DD148720A5 - Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten - Google Patents

Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten Download PDF

Info

Publication number
DD148720A5
DD148720A5 DD80218769A DD21876980A DD148720A5 DD 148720 A5 DD148720 A5 DD 148720A5 DD 80218769 A DD80218769 A DD 80218769A DD 21876980 A DD21876980 A DD 21876980A DD 148720 A5 DD148720 A5 DD 148720A5
Authority
DD
German Democratic Republic
Prior art keywords
formula
alkyl
phenyl
piperidine
amino
Prior art date
Application number
DD80218769A
Other languages
German (de)
English (en)
Inventor
Simon F Campbell
John C Danilewicz
Colin W Greengrass
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DD148720A5 publication Critical patent/DD148720A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DD80218769A 1979-01-31 1980-01-31 Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten DD148720A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7903398 1979-01-31

Publications (1)

Publication Number Publication Date
DD148720A5 true DD148720A5 (de) 1981-06-10

Family

ID=10502852

Family Applications (1)

Application Number Title Priority Date Filing Date
DD80218769A DD148720A5 (de) 1979-01-31 1980-01-31 Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten

Country Status (28)

Country Link
JP (1) JPS55104278A (da)
AR (1) AR222208A1 (da)
AT (1) AT373595B (da)
BE (1) BE881448A (da)
CA (1) CA1131636A (da)
CS (1) CS231970B2 (da)
DD (1) DD148720A5 (da)
DE (1) DE3003323A1 (da)
DK (1) DK540879A (da)
ES (1) ES488129A0 (da)
FI (1) FI63936C (da)
FR (1) FR2447919A1 (da)
GR (1) GR73626B (da)
HU (1) HU184233B (da)
IE (1) IE800178L (da)
IL (1) IL59252A (da)
IT (1) IT1149902B (da)
LU (1) LU82115A1 (da)
NL (1) NL8000571A (da)
NO (1) NO800230L (da)
NZ (1) NZ192744A (da)
PH (1) PH15436A (da)
PL (1) PL121890B1 (da)
PT (1) PT70749A (da)
SE (1) SE8000699L (da)
SU (1) SU895291A3 (da)
YU (1) YU22980A (da)
ZA (1) ZA80557B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2483920A1 (fr) * 1980-06-09 1981-12-11 Synthelabo Nouveaux derives de quinazoline, leur procede de preparation et leur application en therapeutique
ES515338A0 (es) * 1981-09-09 1983-11-01 Orion Yhtymae Oy "metodo para la preparacion de piperidinilquinazolidinas substituidas".
US5280032A (en) * 1989-02-14 1994-01-18 Toyama Chemical Co., Ltd. 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
WO2013070852A2 (en) * 2011-11-08 2013-05-16 Emory University Compounds and compositions used to epigenetically transform cells and methods related thereto

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1088068A (en) * 1977-11-16 1980-10-21 Simon F. Campbell Piperidino-quinazolines
GB2021108B (en) * 1978-05-18 1982-07-21 Pfizer Ltd 6,7 - di - 4 - amino - 2 - quinazolines

Also Published As

Publication number Publication date
NL8000571A (nl) 1980-08-04
GR73626B (da) 1984-03-26
FI63936C (fi) 1983-09-12
AT373595B (de) 1984-02-10
SE8000699L (sv) 1980-08-01
PT70749A (en) 1980-02-01
JPS5728711B2 (da) 1982-06-18
YU22980A (en) 1983-02-28
IT1149902B (it) 1986-12-10
CS60780A2 (en) 1984-01-16
PL121890B1 (en) 1982-06-30
IE800178L (en) 1980-07-31
AR222208A1 (es) 1981-04-30
FI63936B (fi) 1983-05-31
SU895291A3 (ru) 1981-12-30
CA1131636A (en) 1982-09-14
PL221683A1 (da) 1980-12-01
NZ192744A (en) 1984-03-30
DE3003323A1 (de) 1980-08-14
PH15436A (en) 1983-01-18
AU5502480A (en) 1980-08-07
ES8101583A1 (es) 1980-12-16
HU184233B (en) 1984-07-30
DK540879A (da) 1980-08-01
IT8019537A0 (it) 1980-01-29
FR2447919A1 (fr) 1980-08-29
IL59252A (en) 1983-11-30
LU82115A1 (fr) 1980-04-23
JPS55104278A (en) 1980-08-09
FR2447919B1 (da) 1983-02-11
CS231970B2 (en) 1985-01-16
ZA80557B (en) 1981-08-26
IL59252A0 (en) 1980-05-30
FI800252A (fi) 1980-08-01
ATA46980A (de) 1983-06-15
ES488129A0 (es) 1980-12-16
NO800230L (no) 1980-08-01
BE881448A (fr) 1980-07-30

