YU46303A - 6-0-karbamoil ketolidni derivati eritromicina korisni kao antibakterijska sredstva - Google Patents
6-0-karbamoil ketolidni derivati eritromicina korisni kao antibakterijska sredstvaInfo
- Publication number
- YU46303A YU46303A YU46303A YUP46303A YU46303A YU 46303 A YU46303 A YU 46303A YU 46303 A YU46303 A YU 46303A YU P46303 A YUP46303 A YU P46303A YU 46303 A YU46303 A YU 46303A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- carbamoyl
- useful
- antibacterials
- erythromycin
- ketolide derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
6-0-karbamoil ketolidni antibakterijski agensi formule: gde su R1, R2, R3, R4, R5, R6, X, X', Y i Y' definisani u opisu, i u kojima supstituenti imaju značenje naznačeno u opisu. Ova jedinjenja su korisna kao antibakterijski agensi.[6-0-carbamoyl ketolide antibacterials of the formula: wherein R1, R2, R3, R4, R5, R6, X, X', Y, and Y' are as described herein and in which the substituents have the meaning indicated in the description. These compounds are useful as antibacterial agents.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25154700P | 2000-12-06 | 2000-12-06 | |
US09/773,788 US6472372B1 (en) | 2000-12-06 | 2001-02-01 | 6-O-Carbamoyl ketolide antibacterials |
Publications (1)
Publication Number | Publication Date |
---|---|
YU46303A true YU46303A (sh) | 2006-05-25 |
Family
ID=26941686
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU46303A YU46303A (sh) | 2000-12-06 | 2001-12-05 | 6-0-karbamoil ketolidni derivati eritromicina korisni kao antibakterijska sredstva |
Country Status (14)
Country | Link |
---|---|
US (2) | US6472372B1 (sh) |
EP (1) | EP1343798A1 (sh) |
JP (1) | JP2004515504A (sh) |
KR (1) | KR20040008115A (sh) |
CN (1) | CN1310934C (sh) |
AU (1) | AU2002230708A1 (sh) |
BR (1) | BR0116004A (sh) |
CA (1) | CA2431032A1 (sh) |
HR (1) | HRP20030468A2 (sh) |
IL (1) | IL156329A0 (sh) |
MX (1) | MXPA03005028A (sh) |
RU (1) | RU2003117027A (sh) |
WO (1) | WO2002046204A1 (sh) |
YU (1) | YU46303A (sh) |
Families Citing this family (54)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6472372B1 (en) * | 2000-12-06 | 2002-10-29 | Ortho-Mcneil Pharmaceuticals, Inc. | 6-O-Carbamoyl ketolide antibacterials |
PL370714A1 (en) * | 2001-12-05 | 2005-05-30 | Ortho-Mcneil Pharmaceutical, Inc. | 6-o-acyl ketolide derivatives of erythromycine useful as antibacterials |
WO2003090761A1 (en) * | 2002-04-25 | 2003-11-06 | Abbott Laboratories | 9-oxime macrolide antibacterials |
AU2003234650A1 (en) * | 2002-05-31 | 2003-12-19 | Janssen Pharmaceutica N.V. | 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents |
WO2005121160A2 (en) * | 2004-04-26 | 2005-12-22 | Johnson & Johnson Pharmaceutical Research & Development | 11, 12 cyclic thiocarbamate macrolide antibacterial agents |
US20080287376A1 (en) * | 2004-07-28 | 2008-11-20 | Mohammad Salman | Ketolide Derivatives as Antibacterial Agents |
US20090170790A1 (en) * | 2004-10-25 | 2009-07-02 | Biswajit Das | Ketolide derivatives as antibacterial agents |
EP1960413A2 (en) * | 2005-11-23 | 2008-08-27 | Ranbaxy Laboratories Limited | Macrolides derivatives as antibacterial agents |
EP1957508A2 (en) * | 2005-11-23 | 2008-08-20 | Ranbaxy Laboratories Limited | Ketolide derivatives as antibacterial agents |
