CY1112237T1 - Παραγωγα 5-υδροξυ-βενζοθειαζολης που εχουν ενεργοτητα αγωνιστη βητα-2-αδρενοϋποδοχεα - Google Patents

Παραγωγα 5-υδροξυ-βενζοθειαζολης που εχουν ενεργοτητα αγωνιστη βητα-2-αδρενοϋποδοχεα

Info

Publication number
CY1112237T1
CY1112237T1 CY20111101070T CY111101070T CY1112237T1 CY 1112237 T1 CY1112237 T1 CY 1112237T1 CY 20111101070 T CY20111101070 T CY 20111101070T CY 111101070 T CY111101070 T CY 111101070T CY 1112237 T1 CY1112237 T1 CY 1112237T1
Authority
CY
Cyprus
Prior art keywords
beta
hydroxy
agonist activity
benzothiazole derivative
gonadotropin agonist
Prior art date
Application number
CY20111101070T
Other languages
English (en)
Inventor
Robin Alec Fairhurst
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CY1112237T1 publication Critical patent/CY1112237T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Ενώσεις του τύπου (Ι) υπό ελεύθερη μορφή ή υπό μορφή επιδιαλυτωμένου σωματιδίου, όπου Τ έχει την έννοια όπως αναγράφεται στην προδιαγραφή, είναι χρήσιμες για την θεραπεία παθήσεων που προλαμβάνονται ή κατευνάζονται μέσω της ενεργοποίησης του β2-αδρενοϋποδοχέα. Επίσης, περιγράφονται φαρμακευτικές συνθέσεις που περιέχουν τις ενώσεις και μία διεργασία για την παρασκευή των ενώσεων.
CY20111101070T 2004-11-29 2011-11-07 Παραγωγα 5-υδροξυ-βενζοθειαζολης που εχουν ενεργοτητα αγωνιστη βητα-2-αδρενοϋποδοχεα CY1112237T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0426164.0A GB0426164D0 (en) 2004-11-29 2004-11-29 Organic compounds
EP05821742A EP1819686B1 (en) 2004-11-29 2005-11-28 5-hydroxy-benzothiazole derivatives having beta-2-adrenorecptor agonist activity

Publications (1)

Publication Number Publication Date
CY1112237T1 true CY1112237T1 (el) 2015-12-09

Family

ID=33561510

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20111101070T CY1112237T1 (el) 2004-11-29 2011-11-07 Παραγωγα 5-υδροξυ-βενζοθειαζολης που εχουν ενεργοτητα αγωνιστη βητα-2-αδρενοϋποδοχεα

Country Status (19)

Country Link
US (2) US8076489B2 (el)
EP (2) EP2305659A1 (el)
JP (1) JP4648950B2 (el)
KR (1) KR100891415B1 (el)
CN (1) CN101065370B (el)
AT (1) ATE520676T1 (el)
AU (1) AU2005308909C1 (el)
BR (1) BRPI0517894A (el)
CA (1) CA2586443C (el)
CY (1) CY1112237T1 (el)
DK (1) DK1819686T3 (el)
ES (1) ES2370833T3 (el)
GB (1) GB0426164D0 (el)
MX (1) MX2007006374A (el)
PL (1) PL1819686T3 (el)
PT (1) PT1819686E (el)
RU (1) RU2402540C2 (el)
SI (1) SI1819686T1 (el)
WO (1) WO2006056471A1 (el)

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JO3192B1 (ar) * 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
CN106146428A (zh) * 2012-08-30 2016-11-23 诺华股份有限公司 作为β‑2肾上腺受体激动剂的苯并噻唑酮化合物的盐
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KR20070067733A (ko) 2007-06-28
KR100891415B1 (ko) 2009-04-02
AU2005308909C1 (en) 2014-11-27
AU2005308909A1 (en) 2006-06-01
EP1819686A1 (en) 2007-08-22
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EP1819686B1 (en) 2011-08-17
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ATE520676T1 (de) 2011-09-15
EP2305659A1 (en) 2011-04-06
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RU2007124329A (ru) 2009-01-10
JP4648950B2 (ja) 2011-03-09
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