CR20130539A - Triazolopiridinas - Google Patents
TriazolopiridinasInfo
- Publication number
- CR20130539A CR20130539A CR20130539A CR20130539A CR20130539A CR 20130539 A CR20130539 A CR 20130539A CR 20130539 A CR20130539 A CR 20130539A CR 20130539 A CR20130539 A CR 20130539A CR 20130539 A CR20130539 A CR 20130539A
- Authority
- CR
- Costa Rica
- Prior art keywords
- triazolopiridins
- general formula
- triazolopyridine compounds
- triazolopyridine
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Compuestos de Triazolopiridinas de la fórmula general I.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11163342 | 2011-04-21 | ||
EP11167872 | 2011-05-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR20130539A true CR20130539A (es) | 2013-12-04 |
Family
ID=46124297
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR20130539A CR20130539A (es) | 2011-04-21 | 2013-10-21 | Triazolopiridinas |
Country Status (39)
Country | Link |
---|---|
US (1) | US20140120087A1 (es) |
EP (1) | EP2699575B1 (es) |
JP (1) | JP5989091B2 (es) |
KR (1) | KR20140025470A (es) |
CN (1) | CN103608350B (es) |
AP (1) | AP3491A (es) |
AR (1) | AR086191A1 (es) |
AU (1) | AU2012244859B2 (es) |
CA (1) | CA2833657A1 (es) |
CL (1) | CL2013003044A1 (es) |
CO (1) | CO6801751A2 (es) |
CR (1) | CR20130539A (es) |
CY (1) | CY1116439T1 (es) |
DK (1) | DK2699575T3 (es) |
DO (1) | DOP2013000244A (es) |
EA (1) | EA023766B1 (es) |
EC (1) | ECSP13013011A (es) |
ES (1) | ES2539265T3 (es) |
GT (1) | GT201300254A (es) |
HK (1) | HK1190398A1 (es) |
HR (1) | HRP20150517T1 (es) |
HU (1) | HUE025496T2 (es) |
IL (1) | IL228704A0 (es) |
JO (1) | JO3040B1 (es) |
MA (1) | MA35049B1 (es) |
ME (1) | ME02143B (es) |
MX (1) | MX348783B (es) |
MY (1) | MY164939A (es) |
PE (1) | PE20141351A1 (es) |
PL (1) | PL2699575T3 (es) |
PT (1) | PT2699575E (es) |
RS (1) | RS54044B1 (es) |
SA (1) | SA112330466B1 (es) |
SG (1) | SG194003A1 (es) |
SI (1) | SI2699575T1 (es) |
TW (1) | TWI558703B (es) |
UY (1) | UY34034A (es) |
WO (1) | WO2012143329A1 (es) |
ZA (1) | ZA201308707B (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112013027096A2 (pt) | 2011-04-21 | 2016-12-27 | Gilead Sciences Inc | compostos de benzotiazol e seu uso farmacêutico |
UA112096C2 (uk) * | 2011-12-12 | 2016-07-25 | Байєр Інтеллектуал Проперті Гмбх | Заміщені триазолопіридини та їх застосування як інгібіторів ttk |
WO2013103724A1 (en) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | 2- (tert - butoxy) -2- (7 -methylquinolin- 6 - yl) acetic acid derivatives for treating aids |
WO2013103738A1 (en) | 2012-01-04 | 2013-07-11 | Gilead Sciences, Inc. | Napthalene acetic acid derivatives against hiv infection |
EP2825540B1 (en) | 2012-03-14 | 2016-09-14 | Bayer Intellectual Property GmbH | Substituted imidazopyridazines |
AU2013289381A1 (en) | 2012-07-10 | 2015-01-22 | Bayer Pharma Aktiengesellschaft | Method for preparing substituted triazolopyridines |
WO2014020043A1 (en) | 2012-08-02 | 2014-02-06 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer |
WO2014020041A1 (en) | 2012-08-02 | 2014-02-06 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer |
EP3004092B1 (en) * | 2013-06-07 | 2017-03-22 | Bayer Pharma Aktiengesellschaft | Substituted triazolopyridines |
CN105431435A (zh) * | 2013-06-07 | 2016-03-23 | 拜耳制药股份公司 | 具有作为mps-1抑制剂的活性的取代的三唑并吡啶类 |
EA201501175A1 (ru) * | 2013-06-10 | 2016-10-31 | Байер Фарма Акциенгезельшафт | Новые соединения для лечения злокачественного новообразования |
