BR0116004A - Derivados de 6-o-carbamoil cetolida de eritromicina úteis como antibacterianos - Google Patents

Derivados de 6-o-carbamoil cetolida de eritromicina úteis como antibacterianos

Info

Publication number
BR0116004A
BR0116004A BR0116004-4A BR0116004A BR0116004A BR 0116004 A BR0116004 A BR 0116004A BR 0116004 A BR0116004 A BR 0116004A BR 0116004 A BR0116004 A BR 0116004A
Authority
BR
Brazil
Prior art keywords
antibacterials
erythromycin
carbamoyl
derivatives useful
ketolide derivatives
Prior art date
Application number
BR0116004-4A
Other languages
English (en)
Inventor
Todd C Henniger
Xiaodong C Xu
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of BR0116004A publication Critical patent/BR0116004A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

"DERIVADOS DE 6-O-CARBAMOIL CETOLIDA DE ERITROMICINA úTEIS COMO ANTIBACTERIANOS". Antibacterianos do tipo 6-O-carbamoil cetolida da fórmula: onde R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^, R^ 6^, X, X<39>, Y e Y<39> são como descritos no relatório e onde os substituintes têm os significados indicados no relatório. Estes compostos são úteis como agentes bacterianos.
BR0116004-4A 2000-12-06 2001-12-05 Derivados de 6-o-carbamoil cetolida de eritromicina úteis como antibacterianos BR0116004A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25154700P 2000-12-06 2000-12-06
US09/773,788 US6472372B1 (en) 2000-12-06 2001-02-01 6-O-Carbamoyl ketolide antibacterials
PCT/US2001/047530 WO2002046204A1 (en) 2000-12-06 2001-12-05 6-0-carbamoyl ketolide derivatives of erythromycin useful as antibacterials

Publications (1)

Publication Number Publication Date
BR0116004A true BR0116004A (pt) 2004-06-22

Family

ID=26941686

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0116004-4A BR0116004A (pt) 2000-12-06 2001-12-05 Derivados de 6-o-carbamoil cetolida de eritromicina úteis como antibacterianos

Country Status (14)

Country Link
US (2) US6472372B1 (pt)
EP (1) EP1343798A1 (pt)
JP (1) JP2004515504A (pt)
KR (1) KR20040008115A (pt)
CN (1) CN1310934C (pt)
AU (1) AU2002230708A1 (pt)
BR (1) BR0116004A (pt)
CA (1) CA2431032A1 (pt)
HR (1) HRP20030468A2 (pt)
IL (1) IL156329A0 (pt)
MX (1) MXPA03005028A (pt)
RU (1) RU2003117027A (pt)
WO (1) WO2002046204A1 (pt)
YU (1) YU46303A (pt)

