BRPI0719174A2 - preparação de pirimidinas ribofuranosil nucleosídeos - Google Patents

preparação de pirimidinas ribofuranosil nucleosídeos

Info

Publication number
BRPI0719174A2
BRPI0719174A2 BRPI0719174A BRPI0719174A BRPI0719174A2 BR PI0719174 A2 BRPI0719174 A2 BR PI0719174A2 BR PI0719174 A BRPI0719174 A BR PI0719174A BR PI0719174 A BRPI0719174 A BR PI0719174A BR PI0719174 A2 BRPI0719174 A2 BR PI0719174A2
Authority
BR
Brazil
Prior art keywords
pyrimidines
preparation
ribofuranosyl nucleoside
ribofuranosyl
nucleoside
Prior art date
Application number
BRPI0719174A
Other languages
English (en)
Portuguese (pt)
Inventor
Ross Bruce
Chun Byoung-Kwon
Zhu Jiang
Vitale Justin
Sarma Keshab
Jin Qingwu
D Axt Steven
Rachakonda Suguna
Original Assignee
Hoffmann La Roche
Pharmasset Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche, Pharmasset Inc filed Critical Hoffmann La Roche
Publication of BRPI0719174A2 publication Critical patent/BRPI0719174A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • C07H5/02—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BRPI0719174A 2006-10-10 2007-10-05 preparação de pirimidinas ribofuranosil nucleosídeos BRPI0719174A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US85096206P 2006-10-10 2006-10-10
PCT/US2007/021548 WO2008045419A1 (en) 2006-10-10 2007-10-05 Preparation of nucleosides ribofuranosyl pyrimidines

Publications (1)

Publication Number Publication Date
BRPI0719174A2 true BRPI0719174A2 (pt) 2017-06-13

Family

ID=39111500

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0719174A BRPI0719174A2 (pt) 2006-10-10 2007-10-05 preparação de pirimidinas ribofuranosil nucleosídeos

Country Status (18)

Country Link
US (2) US8912321B2 (enExample)
EP (1) EP2084174B1 (enExample)
JP (1) JP5252459B2 (enExample)
KR (1) KR101057239B1 (enExample)
CN (1) CN101600725B (enExample)
AU (1) AU2007307057B2 (enExample)
BR (1) BRPI0719174A2 (enExample)
CA (1) CA2666098C (enExample)
DK (1) DK2084174T3 (enExample)
ES (1) ES2429290T3 (enExample)
GT (1) GT200900080A (enExample)
IL (1) IL198086A (enExample)
MX (1) MX2009003795A (enExample)
PL (1) PL2084174T3 (enExample)
PT (1) PT2084174E (enExample)
RU (1) RU2421461C2 (enExample)
SI (1) SI2084174T1 (enExample)
WO (1) WO2008045419A1 (enExample)

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Also Published As

Publication number Publication date
ES2429290T3 (es) 2013-11-14
IL198086A0 (en) 2009-12-24
EP2084174B1 (en) 2013-07-31
HK1133889A1 (en) 2010-04-09
US8912321B2 (en) 2014-12-16
CN101600725B (zh) 2014-11-26
PT2084174E (pt) 2013-10-08
KR101057239B1 (ko) 2011-08-16
GT200900080A (es) 2012-04-10
US20080139802A1 (en) 2008-06-12
MX2009003795A (es) 2009-06-18
SI2084174T1 (sl) 2013-10-30
KR20090060460A (ko) 2009-06-12
JP2010505954A (ja) 2010-02-25
RU2421461C2 (ru) 2011-06-20
IL198086A (en) 2012-03-29
CN101600725A (zh) 2009-12-09
CA2666098A1 (en) 2008-04-17
RU2009117396A (ru) 2010-11-20
AU2007307057B2 (en) 2011-09-15
PL2084174T3 (pl) 2013-12-31
DK2084174T3 (da) 2013-11-04
US20100056770A1 (en) 2010-03-04
AU2007307057A1 (en) 2008-04-17
CA2666098C (en) 2012-09-25
WO2008045419A1 (en) 2008-04-17
EP2084174A1 (en) 2009-08-05
JP5252459B2 (ja) 2013-07-31

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Legal Events

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B25D Requested change of name of applicant approved

Owner name: F. HOFFMANN-LA ROCHE AG (CH) , GILEAD PHARMASSET L

B25G Requested change of headquarter approved

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