CS259516B2 - Method of new heterocyclic compounds production - Google Patents
Method of new heterocyclic compounds production Download PDFInfo
- Publication number
- CS259516B2 CS259516B2 CS84198A CS19884A CS259516B2 CS 259516 B2 CS259516 B2 CS 259516B2 CS 84198 A CS84198 A CS 84198A CS 19884 A CS19884 A CS 19884A CS 259516 B2 CS259516 B2 CS 259516B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- total
- alkyl
- temperature
- integer
- pyridyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/55—Acids; Esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
- C07D279/06—1,3-Thiazines; Hydrogenated 1,3-thiazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hematology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
- Silicon Polymers (AREA)
- Polyoxymethylene Polymers And Polymers With Carbon-To-Carbon Bonds (AREA)
- Earth Drilling (AREA)
- Materials For Medical Uses (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Peptides Or Proteins (AREA)
- Instructional Devices (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS872469A CS259548B2 (cs) | 1983-01-13 | 1987-04-06 | Způsob výroby nových heierocyklických sloučenin |
| CS872470A CS259549B2 (cs) | 1983-01-13 | 1987-04-06 | Způsob výroby nových heterocyklických sloučenin |
| CS872471A CS259550B2 (cs) | 1984-01-10 | 1987-04-06 | Způsob výroby nové heterocyklické sloučeniny |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8300454A FR2539417A1 (fr) | 1983-01-13 | 1983-01-13 | Nouveaux pyrrolo-1, 2 heterocycles, leur preparation et les medicaments qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CS19884A2 CS19884A2 (en) | 1988-03-15 |
| CS259516B2 true CS259516B2 (en) | 1988-10-14 |
Family
ID=9284899
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS84198A CS259516B2 (en) | 1983-01-13 | 1984-01-10 | Method of new heterocyclic compounds production |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US4546100A (no) |
| EP (1) | EP0118321B1 (no) |
| JP (1) | JPS59134797A (no) |
| KR (1) | KR910001284B1 (no) |
| AT (1) | ATE24321T1 (no) |
| AU (1) | AU562832B2 (no) |
| BG (4) | BG40146A3 (no) |
| CA (1) | CA1222514A (no) |
| CS (1) | CS259516B2 (no) |
| DD (1) | DD216022A5 (no) |
| DE (1) | DE3461713D1 (no) |
| DK (1) | DK13884A (no) |
| ES (3) | ES8502122A1 (no) |
| FI (1) | FI76578C (no) |
| FR (1) | FR2539417A1 (no) |
| GR (1) | GR81680B (no) |
| HU (1) | HU194224B (no) |
| IE (1) | IE56838B1 (no) |
| IL (1) | IL70663A (no) |
| MA (1) | MA20002A1 (no) |
| NO (1) | NO167032C (no) |
| NZ (1) | NZ206809A (no) |
| PL (4) | PL144351B1 (no) |
| PT (1) | PT77951B (no) |
| SU (6) | SU1297730A3 (no) |
| ZA (1) | ZA84234B (no) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2557111B1 (fr) * | 1983-12-21 | 1986-04-11 | Rhone Poulenc Sante | Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent |
| GB8903592D0 (en) * | 1989-02-16 | 1989-04-05 | Boots Co Plc | Therapeutic agents |
| DE3915450A1 (de) * | 1989-05-11 | 1990-11-15 | Gerd Prof Dr Dannhardt | Substituierte pyrrolverbindungen und deren anwendung in der pharmazie |
| US5260451A (en) * | 1989-05-11 | 1993-11-09 | Merckle Gmbh | Substituted pyrrole compounds and use thereof in pharmaceutical compositions |
| JP3061631B2 (ja) * | 1989-10-11 | 2000-07-10 | 山之内製薬株式会社 | 新規なヘテロ環化合物およびその製造法 |
| DE4419246A1 (de) * | 1994-06-01 | 1995-12-07 | Merckle Gmbh | Heteroarylsubstituierte Pyrrolizinverbindungen und deren Anwendung in der Pharmazie |
| DE4419247A1 (de) * | 1994-06-01 | 1995-12-07 | Merckle Gmbh | Sulfonylierte Pyrrolizincarbonsäureamide und deren Anwendung in der Pharmazie |
