DD148220A5 - Verfahren fuer die herstellung einer neuartigen 6'-n-substituierten-3-n-formylkanamycin-zwischenverbindung - Google Patents

Verfahren fuer die herstellung einer neuartigen 6'-n-substituierten-3-n-formylkanamycin-zwischenverbindung Download PDF

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Publication number
DD148220A5
DD148220A5 DD78216901A DD21690178A DD148220A5 DD 148220 A5 DD148220 A5 DD 148220A5 DD 78216901 A DD78216901 A DD 78216901A DD 21690178 A DD21690178 A DD 21690178A DD 148220 A5 DD148220 A5 DD 148220A5
Authority
DD
German Democratic Republic
Prior art keywords
kanamycin
group
compound
acetyl
preparation
Prior art date
Application number
DD78216901A
Other languages
German (de)
English (en)
Inventor
Michael B Thomas
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DD148220A5 publication Critical patent/DD148220A5/de

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
DD78216901A 1977-08-18 1978-08-18 Verfahren fuer die herstellung einer neuartigen 6'-n-substituierten-3-n-formylkanamycin-zwischenverbindung DD148220A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3480877 1977-08-18

Publications (1)

Publication Number Publication Date
DD148220A5 true DD148220A5 (de) 1981-05-13

Family

ID=10370176

Family Applications (2)

Application Number Title Priority Date Filing Date
DD78207368A DD139582A5 (de) 1977-08-18 1978-08-18 Verfahren zur herstellung von 1-n-alkyl-substituierten kanamycin-derivaten
DD78216901A DD148220A5 (de) 1977-08-18 1978-08-18 Verfahren fuer die herstellung einer neuartigen 6'-n-substituierten-3-n-formylkanamycin-zwischenverbindung

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DD78207368A DD139582A5 (de) 1977-08-18 1978-08-18 Verfahren zur herstellung von 1-n-alkyl-substituierten kanamycin-derivaten

Country Status (24)

Country Link
US (1) US4178437A (fi)
JP (1) JPS5459256A (fi)
AR (1) AR218324A1 (fi)
AT (1) AT360154B (fi)
BE (1) BE869761A (fi)
CA (1) CA1106842A (fi)
CS (1) CS201512B2 (fi)
DD (2) DD139582A5 (fi)
DE (1) DE2835759A1 (fi)
DK (1) DK308878A (fi)
EG (1) EG13472A (fi)
ES (2) ES472657A1 (fi)
FI (1) FI782497A (fi)
FR (1) FR2400523A1 (fi)
GR (1) GR70241B (fi)
IE (1) IE47150B1 (fi)
IT (1) IT1098281B (fi)
LU (1) LU80124A1 (fi)
NL (1) NL7808566A (fi)
NO (1) NO782796L (fi)
PL (2) PL114720B1 (fi)
PT (1) PT68427A (fi)
SE (1) SE7808702L (fi)
SU (1) SU873889A3 (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4493831A (en) * 1982-10-25 1985-01-15 Fujisawa Pharmaceutical Co., Ltd. Aminoglycoside derivatives
US7794713B2 (en) 2004-04-07 2010-09-14 Lpath, Inc. Compositions and methods for the treatment and prevention of hyperproliferative diseases
US7862812B2 (en) 2006-05-31 2011-01-04 Lpath, Inc. Methods for decreasing immune response and treating immune conditions
AU2008326297B2 (en) * 2007-11-21 2012-11-08 Cipla USA, Inc. Antibacterial aminoglycoside analogs
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132757A2 (en) * 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
WO2010132765A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE630462A (fi) * 1962-04-03
JPS5644076B2 (fi) * 1973-07-12 1981-10-16
US4029882A (en) * 1974-03-19 1977-06-14 Schering Corporation Selective acylation of the C-1 amino group of aminoglycoside antibiotics
US4044123A (en) * 1975-05-02 1977-08-23 Schering Corporation 6'-N-alkyl-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols, methods for their use as antibacterial agents and compositions useful therefor
NZ184213A (en) * 1976-06-16 1980-05-27 Pfizer 2-deoxystreptamine aminoglycosides and antibacterial pharmaceutical compositions

Also Published As

Publication number Publication date
GR70241B (fi) 1982-09-01
NO782796L (no) 1979-02-20
ES472657A1 (es) 1979-10-16
NL7808566A (nl) 1979-02-20
CS201512B2 (en) 1980-11-28
AT360154B (de) 1980-12-29
BE869761A (fr) 1979-02-16
IT1098281B (it) 1985-09-07
PT68427A (en) 1978-09-01
PL209082A1 (fi) 1980-01-02
SE7808702L (sv) 1979-02-19
IT7826812A0 (it) 1978-08-17
JPS5459256A (en) 1979-05-12
IE47150B1 (en) 1983-12-28
FR2400523A1 (fr) 1979-03-16
IE781653L (en) 1979-02-18
DD139582A5 (de) 1980-01-09
EG13472A (en) 1981-12-31
LU80124A1 (fr) 1980-04-21
FI782497A (fi) 1979-02-19
ATA590278A (de) 1980-05-15
CA1106842A (en) 1981-08-11
AR218324A1 (es) 1980-05-30
DK308878A (da) 1979-02-19
ES479667A1 (es) 1979-08-01
PL114720B1 (en) 1981-02-28
SU873889A3 (ru) 1981-10-15
PL114954B1 (en) 1981-03-31
DE2835759A1 (de) 1979-03-08
US4178437A (en) 1979-12-11

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