BRPI0923126A2 - Compostos inibidores de molécula pequena de necroptose, uso e composição compreendendo os mesmos e método de diminuir necroptose - Google Patents
Compostos inibidores de molécula pequena de necroptose, uso e composição compreendendo os mesmos e método de diminuir necroptose Download PDFInfo
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- BRPI0923126A2 BRPI0923126A2 BRPI0923126-9A BRPI0923126A BRPI0923126A2 BR PI0923126 A2 BRPI0923126 A2 BR PI0923126A2 BR PI0923126 A BRPI0923126 A BR PI0923126A BR PI0923126 A2 BRPI0923126 A2 BR PI0923126A2
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| AR092742A1 (es) | 2012-10-02 | 2015-04-29 | Intermune Inc | Piridinonas antifibroticas |
| TWI638815B (zh) | 2013-02-15 | 2018-10-21 | 英商葛蘭素史克智慧財產發展有限公司 | 作為激酶抑制劑之雜環醯胺類(一) |
| US20160024098A1 (en) * | 2013-03-15 | 2016-01-28 | President And Fellows Of Harvard College | Hybrid necroptosis inhibitors |
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| CN103396376B (zh) * | 2013-07-31 | 2016-08-10 | 杨文茂 | 一种抗菌抗癌活性化合物 |
| CA2927830A1 (en) | 2013-10-23 | 2015-04-30 | Chugai Seiyaku Kabushiki Kaisha | Quinazolinone and isoquinolinone derivative |
| RU2692485C2 (ru) | 2014-04-02 | 2019-06-25 | Интермьюн, Инк. | Противофиброзные пиридиноны |
| EP3229807A4 (en) | 2014-12-11 | 2018-10-17 | President and Fellows of Harvard College | Inhibitors of cellular necrosis and related methods |
| EP3224245B1 (en) | 2014-12-24 | 2018-09-12 | National Institute Of Biological Sciences, Beijing | Necrosis inhibitors |
| KR102606064B1 (ko) | 2014-12-24 | 2023-11-27 | 내셔널 인스티튜트 오브 바이올로지칼 사이언시스, 베이징 | 괴사 억제제 |
| AR103297A1 (es) | 2014-12-30 | 2017-05-03 | Forma Therapeutics Inc | Pirrolo y pirazolopirimidinas como inhibidores de la proteasa 7 específica de ubiquitina |
| MA41291A (fr) | 2014-12-30 | 2017-11-07 | Forma Therapeutics Inc | Dérivés de la pyrrolotriazinone et de l'imidazotriazinone en tant qu'inhibiteurs de la protéase spécifique de l'ubiquitine n° 7 (usp7) pour le traitement d'un cancer |
| JP2018504430A (ja) | 2015-02-05 | 2018-02-15 | フォーマ セラピューティクス,インコーポレイテッド | ユビキチン特異的プロテアーゼ7阻害物質としてのキナゾリノン及びアザキナゾリノン |
| HK1248221A1 (zh) | 2015-02-05 | 2018-10-12 | Forma Therapeutics, Inc. | 异噻唑啉酮类,吡唑并嘧啶酮类和吡咯并嘧啶酮作为泛蛋白特异性蛋白酶7抑制剂 |
| JP2018504431A (ja) | 2015-02-05 | 2018-02-15 | フォーマ セラピューティクス,インコーポレイテッド | ユビキチン特異的プロテアーゼ7阻害物質としてのチエノピリミジノン |
| WO2016133888A1 (en) * | 2015-02-16 | 2016-08-25 | Biota Pharmaceuticals, Inc. | Compounds for treating respiratory syncytial virus infections |
| DE102015212208A1 (de) | 2015-04-24 | 2016-10-27 | Ihp Gmbh-Innovations For High Performance Microelectronics / Leibniz-Institut Für Innovative Mikroelektronik | Hochgeschwindigkeits-Germanium-PIN-Fotodiode |
| TWI730959B (zh) | 2015-05-19 | 2021-06-21 | 英商葛蘭素史克智慧財產發展有限公司 | 作為激酶抑制劑之雜環醯胺 |
| HK1255074A1 (zh) | 2015-07-01 | 2019-08-02 | Crinetics Pharmaceuticals, Inc. | 生长抑素调节剂及其用途 |
| JP6946412B2 (ja) | 2016-07-18 | 2021-10-06 | ヤンセン ファーマシューティカ エヌ.ベー. | タウpet画像化リガンド |
| IL247368A0 (en) | 2016-08-18 | 2016-11-30 | Yeda Res & Dev | Diagnostic and therapeutic uses of exosomes |
| JP2020509009A (ja) | 2017-02-27 | 2020-03-26 | グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドGlaxosmithkline Intellectual Property Development Limited | キナーゼ阻害剤としての複素環式アミド |
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-
2009
- 2009-12-23 CA CA2772760A patent/CA2772760A1/en not_active Abandoned
- 2009-12-23 CN CN201510081043.1A patent/CN104803986A/zh active Pending
- 2009-12-23 US US13/141,545 patent/US20120122889A1/en not_active Abandoned
- 2009-12-23 CN CN2009801569144A patent/CN102316735A/zh active Pending
- 2009-12-23 JP JP2011543689A patent/JP2012513481A/ja active Pending
- 2009-12-23 AU AU2009329879A patent/AU2009329879A1/en not_active Abandoned
- 2009-12-23 EP EP09835866A patent/EP2381775A4/en not_active Withdrawn
- 2009-12-23 WO PCT/US2009/069483 patent/WO2010075561A1/en not_active Ceased
- 2009-12-23 EP EP15001699.6A patent/EP3000468A1/en not_active Withdrawn
- 2009-12-23 BR BRPI0923126-9A patent/BRPI0923126A2/pt not_active IP Right Cessation
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2013
- 2013-09-20 US US14/033,176 patent/US9586880B2/en active Active
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2014
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2016
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- 2016-09-30 HK HK16111463.7A patent/HK1223272A1/en unknown
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2017
- 2017-02-08 US US15/427,699 patent/US20170305824A1/en not_active Abandoned
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2018
- 2018-08-06 US US16/055,898 patent/US20190135718A1/en not_active Abandoned
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| US20120122889A1 (en) | 2012-05-17 |
| EP2381775A4 (en) | 2012-08-15 |
| HK1223272A1 (en) | 2017-07-28 |
| AU2009329879A1 (en) | 2011-08-11 |
| EP2381775A1 (en) | 2011-11-02 |
| US9586880B2 (en) | 2017-03-07 |
| CN104803986A (zh) | 2015-07-29 |
| US20170305824A1 (en) | 2017-10-26 |
| AU2016202262A1 (en) | 2016-05-12 |
| US20140024657A1 (en) | 2014-01-23 |
| US20190135718A1 (en) | 2019-05-09 |
| JP6178777B2 (ja) | 2017-08-09 |
| EP3000468A1 (en) | 2016-03-30 |
| HK1212973A1 (zh) | 2016-06-24 |
| CN102316735A (zh) | 2012-01-11 |
| JP2012513481A (ja) | 2012-06-14 |
| JP2015061853A (ja) | 2015-04-02 |
| CA2772760A1 (en) | 2010-07-01 |
| WO2010075561A1 (en) | 2010-07-01 |
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