CO4650037A1 - Derivados de pirimidina biciclica condensada - Google Patents

Derivados de pirimidina biciclica condensada

Info

Publication number
CO4650037A1
CO4650037A1 CO97068959A CO97068959A CO4650037A1 CO 4650037 A1 CO4650037 A1 CO 4650037A1 CO 97068959 A CO97068959 A CO 97068959A CO 97068959 A CO97068959 A CO 97068959A CO 4650037 A1 CO4650037 A1 CO 4650037A1
Authority
CO
Colombia
Prior art keywords
pirimidine
derivatives
condensed bicyclic
formula
bicyclic
Prior art date
Application number
CO97068959A
Other languages
English (en)
Inventor
Lee Daniel Arnold
Paul Moyer Mikel
Susan Beth Sobolov-Jaynes
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CO4650037A1 publication Critical patent/CO4650037A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Abstract

LA PRESENTE INVENCION SE REFIERE A COMPUESTOS DE FORMULA FIGURA (1) Y A SALES FARMACEUTICAMENTE ACEPTABLES DE LOS MISMOS, EN LA CUAL Z ES UN GRUPO DE FORMULA.
CO97068959A 1996-11-27 1997-11-25 Derivados de pirimidina biciclica condensada CO4650037A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3186296P 1996-11-27 1996-11-27
US4184697P 1997-04-09 1997-04-09

Publications (1)

Publication Number Publication Date
CO4650037A1 true CO4650037A1 (es) 1998-09-03

Family

ID=26707706

Family Applications (1)

Application Number Title Priority Date Filing Date
CO97068959A CO4650037A1 (es) 1996-11-27 1997-11-25 Derivados de pirimidina biciclica condensada

Country Status (24)

Country Link
US (1) US6413971B1 (es)
EP (1) EP0946554A1 (es)
JP (1) JP2000505109A (es)
KR (1) KR20000057228A (es)
CN (1) CN1237177A (es)
AP (1) AP9701146A0 (es)
AR (1) AR010740A1 (es)
AU (1) AU4718997A (es)
BG (1) BG103417A (es)
BR (1) BR9713552A (es)
CA (1) CA2272705C (es)
CO (1) CO4650037A1 (es)
HN (1) HN1997000146A (es)
HR (1) HRP970641A2 (es)
ID (1) ID18958A (es)
IL (1) IL129825A0 (es)
IS (1) IS5041A (es)
MA (1) MA26452A1 (es)
NO (1) NO992524D0 (es)
OA (1) OA11051A (es)
PA (1) PA8442001A1 (es)
PE (1) PE17299A1 (es)
TN (1) TNSN97192A1 (es)
WO (1) WO1998023613A1 (es)

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Also Published As

Publication number Publication date
HN1997000146A (es) 1998-02-26
CA2272705C (en) 2003-03-18
NO992524L (no) 1999-05-26
NO992524D0 (no) 1999-05-26
AU4718997A (en) 1998-06-22
IS5041A (is) 1999-04-30
CN1237177A (zh) 1999-12-01
KR20000057228A (ko) 2000-09-15
WO1998023613A1 (en) 1998-06-04
JP2000505109A (ja) 2000-04-25
ID18958A (id) 1998-05-28
PE17299A1 (es) 1999-02-19
AP9701146A0 (en) 1998-01-31
HRP970641A2 (en) 1998-10-31
US20020045630A1 (en) 2002-04-18
IL129825A0 (en) 2000-02-29
BG103417A (en) 2000-06-30
US6413971B1 (en) 2002-07-02
BR9713552A (pt) 2000-01-25
PA8442001A1 (es) 2000-05-24
CA2272705A1 (en) 1998-06-04
OA11051A (en) 2003-03-07
TNSN97192A1 (fr) 2005-03-15
MA26452A1 (fr) 2004-12-20
EP0946554A1 (en) 1999-10-06
AR010740A1 (es) 2000-07-12

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