PE20160156A1 (es) | 2013-06-11 | 2016-04-20 | Bayer Pharma AG | Derivados de prodroga de triazolpiridinas sustituidas |
EP3007692A1 (en) * | 2013-06-11 | 2016-04-20 | Bayer Pharma Aktiengesellschaft | Combinations for the treatment of cancer comprising a mps-1 kinase inhibitor and a mitotic inhibitor |
EP2860177A3 (en) | 2013-09-20 | 2015-06-10 | Bayer Intellectual Property GmbH | Synthesis of functionalized arenes |
JP6993233B2 (ja) | 2015-04-17 | 2022-01-13 | ネザーランズ トランスレーショナル リサーチ センター ビー.ブイ. | Ttk阻害剤化学療法の為の予後バイオマーカー |
CA3054976A1 (en) * | 2017-03-16 | 2018-09-20 | Jiangsu Hengrui Medicine Co., Ltd. | Heteroaryl[4,3-c]pyrimidine-5-amine derivative, preparation method therefor, and medical uses thereof |
EP3956330A4 (en) | 2019-04-18 | 2023-01-18 | The Johns Hopkins University | SUBSTITUTED 2-AMINO-PYRAZOLYL-[1,2,4]TRIAZOLO[1,5A]PYRIDINE DERIVATIVES AND THEIR USE |
JP2022539208A (ja) | 2019-07-03 | 2022-09-07 | スミトモ ファーマ オンコロジー, インコーポレイテッド | チロシンキナーゼ非受容体1(tnk1)阻害剤およびその使用 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5023252A (en) | 1985-12-04 | 1991-06-11 | Conrex Pharmaceutical Corporation | Transdermal and trans-membrane delivery of drugs |
US5011472A (en) | 1988-09-06 | 1991-04-30 | Brown University Research Foundation | Implantable delivery system for biological factors |
WO2006018325A1 (en) | 2004-08-17 | 2006-02-23 | Galderma Research & Development, S.N.C. | Novel biaromatic compounds which activate receptors of ppar type and their use in cosmetic or pharmaceutical compositions |
SG174086A1 (en) * | 2006-08-30 | 2011-09-29 | Cellzome Ltd | Triazole derivatives as kinase inhibitors |
KR20100049073A (ko) | 2007-07-18 | 2010-05-11 | 노파르티스 아게 | 비시클릭 헤테로아릴 화합물 및 키나제 억제제로서의 그의 용도 |
EP2212326A1 (en) | 2007-08-23 | 2010-08-04 | AstraZeneca AB | 2-anilinopurin-8-ones as inhibitors of ttk/mps1 for the treatment of proliferative disorders |
CA2691448A1 (en) * | 2007-08-31 | 2009-03-05 | Dominique Swinnen | Triazolopyridine compounds and their use as ask inhibitors |
GB0719803D0 (en) * | 2007-10-10 | 2007-11-21 | Cancer Rec Tech Ltd | Therapeutic compounds and their use |
UA102828C2 (en) * | 2007-11-27 | 2013-08-27 | Целльзом Лимитед | Amino triazoles as p13k inhibitors |
KR20110116160A (ko) | 2009-02-13 | 2011-10-25 | 포비어 파마수티칼스 | 카이네이스 저해제로서의 〔1,2,4〕트리아졸로〔1,5-a〕피리딘 |
CA2760077A1 (en) | 2009-04-29 | 2010-11-04 | Marcus Koppitz | Substituted imidazoquinoxalines |
WO2011026579A1 (en) | 2009-09-04 | 2011-03-10 | Bayer Schering Pharma Aktiengesellschaft | Substituted aminoquinoxalines as tyrosine threonine kinase inhibitors |
EP2343297A1 (en) * | 2009-11-30 | 2011-07-13 | Bayer Schering Pharma AG | Triazolopyridines |
UY33452A (es) * | 2010-06-16 | 2012-01-31 | Bayer Schering Pharma Ag | Triazolopiridinas sustituidas |
-
2012
- 2012-04-16 EA EA201301181A patent/EA023766B1/ru not_active IP Right Cessation
- 2012-04-16 AU AU2012244859A patent/AU2012244859B2/en not_active Ceased
- 2012-04-16 AP AP2013007182A patent/AP3491A/xx active
- 2012-04-16 MY MYPI2013701964A patent/MY164939A/en unknown
- 2012-04-16 PE PE2013002378A patent/PE20141351A1/es not_active Application Discontinuation
- 2012-04-16 PT PT127217792T patent/PT2699575E/pt unknown
- 2012-04-16 KR KR1020137030546A patent/KR20140025470A/ko not_active Application Discontinuation
- 2012-04-16 PL PL12721779T patent/PL2699575T3/pl unknown
- 2012-04-16 CN CN201280030682.XA patent/CN103608350B/zh not_active Expired - Fee Related
