CS233736B2 - Processing of derivative of 1,1-dioxid 4-hydroxy-2-methyl-2h-1,2-benzothiazin-3-karboxyl acid - Google Patents

Processing of derivative of 1,1-dioxid 4-hydroxy-2-methyl-2h-1,2-benzothiazin-3-karboxyl acid Download PDF

Info

Publication number
CS233736B2
CS233736B2 CS827096A CS709682A CS233736B2 CS 233736 B2 CS233736 B2 CS 233736B2 CS 827096 A CS827096 A CS 827096A CS 709682 A CS709682 A CS 709682A CS 233736 B2 CS233736 B2 CS 233736B2
Authority
CS
Czechoslovakia
Prior art keywords
methyl
hydroxy
dmso
dmf
reaction
Prior art date
Application number
CS827096A
Other languages
Czech (cs)
English (en)
Other versions
CS709682A2 (en
Inventor
Paul D Weeks
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to CS834592A priority Critical patent/CS233749B2/cs
Publication of CS709682A2 publication Critical patent/CS709682A2/cs
Publication of CS233736B2 publication Critical patent/CS233736B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CS827096A 1981-10-05 1982-10-05 Processing of derivative of 1,1-dioxid 4-hydroxy-2-methyl-2h-1,2-benzothiazin-3-karboxyl acid CS233736B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS834592A CS233749B2 (cs) 1981-10-05 1983-06-22 Způsob výroby 1,1-dioxidů alkyl-4-hydroxy-2-fnethyl-2H-1,2-benzothiazin-3-karboxylótů

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/308,746 US4376204A (en) 1981-10-05 1981-10-05 3-Hydroxy 2-methyl benzisothiazolines as intermediates in production of piroxicam

Publications (2)

Publication Number Publication Date
CS709682A2 CS709682A2 (en) 1984-06-18
CS233736B2 true CS233736B2 (en) 1985-03-14

Family

ID=23195219

Family Applications (1)

Application Number Title Priority Date Filing Date
CS827096A CS233736B2 (en) 1981-10-05 1982-10-05 Processing of derivative of 1,1-dioxid 4-hydroxy-2-methyl-2h-1,2-benzothiazin-3-karboxyl acid

Country Status (6)

Country Link
US (1) US4376204A (ja)
JP (3) JPS5872574A (ja)
CS (1) CS233736B2 (ja)
PL (2) PL135663B1 (ja)
SU (2) SU1192623A3 (ja)
ZA (1) ZA827258B (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4483982A (en) * 1982-09-02 1984-11-20 Pfizer Inc. Processes for preparing piroxicam and intermediates leading thereto
ES2002646A6 (es) * 1987-03-27 1988-09-01 Induspol Sa Procedimiento para la obtencion de 4-hidroxi-2-metil-n-(2-piri-dil)-2h-1,2-benzotiacina-3-carboxamida 1,1-dioxido
US5120334A (en) * 1991-05-23 1992-06-09 Ford Motor Company Air cleaner for internal combustion engine

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987038A (en) * 1975-05-21 1976-10-19 Warner-Lambert Company Process for the preparation of {1-[5-(4-hydroxy-2H-1,2-benzothiazin-3-yl)-1,2,4-oxadiazol-3-yl]methyl}ethanone S,S-dioxide
US4074048A (en) * 1976-05-10 1978-02-14 Warner-Lambert Company Process for the preparation of 4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides
US4213980A (en) * 1978-01-30 1980-07-22 Ciba-Geigy Corporation Azathianaphthalenes
US4289879A (en) * 1980-09-29 1981-09-15 Pfizer Inc. Synthetic method and intermediate for piroxicam
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives

Also Published As

Publication number Publication date
PL135663B1 (en) 1985-11-30
JPS6372685A (ja) 1988-04-02
PL244762A1 (en) 1984-07-16
CS709682A2 (en) 1984-06-18
JPH0316352B2 (ja) 1991-03-05
ZA827258B (en) 1983-08-31
SU1192623A3 (ru) 1985-11-15
JPS5872574A (ja) 1983-04-30
US4376204A (en) 1983-03-08
PL136942B1 (en) 1986-04-30
JPS6372684A (ja) 1988-04-02
JPS6316384B2 (ja) 1988-04-08
PL244763A1 (en) 1984-07-16
JPH0316353B2 (ja) 1991-03-05
SU1240357A3 (ru) 1986-06-23

Similar Documents

Publication Publication Date Title
SU793390A3 (ru) Способ получени производных имидазола, их солей, рацемической смеси диастериоизомеров или антиподов
SU657744A3 (ru) Способ получени производных 3,4-диметил-5-оксо-2,5дигидропиррола
FI72719C (fi) Syntesfoerfarande foer piroxikam samt mellanprodukt.
CA1102341A (en) Isoxazole derivatives, process for their manufacture and agents containing these compounds
FR2589152A1 (fr) Derives pyridine-3-carboxamides et leur application comme inhibiteurs de la croissance des plantes
CS233736B2 (en) Processing of derivative of 1,1-dioxid 4-hydroxy-2-methyl-2h-1,2-benzothiazin-3-karboxyl acid
CA1077934A (en) Process for the preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide and its use as an intermediate
SU715021A3 (ru) Способ получени производных 2,1,3-тиадиазин-4-он-2,2-диоксида
US4090020A (en) Thienothiazine derivatives
US4797482A (en) Process for the preparation of oxazinobenzothiazine 6,6-dioxide derivatives
RU2032679C1 (ru) Производные бензатиазинов
HU197322B (en) Process for producing pyridyl and quinolyl imidazolinones
JPS63152361A (ja) ５‐ピラゾロンの新誘導体、その製造法、除草剤としての使用及びそれを含む組成物
Elgemeie et al. Activated nitriles in heterocyclic synthesis: A novel synthetic route to furyl-and thienyl-substituted pyridine derivatives
US4628109A (en) 2-ketosulfonamides and process for their preparation
US4175085A (en) Thienothiazine derivatives
JPS6034958A (ja) ３，４―ジヒドロ―２―置換―２ｈ―１，２―ベンゾチアジン―カルボン酸　１，１―ジオキサイド誘導体の製造法
KR850001223B1 (ko) 피록시캄 및 그 중간체의 제조방법
US4683306A (en) Process for the preparation of 3,4-dihydro-2-substituted-2H-1,2-thiazine-carboxylic acid 1,1-dioxide derivatives
PL151850B1 (en) Method for manufacturing 6-amine-1,2-dihydro-1-hydroxy-2-amine-4-piperidinepyrimidine
EP0236754A1 (en) Novel process for preparing 4-acetyl isoquinolinone compounds
DE1620249A1 (de) Verfahren zur Herstellung von Pyrimidopyrimidothiazinverbindungen und/oder Thiazinverbindungen
JP2003089691A (ja) ６−（１−フルオロエチル）ピリミジン類及びその製法
Quraishi The synthesis of monomethoxy‐6‐methyl‐7H‐indeno [2, 1‐c] quinolines
JPH05339242A (ja) ５−クロロ−４−ニトロピラゾール誘導体の製造法