| FR2735476B1 (fr) * | 1995-06-14 | 1997-07-18 | Rhone Poulenc Rorer Sa | Nouvelle application de derives du pyrrole |
| DE59908677D1 (de) | 1999-11-23 | 2004-04-01 | Merckle Gmbh | Antiinflammatorische oxo- und hydroxyderivate von pyrrolizinen und deren anwendung in der pharmazie |
| DE10004157A1 (de) | 2000-02-01 | 2001-08-02 | Merckle Gmbh Chem Pharm Fabrik | 4-Pyridyl-und 2,4-Pyrimidinyl-substituierte Pyrrolderivate und ihre Anwendung in der Pharmazie |
| US8424704B2 (en) * | 2004-06-02 | 2013-04-23 | X-Pert Paint Mixing Systems, Inc. | Self-cleaning lid for a paint container fluid pour spout |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1401707A (fr) * | 1963-07-03 | 1965-06-04 | Kodak Pathe | Nouveaux colorants, nouveaux composés intermédiaires servant à les préparer et produits photographiques les contenant |
| BE649903A (no) * | 1963-07-03 | |||
| US3642807A (en) * | 1970-06-18 | 1972-02-15 | Schering Corp | Certain 1-/dilower-alkyl amino-loweralkyl/-2-phenyl indolizines and quaternary salts thereof |
-
1983
- 1983-01-13 FR FR8300454A patent/FR2539417A1/fr active Granted
-
1984
- 1984-01-10 CS CS84198A patent/CS259516B2/cs unknown
- 1984-01-11 IL IL70663A patent/IL70663A/xx unknown
- 1984-01-11 MA MA20223A patent/MA20002A1/fr unknown
- 1984-01-11 AU AU23201/84A patent/AU562832B2/en not_active Ceased
- 1984-01-11 DD DD84259352A patent/DD216022A5/de unknown
- 1984-01-11 ZA ZA84234A patent/ZA84234B/xx unknown
- 1984-01-11 GR GR73492A patent/GR81680B/el unknown
- 1984-01-11 NZ NZ206809A patent/NZ206809A/en unknown
- 1984-01-11 US US06/569,907 patent/US4546100A/en not_active Expired - Lifetime
- 1984-01-12 PT PT77951A patent/PT77951B/pt not_active IP Right Cessation
- 1984-01-12 CA CA000445144A patent/CA1222514A/fr not_active Expired
- 1984-01-12 AT AT84400058T patent/ATE24321T1/de not_active IP Right Cessation
- 1984-01-12 FI FI840107A patent/FI76578C/fi not_active IP Right Cessation
- 1984-01-12 DE DE8484400058T patent/DE3461713D1/de not_active Expired
- 1984-01-12 KR KR1019840000094A patent/KR910001284B1/ko not_active IP Right Cessation
- 1984-01-12 SU SU843692003A patent/SU1297730A3/ru active
- 1984-01-12 HU HU8481A patent/HU194224B/hu unknown
- 1984-01-12 BG BG066789A patent/BG40146A3/xx unknown
- 1984-01-12 SU SU843692010A patent/SU1251805A3/ru active
- 1984-01-12 DK DK13884A patent/DK13884A/da not_active Application Discontinuation
- 1984-01-12 IE IE63/84A patent/IE56838B1/en not_active IP Right Cessation
- 1984-01-12 BG BG063860A patent/BG40968A3/xx unknown
- 1984-01-12 BG BG066790A patent/BG40147A3/xx unknown
- 1984-01-12 BG BG066791A patent/BG40148A3/xx unknown
- 1984-01-12 EP EP84400058A patent/EP0118321B1/fr not_active Expired
- 1984-01-12 NO NO840107A patent/NO167032C/no unknown
- 1984-01-13 JP JP59003685A patent/JPS59134797A/ja active Granted
- 1984-01-13 PL PL1984251479A patent/PL144351B1/pl unknown
- 1984-01-13 PL PL1984251478A patent/PL144350B1/pl unknown
- 1984-01-13 ES ES528874A patent/ES8502122A1/es not_active Expired
- 1984-01-13 PL PL1984245702A patent/PL144341B1/pl unknown
- 1984-01-13 PL PL1984245704A patent/PL142322B1/pl unknown
- 1984-03-28 ES ES531062A patent/ES8504823A1/es not_active Expired
- 1984-03-28 ES ES531063A patent/ES8501771A1/es not_active Expired
- 1984-12-07 SU SU843821204A patent/SU1251808A3/ru active
- 1984-12-14 SU SU843822790A patent/SU1277900A3/ru active
- 1984-12-14 SU SU843823253A patent/SU1282818A3/ru active
- 1984-12-14 SU SU843823559A patent/SU1282819A3/ru active
-
1985
- 1985-04-10 US US06/721,773 patent/US4584297A/en not_active Expired - Fee Related
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