CR20120637A - Triazolopiridinas sustituidas - Google Patents
Triazolopiridinas sustituidasInfo
- Publication number
- CR20120637A CR20120637A CR20120637A CR20120637A CR20120637A CR 20120637 A CR20120637 A CR 20120637A CR 20120637 A CR20120637 A CR 20120637A CR 20120637 A CR20120637 A CR 20120637A CR 20120637 A CR20120637 A CR 20120637A
- Authority
- CR
- Costa Rica
- Prior art keywords
- substituted
- triazolopiridins
- general formula
- triazolopyridine compounds
- substituted triazolopyridine
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A—HUMAN NECESSITIES
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- A61K31/275—Nitriles; Isonitriles
- A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
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- A61K31/282—Platinum compounds
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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- A—HUMAN NECESSITIES
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
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- A—HUMAN NECESSITIES
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
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- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
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- C07D—HETEROCYCLIC COMPOUNDS
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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- C07D491/10—Spiro-condensed systems
- C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Abstract
Compuestos de triazolopiridina sustituida de lafórmula general (I)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10166149 | 2010-06-16 | ||
EP11167139 | 2011-05-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR20120637A true CR20120637A (es) | 2013-03-13 |
Family
ID=44259707
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR20120637A CR20120637A (es) | 2010-06-16 | 2012-12-14 | Triazolopiridinas sustituidas |
Country Status (25)
Country | Link |
---|---|
US (1) | US9555022B2 (es) |
EP (1) | EP2582699A1 (es) |
JP (1) | JP5833644B2 (es) |
KR (1) | KR20130116067A (es) |
CN (1) | CN103189373B (es) |
AR (1) | AR081934A1 (es) |
AU (1) | AU2011267143A1 (es) |
BR (1) | BR112012031837A2 (es) |
CA (1) | CA2802629A1 (es) |
CL (1) | CL2012003540A1 (es) |
CO (1) | CO6650348A2 (es) |
CR (1) | CR20120637A (es) |
CU (1) | CU20120171A7 (es) |
DO (1) | DOP2012000312A (es) |
EA (1) | EA201390010A1 (es) |
EC (1) | ECSP12012338A (es) |
MA (1) | MA34308B1 (es) |
MX (1) | MX2012014766A (es) |
NZ (1) | NZ604443A (es) |
PE (1) | PE20130611A1 (es) |
SG (1) | SG186342A1 (es) |
TN (1) | TN2012000595A1 (es) |
TW (1) | TW201204722A (es) |
UY (1) | UY33452A (es) |
WO (1) | WO2011157688A1 (es) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20120274550A1 (en) | 2010-03-24 | 2012-11-01 | Robert Campbell | Gesture mapping for display device |
EA023766B1 (ru) * | 2011-04-21 | 2016-07-29 | Байер Интеллектчуал Проперти Гмбх | Триазолопиридины |
WO2012160029A1 (en) | 2011-05-23 | 2012-11-29 | Bayer Intellectual Property Gmbh | Substituted triazolopyridines |
UA112096C2 (uk) * | 2011-12-12 | 2016-07-25 | Байєр Інтеллектуал Проперті Гмбх | Заміщені триазолопіридини та їх застосування як інгібіторів ttk |
CN102617339A (zh) * | 2012-03-05 | 2012-08-01 | 山西仟源制药股份有限公司 | 3-环丙基甲氧基-4-卤代苯甲酸或其衍生物及应用 |
AU2013289381A1 (en) | 2012-07-10 | 2015-01-22 | Bayer Pharma Aktiengesellschaft | Method for preparing substituted triazolopyridines |
WO2014020041A1 (en) | 2012-08-02 | 2014-02-06 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer |
WO2014020043A1 (en) | 2012-08-02 | 2014-02-06 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer |
EP3007692A1 (en) * | 2013-06-11 | 2016-04-20 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer comprising a mps-1 kinase inhibitor and a mitotic inhibitor |
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- 2011-06-14 BR BR112012031837A patent/BR112012031837A2/pt not_active IP Right Cessation
- 2011-06-14 AU AU2011267143A patent/AU2011267143A1/en not_active Abandoned
- 2011-06-14 JP JP2013514680A patent/JP5833644B2/ja not_active Expired - Fee Related
- 2011-06-14 CN CN201180039503.4A patent/CN103189373B/zh not_active Expired - Fee Related
- 2011-06-14 SG SG2012091906A patent/SG186342A1/en unknown
- 2011-06-14 EP EP11725437.5A patent/EP2582699A1/en not_active Withdrawn
- 2011-06-14 WO PCT/EP2011/059806 patent/WO2011157688A1/en active Application Filing
- 2011-06-14 MA MA35454A patent/MA34308B1/fr unknown
- 2011-06-14 EA EA201390010A patent/EA201390010A1/ru unknown
- 2011-06-14 PE PE2012002421A patent/PE20130611A1/es not_active Application Discontinuation
- 2011-06-14 KR KR1020137001039A patent/KR20130116067A/ko not_active Application Discontinuation
- 2011-06-14 NZ NZ604443A patent/NZ604443A/en not_active IP Right Cessation
- 2011-06-14 CA CA2802629A patent/CA2802629A1/en not_active Abandoned
- 2011-06-14 MX MX2012014766A patent/MX2012014766A/es not_active Application Discontinuation
- 2011-06-14 US US13/704,859 patent/US9555022B2/en not_active Expired - Fee Related
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2012
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TW201204722A (en) | 2012-02-01 |
MA34308B1 (fr) | 2013-06-01 |
TN2012000595A1 (en) | 2014-04-01 |
CN103189373A (zh) | 2013-07-03 |
CL2012003540A1 (es) | 2013-04-01 |
EP2582699A1 (en) | 2013-04-24 |
SG186342A1 (en) | 2013-01-30 |
CO6650348A2 (es) | 2013-04-15 |
JP5833644B2 (ja) | 2015-12-16 |
CU20120171A7 (es) | 2013-05-31 |
AR081934A1 (es) | 2012-10-31 |
CN103189373B (zh) | 2016-04-06 |
US20130156756A1 (en) | 2013-06-20 |
CA2802629A1 (en) | 2011-12-22 |
JP2013532147A (ja) | 2013-08-15 |
EA201390010A1 (ru) | 2013-06-28 |
NZ604443A (en) | 2014-07-25 |
BR112012031837A2 (pt) | 2016-11-08 |
WO2011157688A1 (en) | 2011-12-22 |
AU2011267143A1 (en) | 2013-01-31 |
KR20130116067A (ko) | 2013-10-22 |
US9555022B2 (en) | 2017-01-31 |
MX2012014766A (es) | 2013-01-29 |
UY33452A (es) | 2012-01-31 |
PE20130611A1 (es) | 2013-05-25 |
DOP2012000312A (es) | 2013-04-15 |
ECSP12012338A (es) | 2012-12-28 |
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