Similar Documents

Publication Publication Date Title
DE60030883T2 (de) Verfahren zur herstellung von alfentanil, sufentanil und remifentanil
DE9101346U1 (de) Neuroprotektive 3-Piperidino-4-hydroxychroman-Derivate
DE2554772A1 (de) Neue 4(1h)-chinolinderivate und verfahren zu ihrer herstellung
DD147537A5 (de) Verfahren zur herstellung von 1,2,4,5-tetra-alkyl-4-aryl-piperidinen
DE1770595B2 (de) 2-(N-Isopropyl aminomethyl)-7-nitro-1,2,3,4-tetrahydrochinolinderivateund deren pharmazeutisch verträgliche Säureadditionssalze
EP0090369B1 (de) Salicylsäurederivate, Verfahren zu ihrer Herstellung, pharmazeutische Präparate auf Basis dieser Verbindungen und ihre Verwendung
DE69102889T2 (de) Chirurgische Nähnadel, Verfahren und Gerät zum Schleifen von chirurgischen Nähnadeln.
DD223452A5 (de) Verfahren zur herstellung von piperidinochinazolinen
DE2919800A1 (de) 4-amino-2-piperidinochinazolin-derivate, verfahren zu ihrer herstellung und solche derivate enthaltende arzneimittel
EP0072960B1 (de) 1,5-Diphenylpyrazolin-3-on-Verbindungen sowie Verfahren und Zwischenprodukte zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DD148720A5 (de) Verfahren zur herstellung von 4-amino-2-piperidinochinazolin-derivaten
DE68902946T2 (de) Heteroarotinoid-derivate, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammenstellungen.
EP0168812A1 (de) 4-Amino-2-phenylchinoline, Verfahren und Zwischenprodukte zu deren Herstellung sowie diese enthaltende Arzneimittel
EP0389425B1 (de) Neue Benzothiopyranylamine
DE1470055A1 (de) Verfahren zur Herstellung von Piperidinderivaten
DE3226921A1 (de) Neue bicyclische verbindungen und verfahren zu ihrer herstellung
DE1949987A1 (de) Neue alpha-Phenylfettsaeureverbindungen
EP0037990A1 (de) Phenyl-chinolizidine, entsprechende pharmazeutische Präparate, die Herstellung der Wirkstoffe sowie entsprechende Ausgangsverbindungen
DE3520104A1 (de) Naphthoxazine, ihre herstellung und verwendung
EP0004260B1 (de) Substituierte Chinolizidin- und Indolizidinmethanolderivate, Verfahren zur Herstellung derselben und Arzneimittel, welche diese enthalten
CH637131A5 (de) 4-amino-2-piperidino-chinazolin-derivate, verfahren zu ihrer herstellung und verwendung solcher derivate in arzneimitteln.
DE1933599A1 (de) Chinolinderivate
DE2160911A1 (de) Verfahren zur Herstellung von Aminoketonen
DE2222931C3 (de) Piperidinoalkylphenthiazine, Verfahren zur Herstellung derselben sowie diese enthaltende pharmazeutische Mittel
DE3115993A1 (de) Neue indol-derivate, verfahren zu ihrer herstellung und pharmazeutische praeparate, die diese verbindungen enthalten