JP2008044880A (ja) | 2006-08-15 | 2008-02-28 | Bayer Cropscience Ag | 殺虫性イソオキサゾリン類 |
AU2007347798A1 (en) * | 2006-08-30 | 2008-09-04 | Long Island University | Antimicrobial compositions |
US8218847B2 (en) | 2008-06-06 | 2012-07-10 | Superdimension, Ltd. | Hybrid registration method |
GB201105633D0 (en) * | 2011-04-01 | 2011-05-18 | Norbrook Lab Ltd | Antibotic compounds |
CN103242239B (zh) * | 2013-05-20 | 2015-09-23 | 洛阳师范学院 | 多取代嘧啶基苯甲醇及其制备方法 |
US9633431B2 (en) | 2014-07-02 | 2017-04-25 | Covidien Lp | Fluoroscopic pose estimation |
US9603668B2 (en) | 2014-07-02 | 2017-03-28 | Covidien Lp | Dynamic 3D lung map view for tool navigation inside the lung |
US9986983B2 (en) | 2014-10-31 | 2018-06-05 | Covidien Lp | Computed tomography enhanced fluoroscopic system, device, and method of utilizing the same |
US10716525B2 (en) | 2015-08-06 | 2020-07-21 | Covidien Lp | System and method for navigating to target and performing procedure on target utilizing fluoroscopic-based local three dimensional volume reconstruction |
US10702226B2 (en) | 2015-08-06 | 2020-07-07 | Covidien Lp | System and method for local three dimensional volume reconstruction using a standard fluoroscope |
US10674982B2 (en) | 2015-08-06 | 2020-06-09 | Covidien Lp | System and method for local three dimensional volume reconstruction using a standard fluoroscope |
US10575754B2 (en) | 2015-09-23 | 2020-03-03 | Covidien Lp | Catheter having a sensor and an extended working channel |
US11529190B2 (en) | 2017-01-30 | 2022-12-20 | Covidien Lp | Enhanced ablation and visualization techniques for percutaneous surgical procedures |
US11793579B2 (en) | 2017-02-22 | 2023-10-24 | Covidien Lp | Integration of multiple data sources for localization and navigation |
CN106928294A (zh) * | 2017-03-22 | 2017-07-07 | 上海启雁实业有限公司 | 制备酮内酯大环内酯类抗生素的方法 |
US10699448B2 (en) | 2017-06-29 | 2020-06-30 | Covidien Lp | System and method for identifying, marking and navigating to a target using real time two dimensional fluoroscopic data |
EP3694412A4 (en) | 2017-10-10 | 2021-08-18 | Covidien LP | SYSTEM AND METHOD FOR IDENTIFYING AND MARKING A TARGET IN A THREE-DIMENSIONAL FLUOROSCOPIC RECONSTRUCTION |
US10930064B2 (en) | 2018-02-08 | 2021-02-23 | Covidien Lp | Imaging reconstruction system and method |
US10905498B2 (en) | 2018-02-08 | 2021-02-02 | Covidien Lp | System and method for catheter detection in fluoroscopic images and updating displayed position of catheter |
US10893842B2 (en) | 2018-02-08 | 2021-01-19 | Covidien Lp | System and method for pose estimation of an imaging device and for determining the location of a medical device with respect to a target |
US10872449B2 (en) | 2018-05-02 | 2020-12-22 | Covidien Lp | System and method for constructing virtual radial ultrasound images from CT data and performing a surgical navigation procedure using virtual ultrasound images |
US11705238B2 (en) | 2018-07-26 | 2023-07-18 | Covidien Lp | Systems and methods for providing assistance during surgery |
US11071591B2 (en) | 2018-07-26 | 2021-07-27 | Covidien Lp | Modeling a collapsed lung using CT data |
US11944388B2 (en) | 2018-09-28 | 2024-04-02 | Covidien Lp | Systems and methods for magnetic interference correction |
US11877806B2 (en) | 2018-12-06 | 2024-01-23 | Covidien Lp | Deformable registration of computer-generated airway models to airway trees |
