CU23874B1 - 4-aril-1,4-dihidro-1,6-naftiridinamidas sustituidas y su uso - Google Patents

4-aril-1,4-dihidro-1,6-naftiridinamidas sustituidas y su uso

Info

Publication number
CU23874B1
CU23874B1 CUP2009000148A CU20090148A CU23874B1 CU 23874 B1 CU23874 B1 CU 23874B1 CU P2009000148 A CUP2009000148 A CU P2009000148A CU 20090148 A CU20090148 A CU 20090148A CU 23874 B1 CU23874 B1 CU 23874B1
Authority
CU
Cuba
Prior art keywords
substituted
naftiridinamids
dihidro
aril
diseases
Prior art date
Application number
CUP2009000148A
Other languages
English (en)
Spanish (es)
Other versions
CU20090148A7 (es
Inventor
Lars Bärfacker
Peter Kolkhof
Karl-Heinz Schlemmer
Rolf Grosser
Adam Nitsche
Martina Klein
Klaus Münter
Barbara Albrecht
Elke Hartmann
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39512753&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU23874(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of CU20090148A7 publication Critical patent/CU20090148A7/es
Publication of CU23874B1 publication Critical patent/CU23874B1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/42—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of mineralocorticosteroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Neurosurgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pigments, Carbon Blacks, Or Wood Stains (AREA)
CUP2009000148A 2007-02-27 2009-08-14 4-aril-1,4-dihidro-1,6-naftiridinamidas sustituidas y su uso CU23874B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007009494A DE102007009494A1 (de) 2007-02-27 2007-02-27 Substituierte 4-Aryl-1, 4-dihydro-1,6-naphthyridinamide und ihre Verwendung
PCT/EP2008/001257 WO2008104306A2 (de) 2007-02-27 2008-02-19 Substituierte 4-aryl-1,4-dihydro-1,6-naphthyridinamide und ihre verwendung

Publications (2)

Publication Number Publication Date
CU20090148A7 CU20090148A7 (es) 2011-04-26
CU23874B1 true CU23874B1 (es) 2013-04-19

Family

ID=39512753

Family Applications (1)

Application Number Title Priority Date Filing Date
CUP2009000148A CU23874B1 (es) 2007-02-27 2009-08-14 4-aril-1,4-dihidro-1,6-naftiridinamidas sustituidas y su uso

Country Status (46)

Country Link
US (2) US8436180B2 (pt-PT)
EP (1) EP2132206B1 (pt-PT)
JP (2) JP5367586B2 (pt-PT)
KR (1) KR101614164B1 (pt-PT)
CN (1) CN101641352B (pt-PT)
AR (1) AR065463A1 (pt-PT)
AU (1) AU2008221071B2 (pt-PT)
BR (2) BR122020008544B8 (pt-PT)
CA (1) CA2679232C (pt-PT)
CL (1) CL2008000502A1 (pt-PT)
CO (1) CO6220951A2 (pt-PT)
CR (1) CR10976A (pt-PT)
CU (1) CU23874B1 (pt-PT)
CY (2) CY1116455T1 (pt-PT)
DE (1) DE102007009494A1 (pt-PT)
DK (1) DK2132206T3 (pt-PT)
DO (1) DOP2009000205A (pt-PT)
EC (1) ECSP099581A (pt-PT)
ES (1) ES2540803T3 (pt-PT)
FR (1) FR22C1017I2 (pt-PT)
GT (1) GT200900230A (pt-PT)
HK (1) HK1140194A1 (pt-PT)
HN (1) HN2009001597A (pt-PT)
HR (1) HRP20150702T1 (pt-PT)
HU (2) HUE026441T2 (pt-PT)
IL (1) IL200060A (pt-PT)
JO (1) JO3018B1 (pt-PT)
LT (1) LTPA2022512I1 (pt-PT)
MA (1) MA31245B1 (pt-PT)
MX (1) MX2009008701A (pt-PT)
MY (2) MY150748A (pt-PT)
NL (1) NL301192I2 (pt-PT)
NO (1) NO2022013I1 (pt-PT)
NZ (1) NZ579230A (pt-PT)
PA (1) PA8770101A1 (pt-PT)
PE (1) PE20090724A1 (pt-PT)
PL (1) PL2132206T3 (pt-PT)
PT (1) PT2132206E (pt-PT)
SA (1) SA08290071B1 (pt-PT)
SI (1) SI2132206T1 (pt-PT)
TN (1) TN2009000318A1 (pt-PT)
TW (2) TWI474821B (pt-PT)
UA (1) UA102065C2 (pt-PT)
UY (3) UY38953A (pt-PT)
WO (1) WO2008104306A2 (pt-PT)
ZA (1) ZA200905730B (pt-PT)

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DE102017008472A1 (de) 2017-09-08 2018-05-03 Bayer Pharma Aktiengesellschaft Kombination enthaltend PDE5 Inhibitoren und Mineralocorticoid-Rezeptor-Antagonisten
CN109721536B (zh) * 2017-10-27 2020-11-24 广东东阳光药业有限公司 苯基取代的稠合三环类化合物及其用途
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CN110917195A (zh) * 2018-08-20 2020-03-27 山西惠尔健生物科技有限公司 肌松剂阿库氯铵（Alcuronium chloride）可作为抗心律失常药物
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