CN101613321A - 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物 - Google Patents

抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物 Download PDF

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CN101613321A
CN101613321A CN200910150500A CN200910150500A CN101613321A CN 101613321 A CN101613321 A CN 101613321A CN 200910150500 A CN200910150500 A CN 200910150500A CN 200910150500 A CN200910150500 A CN 200910150500A CN 101613321 A CN101613321 A CN 101613321A
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group
phenyl
aryl
alkylidene group
heteroaryl
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Chinese (zh)
Inventor
阿德南·M·M·米亚里
罗伯特·C·安德鲁
拉梅什·高伯拉斯瓦米
安尼塔·哈里
夸西·阿沃
加桑·卡巴加
郭晓川
苏帕纳·古普塔
大卫·R·琼斯
陈新
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vTv Therapeutics LLC
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Trans Tech Pharma Inc
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Publication of CN101613321A publication Critical patent/CN101613321A/zh
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    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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CN200910150500A 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物 Pending CN101613321A (zh)

Applications Claiming Priority (2)

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US36198302P 2002-03-05 2002-03-05
US60/361,983 2002-03-05

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CNB038052040A Division CN100525763C (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物

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CN101613321A true CN101613321A (zh) 2009-12-30

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CN200910150500A Pending CN101613321A (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物
CNA2009101508570A Pending CN101597262A (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物
CNB038052040A Expired - Fee Related CN100525763C (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物

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CNA2009101508570A Pending CN101597262A (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物
CNB038052040A Expired - Fee Related CN100525763C (zh) 2002-03-05 2003-03-05 抑制配体与高级糖化终产物受体相互作用的单和双环吡咯衍生物

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US (5) US7361678B2 (https=)
EP (2) EP2324830A1 (https=)
JP (2) JP4481011B2 (https=)
CN (3) CN101613321A (https=)
AT (1) ATE529110T1 (https=)
AU (2) AU2007202350B2 (https=)
CA (1) CA2476594C (https=)
DK (1) DK1482931T3 (https=)
ES (1) ES2373875T3 (https=)
WO (1) WO2003075921A2 (https=)

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EP1482931A2 (en) 2004-12-08
AU2009202814B2 (en) 2011-07-14
AU2007202350A1 (en) 2007-06-14
US20100256119A1 (en) 2010-10-07
US7737285B2 (en) 2010-06-15
CN1633290A (zh) 2005-06-29
WO2003075921A2 (en) 2003-09-18
ATE529110T1 (de) 2011-11-15
US20040082542A1 (en) 2004-04-29
WO2003075921A3 (en) 2003-12-04
DK1482931T3 (da) 2011-12-19
AU2003217943A1 (en) 2003-09-22
CN100525763C (zh) 2009-08-12
HK1069549A1 (en) 2005-05-27
JP2009096806A (ja) 2009-05-07
JP2005525378A (ja) 2005-08-25
US7361678B2 (en) 2008-04-22
US20070213347A1 (en) 2007-09-13
US20120088778A1 (en) 2012-04-12
US7714013B2 (en) 2010-05-11
CN101597262A (zh) 2009-12-09
AU2009202814A1 (en) 2009-08-06
CA2476594C (en) 2012-10-09
ES2373875T3 (es) 2012-02-09
AU2007202350B2 (en) 2009-07-30
CA2476594A1 (en) 2003-09-18
EP1482931B1 (en) 2011-10-19

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