DD148720A5 - Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten - Google Patents

Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten Download PDF

Info

Publication number
DD148720A5
DD148720A5 DD80218769A DD21876980A DD148720A5 DD 148720 A5 DD148720 A5 DD 148720A5 DD 80218769 A DD80218769 A DD 80218769A DD 21876980 A DD21876980 A DD 21876980A DD 148720 A5 DD148720 A5 DD 148720A5
Authority
DD
German Democratic Republic
Prior art keywords
formula
alkyl
phenyl
piperidine
amino
Prior art date
Application number
DD80218769A
Other languages
German (de)
English (en)
Inventor
Simon F Campbell
John C Danilewicz
Colin W Greengrass
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DD148720A5 publication Critical patent/DD148720A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DD80218769A 1979-01-31 1980-01-31 Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten DD148720A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7903398 1979-01-31

Publications (1)

Publication Number Publication Date
DD148720A5 true DD148720A5 (de) 1981-06-10

Family

ID=10502852

Family Applications (1)

Application Number Title Priority Date Filing Date
DD80218769A DD148720A5 (de) 1979-01-31 1980-01-31 Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten

Country Status (28)

Country Link
JP (1) JPS55104278A (ja)
AR (1) AR222208A1 (ja)
AT (1) AT373595B (ja)
BE (1) BE881448A (ja)
CA (1) CA1131636A (ja)
CS (1) CS231970B2 (ja)
DD (1) DD148720A5 (ja)
DE (1) DE3003323A1 (ja)
DK (1) DK540879A (ja)
ES (1) ES488129A0 (ja)
FI (1) FI63936C (ja)
FR (1) FR2447919A1 (ja)
GR (1) GR73626B (ja)
HU (1) HU184233B (ja)
IE (1) IE800178L (ja)
IL (1) IL59252A (ja)
IT (1) IT1149902B (ja)
LU (1) LU82115A1 (ja)
NL (1) NL8000571A (ja)
NO (1) NO800230L (ja)
NZ (1) NZ192744A (ja)
PH (1) PH15436A (ja)
PL (1) PL121890B1 (ja)
PT (1) PT70749A (ja)
SE (1) SE8000699L (ja)
SU (1) SU895291A3 (ja)
YU (1) YU22980A (ja)
ZA (1) ZA80557B (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2483920A1 (fr) * 1980-06-09 1981-12-11 Synthelabo Nouveaux derives de quinazoline, leur procede de preparation et leur application en therapeutique
ES515338A0 (es) * 1981-09-09 1983-11-01 Orion Yhtymae Oy "metodo para la preparacion de piperidinilquinazolidinas substituidas".
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
WO2013070852A2 (en) * 2011-11-08 2013-05-16 Emory University Compounds and compositions used to epigenetically transform cells and methods related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1088068A (en) * 1977-11-16 1980-10-21 Simon F. Campbell Piperidino-quinazolines
GB2021108B (en) * 1978-05-18 1982-07-21 Pfizer Ltd 6,7 - di - 4 - amino - 2 - quinazolines

Also Published As

Publication number Publication date
NL8000571A (nl) 1980-08-04
GR73626B (ja) 1984-03-26
FI63936C (fi) 1983-09-12
AT373595B (de) 1984-02-10
SE8000699L (sv) 1980-08-01
PT70749A (en) 1980-02-01
JPS5728711B2 (ja) 1982-06-18
YU22980A (en) 1983-02-28
IT1149902B (it) 1986-12-10
CS60780A2 (en) 1984-01-16
PL121890B1 (en) 1982-06-30
IE800178L (en) 1980-07-31
AR222208A1 (es) 1981-04-30
FI63936B (fi) 1983-05-31
SU895291A3 (ru) 1981-12-30
CA1131636A (en) 1982-09-14
PL221683A1 (ja) 1980-12-01
NZ192744A (en) 1984-03-30
DE3003323A1 (de) 1980-08-14
PH15436A (en) 1983-01-18
AU5502480A (en) 1980-08-07
ES8101583A1 (es) 1980-12-16
HU184233B (en) 1984-07-30
DK540879A (da) 1980-08-01
IT8019537A0 (it) 1980-01-29
FR2447919A1 (fr) 1980-08-29
IL59252A (en) 1983-11-30
LU82115A1 (fr) 1980-04-23
JPS55104278A (en) 1980-08-09
FR2447919B1 (ja) 1983-02-11
CS231970B2 (en) 1985-01-16
ZA80557B (en) 1981-08-26
IL59252A0 (en) 1980-05-30
FI800252A (fi) 1980-08-01
ATA46980A (de) 1983-06-15
ES488129A0 (es) 1980-12-16
NO800230L (no) 1980-08-01
BE881448A (fr) 1980-07-30

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