CA2639910A1 - Thiazole and thiadiazole compounds for inflammation and immune-related uses - Google Patents

Thiazole and thiadiazole compounds for inflammation and immune-related uses Download PDF

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Publication number
CA2639910A1
CA2639910A1 CA002639910A CA2639910A CA2639910A1 CA 2639910 A1 CA2639910 A1 CA 2639910A1 CA 002639910 A CA002639910 A CA 002639910A CA 2639910 A CA2639910 A CA 2639910A CA 2639910 A1 CA2639910 A1 CA 2639910A1
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Canada
Prior art keywords
optionally substituted
compound
phenyl
methyl
thiazol
Prior art date
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Abandoned
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CA002639910A
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English (en)
French (fr)
Inventor
Nha Huu Vo
Shoujun Chen
Qinglin Che
Yu Xie
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Synta Phamaceuticals Corp
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Individual
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Publication of CA2639910A1 publication Critical patent/CA2639910A1/en
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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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US9725452B2 (en) 2013-03-15 2017-08-08 Presidents And Fellows Of Harvard College Substituted indoles and pyrroles as RIP kinase inhibitors

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