CH618180A5 - Process for the preparation of a derivative of the antibiotic XK-62-2. - Google Patents

Process for the preparation of a derivative of the antibiotic XK-62-2. Download PDF

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Publication number
CH618180A5
CH618180A5 CH1657774A CH1657774A CH618180A5 CH 618180 A5 CH618180 A5 CH 618180A5 CH 1657774 A CH1657774 A CH 1657774A CH 1657774 A CH1657774 A CH 1657774A CH 618180 A5 CH618180 A5 CH 618180A5
Authority
CH
Switzerland
Prior art keywords
compound
hydrogen
compounds
choh
formula
Prior art date
Application number
CH1657774A
Other languages
German (de)
English (en)
Inventor
Kunikatsu Shirahata
Shinji Tomioka
Takashi Nara
Hideo Matsushima
Isao Matsubara
Original Assignee
Kyowa Hakko Kogyo Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyowa Hakko Kogyo Kk filed Critical Kyowa Hakko Kogyo Kk
Publication of CH618180A5 publication Critical patent/CH618180A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
CH1657774A 1973-12-12 1974-12-12 Process for the preparation of a derivative of the antibiotic XK-62-2. CH618180A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP13782773A JPS5635193B2 (ja) 1973-12-12 1973-12-12

Publications (1)

Publication Number Publication Date
CH618180A5 true CH618180A5 (en) 1980-07-15

Family

ID=15207762

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1657774A CH618180A5 (en) 1973-12-12 1974-12-12 Process for the preparation of a derivative of the antibiotic XK-62-2.

Country Status (15)

Country Link
JP (1) JPS5635193B2 (ja)
AT (1) AT337894B (ja)
CA (1) CA1030530A (ja)
CH (1) CH618180A5 (ja)
DE (1) DE2458921C3 (ja)
DK (1) DK644174A (ja)
ES (1) ES432862A1 (ja)
FR (1) FR2254565B1 (ja)
GB (1) GB1470329A (ja)
IN (1) IN141068B (ja)
NL (1) NL7416211A (ja)
NO (1) NO139562C (ja)
PH (1) PH15160A (ja)
SE (1) SE417825B (ja)
ZA (1) ZA747907B (ja)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI425947B (zh) 2007-11-21 2014-02-11 Achaogen Inc 抗菌性胺基糖苷類似物
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
WO2010132757A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132765A2 (en) * 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs

Also Published As

Publication number Publication date
DK644174A (ja) 1975-08-25
ATA991874A (de) 1976-11-15
NO139562B (no) 1978-12-27
FR2254565A1 (ja) 1975-07-11
AU7636074A (en) 1976-06-17
ZA747907B (en) 1976-01-28
CA1030530A (en) 1978-05-02
JPS5088050A (ja) 1975-07-15
PH15160A (en) 1982-08-27
NO139562C (no) 1979-04-04
GB1470329A (en) 1977-04-14
DE2458921B2 (de) 1977-08-04
DE2458921A1 (de) 1975-06-26
NO744447L (ja) 1975-07-07
DE2458921C3 (de) 1978-04-06
SE7415609L (ja) 1975-06-13
SE417825B (sv) 1981-04-13
NL7416211A (nl) 1975-06-16
JPS5635193B2 (ja) 1981-08-15
AT337894B (de) 1977-07-25
ES432862A1 (es) 1977-04-01
IN141068B (ja) 1977-01-15
FR2254565B1 (ja) 1979-08-10

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