DD218362A5 - Verfahren zur herstellung von neuen 1h, 3h-pyrrolo (1,2-c) thiasol-derivaten - Google Patents

Verfahren zur herstellung von neuen 1h, 3h-pyrrolo (1,2-c) thiasol-derivaten Download PDF

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Publication number
DD218362A5
DD218362A5 DD84259351A DD25935184A DD218362A5 DD 218362 A5 DD218362 A5 DD 218362A5 DD 84259351 A DD84259351 A DD 84259351A DD 25935184 A DD25935184 A DD 25935184A DD 218362 A5 DD218362 A5 DD 218362A5
Authority
DD
German Democratic Republic
Prior art keywords
temperature
general formula
radical
product
defined above
Prior art date
Application number
DD84259351A
Other languages
German (de)
English (en)
Inventor
Jean-Louis Fabre
Daniel Farge
Claude James
Daniel Lave
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of DD218362A5 publication Critical patent/DD218362A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
DD84259351A 1983-01-13 1984-01-11 Verfahren zur herstellung von neuen 1h, 3h-pyrrolo (1,2-c) thiasol-derivaten DD218362A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8300453A FR2541280B1 (fr) 1983-01-13 1983-01-13 Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent

Publications (1)

Publication Number Publication Date
DD218362A5 true DD218362A5 (de) 1985-02-06

Family

ID=9284898

Family Applications (1)

Application Number Title Priority Date Filing Date
DD84259351A DD218362A5 (de) 1983-01-13 1984-01-11 Verfahren zur herstellung von neuen 1h, 3h-pyrrolo (1,2-c) thiasol-derivaten

Country Status (28)

Country Link
US (1) US4529728A (ja)
EP (1) EP0115979B1 (ja)
JP (2) JPS59137490A (ja)
KR (1) KR910001482B1 (ja)
AR (1) AR240828A1 (ja)
AT (1) ATE21248T1 (ja)
AU (1) AU562795B2 (ja)
BG (3) BG40145A3 (ja)
CA (1) CA1229603A (ja)
CS (1) CS262417B2 (ja)
DD (1) DD218362A5 (ja)
DE (1) DE3460401D1 (ja)
DK (1) DK13984A (ja)
ES (2) ES8407058A1 (ja)
FI (1) FI76577C (ja)
FR (1) FR2541280B1 (ja)
GR (1) GR81679B (ja)
HU (1) HU193277B (ja)
IE (1) IE56839B1 (ja)
IL (1) IL70664A (ja)
MA (1) MA20001A1 (ja)
MX (5) MX160610A (ja)
NO (1) NO167031C (ja)
NZ (1) NZ206807A (ja)
PL (2) PL140595B1 (ja)
PT (1) PT77952B (ja)
SU (3) SU1245263A3 (ja)
ZA (2) ZA84233B (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2557111B1 (fr) * 1983-12-21 1986-04-11 Rhone Poulenc Sante Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent
FR2601015B1 (fr) * 1986-07-04 1988-08-05 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
CN1030415A (zh) * 1987-02-20 1989-01-18 山之内制药株式会社 饱和的杂环碳酰胺衍生物和它的制备方法
FR2617484B1 (fr) * 1987-07-02 1989-10-20 Rhone Poulenc Sante Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2626004B1 (fr) * 1988-01-20 1991-08-02 Rhone Poulenc Sante Procede de preparation du (pyridyl-3)-3 1h, 3h-pyrrolo (1,2-c) thiazolecarbonitrile-7
FR2644456B1 (fr) * 1989-03-17 1991-07-05 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
JPH05501103A (ja) * 1989-06-26 1993-03-04 ザ・リサーチ・ファウンデーション・オヴ・ステイト・ユニヴァーシティ・オヴ・ニューヨーク ビス―アシルオキシメチル誘導体
FR2678834A1 (fr) * 1991-07-09 1993-01-15 Rhone Poulenc Rorer Sa Nouvelle application therapeutique du pyridylpyrrolothiazole carboxamide.
US5459152A (en) * 1991-07-17 1995-10-17 Abbott Laboratories Platelet activating factor antagonists
HU230518B1 (hu) * 2005-12-20 2016-10-28 Richter Gedeon Nyrt. Bradykinin B1 receptor szelektív antagonista hatással rendelkező új fenatridin származékok, eljárás előállításukra, és az ezeket tartalmazó gyógyszerkészítmények

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3544590A (en) * 1967-04-28 1970-12-01 Exxon Research Engineering Co Cyclic amines and the process for their formation
US3865839A (en) * 1973-03-01 1975-02-11 Hoechst Co American Thiopyranopyrrolylsalicyclic acids and derivatives thereof

Also Published As

Publication number Publication date
ES528873A0 (es) 1984-08-16
US4529728A (en) 1985-07-16
PL251304A1 (en) 1985-09-24
SU1284459A3 (ru) 1987-01-15
ZA84233B (en) 1984-09-26
IE56839B1 (en) 1992-01-01
JPH0547548B2 (ja) 1993-07-19
PT77952B (fr) 1986-07-14
PL245701A1 (en) 1985-05-07
ZA84235B (en) 1984-09-26
KR910001482B1 (ko) 1991-03-09
PL140595B1 (en) 1987-05-30
FI840106A (fi) 1984-07-14
SU1266472A3 (ru) 1986-10-23
FI76577B (fi) 1988-07-29
JPS59137490A (ja) 1984-08-07
ES8502123A1 (es) 1984-12-16
ES531518A0 (es) 1984-12-16
AR240828A2 (es) 1991-02-28
FI76577C (fi) 1988-11-10
HUT34986A (en) 1985-05-28
MX13463A (es) 1993-10-01
MX160610A (es) 1990-03-28
FR2541280B1 (fr) 1985-06-21
NO167031C (no) 1991-09-25
IL70664A0 (en) 1984-04-30
AR240828A1 (es) 1991-02-28
KR840007419A (ko) 1984-12-07
JPH0653748B2 (ja) 1994-07-20
NO167031B (no) 1991-06-17
PL141846B1 (en) 1987-08-31
EP0115979A1 (fr) 1984-08-15
MX13292A (es) 1993-11-01
BG40144A3 (en) 1986-10-15
AU2320284A (en) 1984-07-19
FI840106A0 (fi) 1984-01-12
SU1245263A3 (ru) 1986-07-15
IL70664A (en) 1986-10-31
HU193277B (en) 1987-09-28
ATE21248T1 (de) 1986-08-15
MX13291A (es) 1993-11-01
ES8407058A1 (es) 1984-08-16
EP0115979B1 (fr) 1986-08-06
BG40145A3 (en) 1986-10-15
DK13984A (da) 1984-07-14
CS262417B2 (en) 1989-03-14
BG39639A3 (bg) 1986-07-15
GR81679B (ja) 1984-12-12
DK13984D0 (da) 1984-01-12
MA20001A1 (fr) 1984-10-01
NO840106L (no) 1984-07-16
AU562795B2 (en) 1987-06-18
MX13462A (es) 1993-08-01
DE3460401D1 (en) 1986-09-11
FR2541280A1 (fr) 1984-08-24
CA1229603A (fr) 1987-11-24
PT77952A (fr) 1984-02-01
IE840064L (en) 1984-07-13
NZ206807A (en) 1985-12-13
JPS59134798A (ja) 1984-08-02
CS19784A2 (en) 1988-08-16

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Legal Events

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PJ Ceased due to non-payment of renewal fee (addendum to changes before extension act)