EA021568B1 - Конденсированные гетероароматические пирролидиноны как ингибиторы syk - Google Patents

Конденсированные гетероароматические пирролидиноны как ингибиторы syk Download PDF

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EA021568B1
EA021568B1 EA201290555A EA201290555A EA021568B1 EA 021568 B1 EA021568 B1 EA 021568B1 EA 201290555 A EA201290555 A EA 201290555A EA 201290555 A EA201290555 A EA 201290555A EA 021568 B1 EA021568 B1 EA 021568B1
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Eurasian Patent Office
Prior art keywords
pyrrolo
pyridin
fluoro
methyl
ylamino
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EA201290555A
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English (en)
Russian (ru)
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EA201290555A1 (ru
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Ясуёси Арикава
Бенджамин Джоунз
Бетти Лэм
Чжэ Не
Кристофер Смит
Масаси Такахаси
Цин Дун
Виктория Феер
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Такеда Фармасьютикал Компани Лимитед
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Application filed by Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютикал Компани Лимитед
Publication of EA201290555A1 publication Critical patent/EA201290555A1/ru
Publication of EA021568B1 publication Critical patent/EA021568B1/ru

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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EA201290555A 2009-12-23 2010-12-17 Конденсированные гетероароматические пирролидиноны как ингибиторы syk EA021568B1 (ru)

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US28996909P 2009-12-23 2009-12-23
US38696410P 2010-09-27 2010-09-27
PCT/US2010/061146 WO2011079051A1 (en) 2009-12-23 2010-12-17 Fused heteroaromatic pyrrolidinones as syk inhibitors

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EA201290555A1 EA201290555A1 (ru) 2013-01-30
EA021568B1 true EA021568B1 (ru) 2015-07-30

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