US11045075B2 (en) | 2018-12-10 | 2021-06-29 | Covidien Lp | System and method for generating a three-dimensional model of a surgical site |
US11617493B2 (en) | 2018-12-13 | 2023-04-04 | Covidien Lp | Thoracic imaging, distance measuring, surgical awareness, and notification system and method |
US11801113B2 (en) | 2018-12-13 | 2023-10-31 | Covidien Lp | Thoracic imaging, distance measuring, and notification system and method |
US11357593B2 (en) | 2019-01-10 | 2022-06-14 | Covidien Lp | Endoscopic imaging with augmented parallax |
US11625825B2 (en) | 2019-01-30 | 2023-04-11 | Covidien Lp | Method for displaying tumor location within endoscopic images |
US11564751B2 (en) | 2019-02-01 | 2023-01-31 | Covidien Lp | Systems and methods for visualizing navigation of medical devices relative to targets |
US11925333B2 (en) | 2019-02-01 | 2024-03-12 | Covidien Lp | System for fluoroscopic tracking of a catheter to update the relative position of a target and the catheter in a 3D model of a luminal network |
US11744643B2 (en) | 2019-02-04 | 2023-09-05 | Covidien Lp | Systems and methods facilitating pre-operative prediction of post-operative tissue function |
US11819285B2 (en) | 2019-04-05 | 2023-11-21 | Covidien Lp | Magnetic interference detection systems and methods |
US11975157B2 (en) | 2019-04-12 | 2024-05-07 | Covidien Lp | Method of manufacturing an elongated catheter having multiple sensors for three-dimensional location of the catheter |
US11269173B2 (en) | 2019-08-19 | 2022-03-08 | Covidien Lp | Systems and methods for displaying medical video images and/or medical 3D models |
US11931111B2 (en) | 2019-09-09 | 2024-03-19 | Covidien Lp | Systems and methods for providing surgical guidance |
US11864935B2 (en) | 2019-09-09 | 2024-01-09 | Covidien Lp | Systems and methods for pose estimation of a fluoroscopic imaging device and for three-dimensional imaging of body structures |
US11627924B2 (en) | 2019-09-24 | 2023-04-18 | Covidien Lp | Systems and methods for image-guided navigation of percutaneously-inserted devices |
US11847730B2 (en) | 2020-01-24 | 2023-12-19 | Covidien Lp | Orientation detection in fluoroscopic images |
US11380060B2 (en) | 2020-01-24 | 2022-07-05 | Covidien Lp | System and method for linking a segmentation graph to volumetric data |
US11922581B2 (en) | 2020-05-08 | 2024-03-05 | Coviden Lp | Systems and methods of controlling an operating room display using an augmented reality headset |
US11701492B2 (en) | 2020-06-04 | 2023-07-18 | Covidien Lp | Active distal tip drive |
US11950950B2 (en) | 2020-07-24 | 2024-04-09 | Covidien Lp | Zoom detection and fluoroscope movement detection for target overlay |
CN112300221B (zh) * | 2020-11-11 | 2022-04-15 | 艾美科健(中国)生物医药有限公司 | 一种加米霉素的合成方法 |
Family Cites Families (20)
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GB8521402D0 (en) * | 1985-08-28 | 1985-10-02 | Beecham Group Plc | Chemical compounds |
IL99995A (en) * | 1990-11-21 | 1997-11-20 | Roussel Uclaf | Erythromycin derivatives, their preparation and pharmaceutical compositions containing them |
US5559256A (en) * | 1992-07-20 | 1996-09-24 | E. R. Squibb & Sons, Inc. | Aminediol protease inhibitors |
ES2218604T3 (es) | 1995-11-08 | 2004-11-16 | Abbott Laboratories | Derivados triciclicos de eritromicina. |
