CO6592058A2 - Pirrolidinonas heteroaromaticas fusionadas - Google Patents

Pirrolidinonas heteroaromaticas fusionadas

Info

Publication number
CO6592058A2
CO6592058A2 CO12121953A CO12121953A CO6592058A2 CO 6592058 A2 CO6592058 A2 CO 6592058A2 CO 12121953 A CO12121953 A CO 12121953A CO 12121953 A CO12121953 A CO 12121953A CO 6592058 A2 CO6592058 A2 CO 6592058A2
Authority
CO
Colombia
Prior art keywords
diseases
compounds
formula
conditions
fused heteroaromatic
Prior art date
Application number
CO12121953A
Other languages
English (en)
Spanish (es)
Inventor
Yasuyoshi Arikawa
Benjamin Jones
Betty Lam
Zhe Nie
Christopher Smith
Masashi Takahashi
Quing Dong
Victoria Feher
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43618073&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6592058(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of CO6592058A2 publication Critical patent/CO6592058A2/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/33Heterocyclic compounds
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/527Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim spiro-condensed
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
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  • Immunology (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
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  • Ophthalmology & Optometry (AREA)
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CO12121953A 2009-12-23 2012-07-19 Pirrolidinonas heteroaromaticas fusionadas CO6592058A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28996909P 2009-12-23 2009-12-23
US38696410P 2010-09-27 2010-09-27

Publications (1)

Publication Number Publication Date
CO6592058A2 true CO6592058A2 (es) 2013-01-02

Family

ID=43618073

Family Applications (1)

Application Number Title Priority Date Filing Date
CO12121953A CO6592058A2 (es) 2009-12-23 2012-07-19 Pirrolidinonas heteroaromaticas fusionadas

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Country Link
US (7) US8440689B2 (enExample)
EP (4) EP3489236B1 (enExample)
JP (7) JP5658274B2 (enExample)
KR (1) KR101790255B1 (enExample)
CN (1) CN102753548B (enExample)
AR (1) AR081797A1 (enExample)
AU (1) AU2010333804B2 (enExample)
BR (1) BR112012015651B1 (enExample)
CA (1) CA2786950C (enExample)
CL (1) CL2012001745A1 (enExample)
CO (1) CO6592058A2 (enExample)
CR (1) CR20120392A (enExample)
CY (1) CY1116736T1 (enExample)
DK (1) DK2516434T3 (enExample)
DO (1) DOP2012000180A (enExample)
EA (1) EA021568B1 (enExample)
EC (1) ECSP12012057A (enExample)
ES (1) ES2545616T3 (enExample)
GE (1) GEP20156243B (enExample)
HR (1) HRP20150878T1 (enExample)
HU (1) HUE025177T2 (enExample)
IL (1) IL220509A (enExample)
JO (1) JO3108B1 (enExample)
MA (1) MA33909B1 (enExample)
ME (1) ME02186B (enExample)
MX (1) MX2012007402A (enExample)
MY (1) MY159257A (enExample)
NZ (1) NZ601267A (enExample)
PE (1) PE20130188A1 (enExample)
PH (1) PH12012501311A1 (enExample)
PL (1) PL2516434T3 (enExample)
PT (1) PT2516434E (enExample)
RS (1) RS54180B1 (enExample)
SG (1) SG181857A1 (enExample)
SI (1) SI2516434T1 (enExample)
SM (1) SMT201500199B (enExample)
TN (1) TN2012000316A1 (enExample)
TW (1) TWI457339B (enExample)
UA (1) UA107100C2 (enExample)
UY (1) UY33151A (enExample)
WO (1) WO2011079051A1 (enExample)
ZA (1) ZA201205428B (enExample)

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BR112013024901A2 (pt) * 2011-03-28 2017-11-07 Hoffmann La Roche compostos de tiazolopirimidina
EP2723739B1 (en) 2011-06-22 2016-08-24 Takeda Pharmaceutical Company Limited Substituted 6-aza-isoindolin-1-one derivatives
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US9533986B2 (en) 2012-09-27 2017-01-03 Portola Pharmaceuticals, Inc. Bicyclic dihydropyridone kinase inhibitors
CN105102000B (zh) 2012-11-01 2021-10-22 无限药品公司 使用pi3激酶亚型调节剂的癌症疗法
EP2970194A1 (en) 2013-03-15 2016-01-20 Infinity Pharmaceuticals, Inc. Salts and solid forms of isoquinolinones and composition comprising and methods of using the same
SG10201709926VA (en) 2013-05-30 2017-12-28 Infinity Pharmaceuticals Inc Treatment of cancers using pi3 kinase isoform modulators
SG11201600373YA (en) * 2013-07-31 2016-02-26 Gilead Sciences Inc Syk inhibitors
US9751888B2 (en) 2013-10-04 2017-09-05 Infinity Pharmaceuticals, Inc. Heterocyclic compounds and uses thereof
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