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US11172989B2 (en) 2014-07-02 2021-11-16 Covidien Lp Dynamic 3D lung map view for tool navigation inside the lung
US11253325B2 (en) 2018-02-08 2022-02-22 Covidien Lp System and method for catheter detection in fluoroscopic images and updating displayed position of catheter
US11269173B2 (en) 2019-08-19 2022-03-08 Covidien Lp Systems and methods for displaying medical video images and/or medical 3D models
US11282251B2 (en) 2018-05-02 2022-03-22 Covidien Lp System and method for constructing virtual radial ultrasound images from CT data and performing a surgical navigation procedure using virtual ultrasound images
US11341692B2 (en) 2017-06-29 2022-05-24 Covidien Lp System and method for identifying, marking and navigating to a target using real time two dimensional fluoroscopic data
US11341720B2 (en) 2018-02-08 2022-05-24 Covidien Lp Imaging reconstruction system and method
US11357593B2 (en) 2019-01-10 2022-06-14 Covidien Lp Endoscopic imaging with augmented parallax
US11364004B2 (en) 2018-02-08 2022-06-21 Covidien Lp System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target
US11380060B2 (en) 2020-01-24 2022-07-05 Covidien Lp System and method for linking a segmentation graph to volumetric data
US11529190B2 (en) 2017-01-30 2022-12-20 Covidien Lp Enhanced ablation and visualization techniques for percutaneous surgical procedures
US11547377B2 (en) 2015-08-06 2023-01-10 Covidien Lp System and method for navigating to target and performing procedure on target utilizing fluoroscopic-based local three dimensional volume reconstruction
US11559266B2 (en) 2015-08-06 2023-01-24 Covidien Lp System and method for local three dimensional volume reconstruction using a standard fluoroscope
US11564751B2 (en) 2019-02-01 2023-01-31 Covidien Lp Systems and methods for visualizing navigation of medical devices relative to targets
US11564649B2 (en) 2017-10-10 2023-01-31 Covidien Lp System and method for identifying and marking a target in a fluoroscopic three-dimensional reconstruction
US11617493B2 (en) 2018-12-13 2023-04-04 Covidien Lp Thoracic imaging, distance measuring, surgical awareness, and notification system and method
US11625825B2 (en) 2019-01-30 2023-04-11 Covidien Lp Method for displaying tumor location within endoscopic images
US11627924B2 (en) 2019-09-24 2023-04-18 Covidien Lp Systems and methods for image-guided navigation of percutaneously-inserted devices
US11701492B2 (en) 2020-06-04 2023-07-18 Covidien Lp Active distal tip drive
US11701179B2 (en) 2018-07-26 2023-07-18 Covidien Lp Modeling a collapsed lung using CT data
US11705238B2 (en) 2018-07-26 2023-07-18 Covidien Lp Systems and methods for providing assistance during surgery
US11707241B2 (en) 2015-08-06 2023-07-25 Covidien Lp System and method for local three dimensional volume reconstruction using a standard fluoroscope
US11744643B2 (en) 2019-02-04 2023-09-05 Covidien Lp Systems and methods facilitating pre-operative prediction of post-operative tissue function
US11793402B2 (en) 2018-12-10 2023-10-24 Covidien Lp System and method for generating a three-dimensional model of a surgical site
US11798178B2 (en) 2014-07-02 2023-10-24 Covidien Lp Fluoroscopic pose estimation
US11793579B2 (en) 2017-02-22 2023-10-24 Covidien Lp Integration of multiple data sources for localization and navigation
US11801113B2 (en) 2018-12-13 2023-10-31 Covidien Lp Thoracic imaging, distance measuring, and notification system and method
US11819285B2 (en) 2019-04-05 2023-11-21 Covidien Lp Magnetic interference detection systems and methods
US11847730B2 (en) 2020-01-24 2023-12-19 Covidien Lp Orientation detection in fluoroscopic images
US11864935B2 (en) 2019-09-09 2024-01-09 Covidien Lp Systems and methods for pose estimation of a fluoroscopic imaging device and for three-dimensional imaging of body structures
US11871913B2 (en) 2014-10-31 2024-01-16 Covidien Lp Computed tomography enhanced fluoroscopic system, device, and method of utilizing the same
US11877806B2 (en) 2018-12-06 2024-01-23 Covidien Lp Deformable registration of computer-generated airway models to airway trees
US11918338B2 (en) 2015-09-23 2024-03-05 Coviden Lp Elongated catheter having sensor and an extended working channel
US11922581B2 (en) 2020-05-08 2024-03-05 Coviden Lp Systems and methods of controlling an operating room display using an augmented reality headset
US11925333B2 (en) 2019-02-01 2024-03-12 Covidien Lp System for fluoroscopic tracking of a catheter to update the relative position of a target and the catheter in a 3D model of a luminal network
US11931111B2 (en) 2019-09-09 2024-03-19 Covidien Lp Systems and methods for providing surgical guidance
US11931141B2 (en) 2008-06-06 2024-03-19 Covidien Lp Hybrid registration method
US11944388B2 (en) 2018-09-28 2024-04-02 Covidien Lp Systems and methods for magnetic interference correction
US11950950B2 (en) 2020-07-24 2024-04-09 Covidien Lp Zoom detection and fluoroscope movement detection for target overlay
US11975157B2 (en) 2019-04-12 2024-05-07 Covidien Lp Method of manufacturing an elongated catheter having multiple sensors for three-dimensional location of the catheter
US12008760B2 (en) 2020-07-24 2024-06-11 Covidien Lp Systems and methods for estimating the movement of a target using a universal deformation model for anatomic tissue
US12051156B2 (en) 2022-06-23 2024-07-30 Covidien Lp System and method for linking a segmentation graph to volumetric data

