper or the like
US4705799A (en) * 1983-06-07 1987-11-10 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4985429A (en) * 1987-10-09 1991-01-15 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A (en) * 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents

Also Published As

Publication number Publication date
FR2021204B1 (enExample) 1973-06-08
FR2021204A1 (enExample) 1970-07-17
DE1951273A1 (de) 1970-05-06
US3687965A (en) 1972-08-29
NL6915339A (enExample) 1970-04-24
ES372342A1 (es) 1972-01-16
CH498853A (fr) 1970-11-15
LU59620A1 (enExample) 1970-04-10
BE740092A (enExample) 1970-04-10

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