CY2270B1 - Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters - Google Patents

Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters

Info

Publication number
CY2270B1
CY2270B1 CY0200021A CY0200021A CY2270B1 CY 2270 B1 CY2270 B1 CY 2270B1 CY 0200021 A CY0200021 A CY 0200021A CY 0200021 A CY0200021 A CY 0200021A CY 2270 B1 CY2270 B1 CY 2270B1
Authority
CY
Cyprus
Prior art keywords
fatty acid
acid esters
aqueous suspensions
hydroxyrisperidone fatty
hydroxyrisperidone
Prior art date
Application number
CY0200021A
Other languages
English (en)
Inventor
Marc Karel Jozef Francois
Roger Carolus August Embrechts
Herman Karel Borghijs
Johan Monbaliu
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8224016&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2270(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CY2270B1 publication Critical patent/CY2270B1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CY0200021A 1996-05-20 2002-04-25 Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters CY2270B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP96201429 1996-05-20

Publications (1)

Publication Number Publication Date
CY2270B1 true CY2270B1 (en) 2003-07-04

Family

ID=8224016

Family Applications (2)

Application Number Title Priority Date Filing Date
CY0200021A CY2270B1 (en) 1996-05-20 2002-04-25 Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
CY2011011C CY2011011I2 (el) 1996-05-20 2011-08-18 Υδατικα εναιωρηματα εστερων λιπαρων οξεων με 9-υδροξυρισπεριδονη

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY2011011C CY2011011I2 (el) 1996-05-20 2011-08-18 Υδατικα εναιωρηματα εστερων λιπαρων οξεων με 9-υδροξυρισπεριδονη

Country Status (38)

Country Link
US (1) US6077843A (pl)
EP (1) EP0904081B1 (pl)
JP (1) JP3274687B2 (pl)
KR (1) KR100358373B1 (pl)
CN (1) CN1093762C (pl)
AR (1) AR007194A1 (pl)
AT (1) ATE208619T1 (pl)
AU (1) AU715572B2 (pl)
BG (1) BG62684B1 (pl)
BR (1) BR9706824B8 (pl)
CA (1) CA2236691C (pl)
CY (2) CY2270B1 (pl)
CZ (1) CZ291284B6 (pl)
DE (2) DE122011100027I1 (pl)
DK (1) DK0904081T3 (pl)
EA (1) EA000536B1 (pl)
EE (1) EE03594B1 (pl)
ES (1) ES2167745T3 (pl)
FR (1) FR11C0035I2 (pl)
HK (1) HK1017852A1 (pl)
HR (1) HRP970276B1 (pl)
HU (2) HU224025B1 (pl)
ID (1) ID16927A (pl)
IL (1) IL124551A (pl)
LU (1) LU91842I2 (pl)
MX (1) MX9804816A (pl)
MY (1) MY126302A (pl)
NO (2) NO315931B1 (pl)
NZ (1) NZ330369A (pl)
PL (1) PL188309B1 (pl)
PT (1) PT904081E (pl)
SI (1) SI0904081T1 (pl)
SK (1) SK284013B6 (pl)
TR (1) TR199800923T2 (pl)
TW (1) TW487572B (pl)
UA (1) UA61898C2 (pl)
WO (1) WO1997044039A1 (pl)
ZA (1) ZA974331B (pl)

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US8329203B2 (en) * 2004-01-12 2012-12-11 The Trustees Of The University Of Pennsylvania Drug-containing implants and methods of use thereof
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JP2023551009A (ja) 2020-11-30 2023-12-06 ヤンセン ファーマシューティカ エヌ．ベー． 持続放出パリペリドン注射可能製剤に関連する投与レジメン
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Also Published As

Publication number Publication date
NO315931B1 (no) 2003-11-17
CA2236691A1 (en) 1997-11-27
NO2011015I1 (no) 2011-09-19
PL327995A1 (en) 1999-01-04
DE122011100027I1 (de) 2011-11-17
NO981984D0 (no) 1998-04-30
TR199800923T2 (xx) 1999-09-21
DE69708284D1 (de) 2001-12-20
PL188309B1 (pl) 2005-01-31
HRP970276A2 (en) 1998-04-30
CA2236691C (en) 2007-01-02
CN1093762C (zh) 2002-11-06
BG102443A (en) 1999-06-30
WO1997044039A1 (en) 1997-11-27
HUP9901319A3 (en) 1999-11-29
HUP9901319A2 (hu) 1999-08-30
SI0904081T1 (en) 2002-04-30
CY2011011I1 (el) 2016-12-14
AU715572B2 (en) 2000-02-03
NO2011015I2 (no) 2013-03-11
JP2000513718A (ja) 2000-10-17
EE03594B1 (et) 2002-02-15
EP0904081A1 (en) 1999-03-31
MY126302A (en) 2006-09-29
BR9706824B8 (pt) 2015-02-18
CY2011011I2 (el) 2016-12-14
DK0904081T3 (da) 2002-02-25
HU224025B1 (hu) 2005-05-30
AU2955997A (en) 1997-12-09
DE69708284T2 (de) 2002-07-25
LU91842I2 (fr) 2011-09-20
EE9800136A (et) 1998-10-15
ES2167745T3 (es) 2002-05-16
MX9804816A (es) 1998-10-31
IL124551A0 (en) 1998-12-06
EP0904081B1 (en) 2001-11-14
BR9706824A (pt) 1999-03-23
KR19990067603A (ko) 1999-08-25
CZ140198A3 (cs) 1999-04-14
JP3274687B2 (ja) 2002-04-15
SK284013B6 (sk) 2004-08-03
EA199800531A1 (ru) 1998-12-24
HUS1100013I1 (hu) 2017-03-28
NO981984L (no) 1998-11-19
ZA974331B (en) 1998-11-19
US6077843A (en) 2000-06-20
CZ291284B6 (cs) 2003-01-15
SK62098A3 (en) 2000-04-10
UA61898C2 (en) 2003-12-15
HK1017852A1 (en) 1999-12-03
AR007194A1 (es) 1999-10-13
PT904081E (pt) 2002-04-29
EA000536B1 (ru) 1999-10-28
FR11C0035I2 (fr) 2013-08-16
TW487572B (en) 2002-05-21
NZ330369A (en) 2000-04-28
ID16927A (id) 1997-11-20
FR11C0035I1 (pl) 2011-07-10
KR100358373B1 (ko) 2003-02-11
BG62684B1 (bg) 2000-05-31
ATE208619T1 (de) 2001-11-15
IL124551A (en) 2001-08-26
HRP970276B1 (en) 2002-04-30
CN1206347A (zh) 1999-01-27

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