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CN103242239B (zh) * 2013-05-20 2015-09-23 洛阳师范学院 多取代嘧啶基苯甲醇及其制备方法
CN106928294A (zh) * 2017-03-22 2017-07-07 上海启雁实业有限公司 制备酮内酯大环内酯类抗生素的方法
CN112300221B (zh) * 2020-11-11 2022-04-15 艾美科健（中国）生物医药有限公司 一种加米霉素的合成方法

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US11547485B2 (en) 2014-07-02 2023-01-10 Covidien Lp Dynamic 3D lung map view for tool navigation inside the lung
US11529192B2 (en) 2014-07-02 2022-12-20 Covidien Lp Dynamic 3D lung map view for tool navigation inside the lung
US11389247B2 (en) 2014-07-02 2022-07-19 Covidien Lp Methods for navigation of a probe inside a lung
US11607276B2 (en) 2014-07-02 2023-03-21 Covidien Lp Dynamic 3D lung map view for tool navigation inside the lung
US11172989B2 (en) 2014-07-02 2021-11-16 Covidien Lp Dynamic 3D lung map view for tool navigation inside the lung
US11798178B2 (en) 2014-07-02 2023-10-24 Covidien Lp Fluoroscopic pose estimation
US11877804B2 (en) 2014-07-02 2024-01-23 Covidien Lp Methods for navigation of catheters inside lungs
US11871913B2 (en) 2014-10-31 2024-01-16 Covidien Lp Computed tomography enhanced fluoroscopic system, device, and method of utilizing the same
US11992349B2 (en) 2015-08-06 2024-05-28 Covidien Lp System and method for local three dimensional volume reconstruction using a standard fluoroscope
US11707241B2 (en) 2015-08-06 2023-07-25 Covidien Lp System and method for local three dimensional volume reconstruction using a standard fluoroscope
US11547377B2 (en) 2015-08-06 2023-01-10 Covidien Lp System and method for navigating to target and performing procedure on target utilizing fluoroscopic-based local three dimensional volume reconstruction
US11559266B2 (en) 2015-08-06 2023-01-24 Covidien Lp System and method for local three dimensional volume reconstruction using a standard fluoroscope
US11918338B2 (en) 2015-09-23 2024-03-05 Coviden Lp Elongated catheter having sensor and an extended working channel
US11529190B2 (en) 2017-01-30 2022-12-20 Covidien Lp Enhanced ablation and visualization techniques for percutaneous surgical procedures
US11793579B2 (en) 2017-02-22 2023-10-24 Covidien Lp Integration of multiple data sources for localization and navigation
US11341692B2 (en) 2017-06-29 2022-05-24 Covidien Lp System and method for identifying, marking and navigating to a target using real time two dimensional fluoroscopic data
US11564649B2 (en) 2017-10-10 2023-01-31 Covidien Lp System and method for identifying and marking a target in a fluoroscopic three-dimensional reconstruction
US11712213B2 (en) 2018-02-08 2023-08-01 Covidien Lp System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target
US11341720B2 (en) 2018-02-08 2022-05-24 Covidien Lp Imaging reconstruction system and method
US11896414B2 (en) 2018-02-08 2024-02-13 Covidien Lp System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target
US11989830B2 (en) 2018-02-08 2024-05-21 Covidien Lp Imaging reconstruction system and method
US11701184B2 (en) 2018-02-08 2023-07-18 Covidien Lp System and method for catheter detection in fluoroscopic images and updating displayed position of catheter
US11364004B2 (en) 2018-02-08 2022-06-21 Covidien Lp System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target
US11253325B2 (en) 2018-02-08 2022-02-22 Covidien Lp System and method for catheter detection in fluoroscopic images and updating displayed position of catheter
US11282251B2 (en) 2018-05-02 2022-03-22 Covidien Lp System and method for constructing virtual radial ultrasound images from CT data and performing a surgical navigation procedure using virtual ultrasound images
US12004815B2 (en) 2018-07-26 2024-06-11 Covidien Lp Modeling a collapsed lung using CT data
US11705238B2 (en) 2018-07-26 2023-07-18 Covidien Lp Systems and methods for providing assistance during surgery
US11701179B2 (en) 2018-07-26 2023-07-18 Covidien Lp Modeling a collapsed lung using CT data
