CL2012003540A1 - Compuestos derivados de triazolopiridinas sustituidas; metodo de preparacion; compuestos intermediarios; composicion farmaceutica que los comprende; uso del compuesto para la profilaxis o el tratamiento de leucemia, linfomas malignos, tumores de cabeza y cuello, tumores del torax, tumores gastrointestinales, entre otros. - Google Patents

Compuestos derivados de triazolopiridinas sustituidas; metodo de preparacion; compuestos intermediarios; composicion farmaceutica que los comprende; uso del compuesto para la profilaxis o el tratamiento de leucemia, linfomas malignos, tumores de cabeza y cuello, tumores del torax, tumores gastrointestinales, entre otros.

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Publication number
CL2012003540A1
CL2012003540A1 CL2012003540A CL2012003540A CL2012003540A1 CL 2012003540 A1 CL2012003540 A1 CL 2012003540A1 CL 2012003540 A CL2012003540 A CL 2012003540A CL 2012003540 A CL2012003540 A CL 2012003540A CL 2012003540 A1 CL2012003540 A1 CL 2012003540A1
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CL
Chile
Prior art keywords
tumors
compounds
prophylaxis
leukemia
compound
Prior art date
Application number
CL2012003540A
Other languages
English (en)
Inventor
Gerhard Siemeister
Antje Margret Wengner
Volker Schulze
Dirk Kosemund
Hartmut Schirok
Benjamin Bader
Hans Briem
Simon Holton
Marcus Koppitz
Detlef Stockigt
Olaf Prien
Philip Lieneau
Stefan Prechtl
Original Assignee
Bayer Ip Gmbh
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Publication date
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Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of CL2012003540A1 publication Critical patent/CL2012003540A1/es

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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Abstract

Compuestos derivados de triazolopiridinas sustituidas; método de preparación; compuestos intermediarios; composición farmacéutica que los comprende; uso del compuesto para la profilaxis o el tratamiento de leucemia, linfomas malignos, tumores de cabeza y cuello, tumores del tórax, tumores gastrointestinales, entre otros.
CL2012003540A 2010-06-16 2012-12-14 Compuestos derivados de triazolopiridinas sustituidas; metodo de preparacion; compuestos intermediarios; composicion farmaceutica que los comprende; uso del compuesto para la profilaxis o el tratamiento de leucemia, linfomas malignos, tumores de cabeza y cuello, tumores del torax, tumores gastrointestinales, entre otros. CL2012003540A1 (es)

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CO6650348A2 (es) 2013-04-15
MA34308B1 (fr) 2013-06-01
KR20130116067A (ko) 2013-10-22
CR20120637A (es) 2013-03-13
CN103189373B (zh) 2016-04-06
EA201390010A1 (ru) 2013-06-28
DOP2012000312A (es) 2013-04-15
AR081934A1 (es) 2012-10-31
TW201204722A (en) 2012-02-01
PE20130611A1 (es) 2013-05-25
CU20120171A7 (es) 2013-05-31
JP2013532147A (ja) 2013-08-15
SG186342A1 (en) 2013-01-30
EP2582699A1 (en) 2013-04-24
JP5833644B2 (ja) 2015-12-16
UY33452A (es) 2012-01-31
BR112012031837A2 (pt) 2016-11-08
TN2012000595A1 (en) 2014-04-01
NZ604443A (en) 2014-07-25
MX2012014766A (es) 2013-01-29
AU2011267143A1 (en) 2013-01-31
US9555022B2 (en) 2017-01-31
CA2802629A1 (en) 2011-12-22
CN103189373A (zh) 2013-07-03
US20130156756A1 (en) 2013-06-20
ECSP12012338A (es) 2012-12-28
WO2011157688A1 (en) 2011-12-22

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