BR112014019699B1 - Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende - Google Patents

Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende Download PDF

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BR112014019699B1
BR112014019699B1 BR112014019699-0A BR112014019699A BR112014019699B1 BR 112014019699 B1 BR112014019699 B1 BR 112014019699B1 BR 112014019699 A BR112014019699 A BR 112014019699A BR 112014019699 B1 BR112014019699 B1 BR 112014019699B1
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formula
compound
alkyl
substituted
pharmaceutical composition
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BR112014019699-0A
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Portuguese (pt)
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BR112014019699A8 (pt
BR112014019699A2 (https=
Inventor
Tim Hugo Maria Jonckers
David Craig Mc Gowan
Pierre Jean-Marie Bernard Raboisson
Mourad Daoubi Khamlichi
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Janssen Sciences Ireland Uc
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Publication of BR112014019699A8 publication Critical patent/BR112014019699A8/pt
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112014019699-0A 2012-02-08 2013-02-07 Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende BR112014019699B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12154474 2012-02-08
EP12154474.6 2012-02-08
PCT/EP2013/052372 WO2013117615A1 (en) 2012-02-08 2013-02-07 Piperidino-pyrimidine derivatives for the treatment of viral infections

Publications (3)

Publication Number Publication Date
BR112014019699A2 BR112014019699A2 (https=) 2017-06-20
BR112014019699A8 BR112014019699A8 (pt) 2021-10-19
BR112014019699B1 true BR112014019699B1 (pt) 2021-12-07

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ID=47678822

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Application Number Title Priority Date Filing Date
BR112014019699-0A BR112014019699B1 (pt) 2012-02-08 2013-02-07 Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende

Country Status (22)

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US (2) US9133192B2 (https=)
EP (1) EP2812331B1 (https=)
JP (1) JP6283320B2 (https=)
KR (1) KR102064807B1 (https=)
CN (1) CN104245695B (https=)
AU (1) AU2013218072B2 (https=)
BR (1) BR112014019699B1 (https=)
CA (1) CA2862823C (https=)
CL (1) CL2014002093A1 (https=)
DK (1) DK2812331T3 (https=)
EA (2) EA033907B1 (https=)
ES (1) ES2716811T3 (https=)
IL (1) IL233499B (https=)
IN (1) IN2014MN01736A (https=)
MX (1) MX357296B (https=)
MY (1) MY169159A (https=)
NZ (1) NZ627036A (https=)
PH (1) PH12014501738B1 (https=)
SG (1) SG11201404743TA (https=)
UA (1) UA112668C2 (https=)
WO (1) WO2013117615A1 (https=)
ZA (1) ZA201405820B (https=)

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