US11944388B2 (en) 2018-09-28 2024-04-02 Covidien Lp Systems and methods for magnetic interference correction
US11877806B2 (en) 2018-12-06 2024-01-23 Covidien Lp Deformable registration of computer-generated airway models to airway trees
US11793402B2 (en) 2018-12-10 2023-10-24 Covidien Lp System and method for generating a three-dimensional model of a surgical site
US11617493B2 (en) 2018-12-13 2023-04-04 Covidien Lp Thoracic imaging, distance measuring, surgical awareness, and notification system and method
US11801113B2 (en) 2018-12-13 2023-10-31 Covidien Lp Thoracic imaging, distance measuring, and notification system and method
US11357593B2 (en) 2019-01-10 2022-06-14 Covidien Lp Endoscopic imaging with augmented parallax
US11793390B2 (en) 2019-01-10 2023-10-24 Covidien Lp Endoscopic imaging with augmented parallax
US11625825B2 (en) 2019-01-30 2023-04-11 Covidien Lp Method for displaying tumor location within endoscopic images
US11564751B2 (en) 2019-02-01 2023-01-31 Covidien Lp Systems and methods for visualizing navigation of medical devices relative to targets
US11925333B2 (en) 2019-02-01 2024-03-12 Covidien Lp System for fluoroscopic tracking of a catheter to update the relative position of a target and the catheter in a 3D model of a luminal network
US11744643B2 (en) 2019-02-04 2023-09-05 Covidien Lp Systems and methods facilitating pre-operative prediction of post-operative tissue function
US11819285B2 (en) 2019-04-05 2023-11-21 Covidien Lp Magnetic interference detection systems and methods
US11975157B2 (en) 2019-04-12 2024-05-07 Covidien Lp Method of manufacturing an elongated catheter having multiple sensors for three-dimensional location of the catheter
US12016737B2 (en) 2019-08-19 2024-06-25 Covidien Lp Systems and methods for displaying medical video images and/or medical 3D models
US11269173B2 (en) 2019-08-19 2022-03-08 Covidien Lp Systems and methods for displaying medical video images and/or medical 3D models
US11864935B2 (en) 2019-09-09 2024-01-09 Covidien Lp Systems and methods for pose estimation of a fluoroscopic imaging device and for three-dimensional imaging of body structures
US11931111B2 (en) 2019-09-09 2024-03-19 Covidien Lp Systems and methods for providing surgical guidance
US11627924B2 (en) 2019-09-24 2023-04-18 Covidien Lp Systems and methods for image-guided navigation of percutaneously-inserted devices
US11847730B2 (en) 2020-01-24 2023-12-19 Covidien Lp Orientation detection in fluoroscopic images
US11380060B2 (en) 2020-01-24 2022-07-05 Covidien Lp System and method for linking a segmentation graph to volumetric data
US11922581B2 (en) 2020-05-08 2024-03-05 Coviden Lp Systems and methods of controlling an operating room display using an augmented reality headset
US11701492B2 (en) 2020-06-04 2023-07-18 Covidien Lp Active distal tip drive
US11950950B2 (en) 2020-07-24 2024-04-09 Covidien Lp Zoom detection and fluoroscope movement detection for target overlay
US12008760B2 (en) 2020-07-24 2024-06-11 Covidien Lp Systems and methods for estimating the movement of a target using a universal deformation model for anatomic tissue
US12051156B2 (en) 2022-06-23 2024-07-30 Covidien Lp System and method for linking a segmentation graph to volumetric data

Also Published As

Publication number Publication date
US20030013663A1 (en) 2003-01-16
JP2004515504A (ja) 2004-05-27
KR20040008115A (ko) 2004-01-28
HRP20030468A2 (en) 2005-04-30
IL156329A0 (en) 2004-01-04
US20020115620A1 (en) 2002-08-22
MXPA03005028A (es) 2004-01-29
EP1343798A1 (en) 2003-09-17
CA2431032A1 (en) 2002-06-13
RU2003117027A (ru) 2004-12-10
US6613747B2 (en) 2003-09-02
WO2002046204A1 (en) 2002-06-13
US6472372B1 (en) 2002-10-29
CN1310934C (zh) 2007-04-18
YU46303A (sh) 2006-05-25
CN1543472A (zh) 2004-11-03
AU2002230708A1 (en) 2002-06-18

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