- 2012-04-16 JP JP2014505584A patent/JP5989091B2/ja not_active Expired - Fee Related
- 2012-04-16 MX MX2013012289A patent/MX348783B/es active IP Right Grant
- 2012-04-16 DK DK12721779.2T patent/DK2699575T3/da active
- 2012-04-16 CA CA2833657A patent/CA2833657A1/en not_active Abandoned
- 2012-04-16 ES ES12721779.2T patent/ES2539265T3/es active Active
- 2012-04-16 WO PCT/EP2012/056914 patent/WO2012143329A1/en active Application Filing
- 2012-04-16 RS RS20150345A patent/RS54044B1/en unknown
- 2012-04-16 EP EP12721779.2A patent/EP2699575B1/en active Active
- 2012-04-16 SI SI201230220T patent/SI2699575T1/sl unknown
- 2012-04-16 HU HUE12721779A patent/HUE025496T2/en unknown
- 2012-04-16 SG SG2013073044A patent/SG194003A1/en unknown
- 2012-04-16 US US14/113,017 patent/US20140120087A1/en not_active Abandoned
- 2012-04-16 MA MA36344A patent/MA35049B1/fr unknown
- 2012-04-16 ME MEP-2015-80A patent/ME02143B/me unknown
- 2012-04-18 SA SA112330466A patent/SA112330466B1/ar unknown
- 2012-04-18 JO JOP/2012/0093A patent/JO3040B1/ar active
- 2012-04-20 UY UY0001034034A patent/UY34034A/es not_active Application Discontinuation
- 2012-04-20 AR ARP120101355A patent/AR086191A1/es active Pending
- 2012-04-20 TW TW101114259A patent/TWI558703B/zh not_active IP Right Cessation
-
2013
- 2013-10-03 IL IL228704A patent/IL228704A0/en unknown
- 2013-10-18 GT GT201300254A patent/GT201300254A/es unknown
- 2013-10-21 DO DO2013000244A patent/DOP2013000244A/es unknown
- 2013-10-21 CL CL2013003044A patent/CL2013003044A1/es unknown
- 2013-10-21 CO CO13248763A patent/CO6801751A2/es active IP Right Grant
- 2013-10-21 CR CR20130539A patent/CR20130539A/es unknown
- 2013-11-05 EC ECSP13013011 patent/ECSP13013011A/es unknown
- 2013-11-20 ZA ZA2013/08707A patent/ZA201308707B/en unknown
-
2014
- 2014-04-15 HK HK14103581.3A patent/HK1190398A1/zh not_active IP Right Cessation
-
2015
- 2015-05-14 HR HRP20150517TT patent/HRP20150517T1/hr unknown
- 2015-06-12 CY CY20151100512T patent/CY1116439T1/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CR20130539A (es) | Triazolopiridinas | |
CR20120295A (es) | Triazolopiridinas | |
CR20140468A (es) | Inhibidores de diacilglicerol aciltransferasa 2 | |
UY34365A (es) | Compuestos heterociclicos | |
UY33958A (es) | Inhibidores de la glucosilceramida sintasa | |
CR20120637A (es) | Triazolopiridinas sustituidas | |
UY34145A (es) | Compuestos inhibidores de metaloenzimas | |
UY34156A (es) | Compuestos inhibidores de metaloenzimas | |
UY34146A (es) | Compuestos inhibidores de metaloenzimas | |
UY34177A (es) | Nuevos compuestos inhibidores de la fosfodiesterasa tipo 10a | |
UY34472A (es) | Derivados modificados de 4-fenil-piridina | |
CL2012002979A1 (es) | Derivados de n3-sustituido-n1-sulfonil-5-fluorpirimidinona. | |
UY34523A (es) | Derivados de betulina | |
UY34654A (es) | Inhibidores de la beta-secretasa | |
CR20140229A (es) | Nuevos derivados bicíclicos de dihidroisoquinolin-1-ona | |
UY34445A (es) | Nuevos compuestos inhibidores de la fosfodiesterasa del tipo 10a | |
UY34206A (es) | Anticuerpo monoclonal de interleucina-31 | |
UY34550A (es) | Bencilpirazoles sustituidos | |
UY33930A (es) | Inhibidores novedosos de quinasas | |
UY34817A (es) | Tienopirimidinas | |
UY34027A (es) | Inhibidores sustituidos de acetil-coa carboxilasa. | |
UY34013A (es) | ?compuestos de cromenona con actividad anti-tumoral?. | |
UY34442A (es) | 2-tiopirimidinonas. | |
BR112014003027A2 (pt) | formulação herbicida melhorada | |
UY34329A (es) | Compuestos de triazolopiridina |