TR199801254T2 (xx) * | 1995-12-29 | 1998-10-21 | Smithkline Beecham Corporation | Vitronektin resept�r� antagonistleri. |
CN100441591C (zh) | 1996-09-04 | 2008-12-10 | 艾博特公司 | 酮基内酯类化合物,其用途和制备方法以及药用组合物 |
UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
AU4033297A (en) * | 1996-09-06 | 1998-03-26 | Nisshin Oil Mills, Ltd., The | Sulfated glycolipid derivatives and medicinal compositions thereof |
CZ180799A3 (cs) | 1996-11-27 | 1999-09-15 | Taisho Pharmaceutical Co., Ltd. | Deriváty erythromycinu A |
FR2757168B1 (fr) * | 1996-12-12 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
UA59384C2 (uk) * | 1996-12-20 | 2003-09-15 | Пфайзер, Інк. | Похідні сульфонамідів та амідів як агоністи простагландину, фармацевтична композиція та способи лікування на їх основі |
AR015986A1 (es) * | 1997-10-29 | 2001-05-30 | Abbott Lab | Derivados de eritromicina puenteados en 6,11, composiciones farmaceuticas que los contienen, su uso para la manufactura de un medicamento y procedimientospara su preparacion |
CO4990960A1 (es) * | 1997-10-29 | 2000-12-26 | Abbott Lab | Derivados de cetolidos 2-halo-6-o sustituidos |
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US6399582B1 (en) | 1999-04-16 | 2002-06-04 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
MXPA01010524A (es) | 1999-04-16 | 2002-03-14 | Kosan Biosciences Inc | Agentes macrolidos anti-infecciosos. |
JP2003501439A (ja) | 1999-06-07 | 2003-01-14 | アボット・ラボラトリーズ | 6−o−カルバメートケトライド誘導体 |
CA2391297C (en) | 1999-12-02 | 2009-01-06 | Abbott Laboratories | 6-o-alkyl-2-nor-2-substituted ketolide derivatives |
EP1146051A3 (en) | 2000-04-10 | 2001-10-31 | Pfizer Products Inc. | Erythromycin A derivatives |
US6472372B1 (en) * | 2000-12-06 | 2002-10-29 | Ortho-Mcneil Pharmaceuticals, Inc. | 6-O-Carbamoyl ketolide antibacterials |
-
2001
- 2001-02-01 US US09/773,788 patent/US6472372B1/en not_active Expired - Lifetime
- 2001-12-05 AU AU2002230708A patent/AU2002230708A1/en not_active Abandoned
- 2001-12-05 EP EP01990950A patent/EP1343798A1/en not_active Withdrawn
- 2001-12-05 US US10/011,937 patent/US6613747B2/en not_active Expired - Lifetime
- 2001-12-05 WO PCT/US2001/047530 patent/WO2002046204A1/en active Application Filing
- 2001-12-05 JP JP2002547941A patent/JP2004515504A/ja active Pending
- 2001-12-05 MX MXPA03005028A patent/MXPA03005028A/es active IP Right Grant
- 2001-12-05 CA CA002431032A patent/CA2431032A1/en not_active Abandoned
- 2001-12-05 KR KR10-2003-7007629A patent/KR20040008115A/ko not_active Application Discontinuation
- 2001-12-05 CN CNB018223087A patent/CN1310934C/zh not_active Expired - Fee Related
- 2001-12-05 BR BR0116004-4A patent/BR0116004A/pt not_active IP Right Cessation
- 2001-12-05 YU YU46303A patent/YU46303A/sh unknown
- 2001-12-05 IL IL15632901A patent/IL156329A0/xx unknown
- 2001-12-05 RU RU2003117027/04A patent/RU2003117027A/ru not_active Application Discontinuation
-
2003
- 2003-06-06 HR HR20030468A patent/HRP20030468A2/hr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
MXPA03005028A (es) | 2004-01-29 |
HRP20030468A2 (en) | 2005-04-30 |
KR20040008115A (ko) | 2004-01-28 |
JP2004515504A (ja) | 2004-05-27 |
IL156329A0 (en) | 2004-01-04 |
US6613747B2 (en) | 2003-09-02 |
RU2003117027A (ru) | 2004-12-10 |
US20020115620A1 (en) | 2002-08-22 |
US6472372B1 (en) | 2002-10-29 |
BR0116004A (pt) | 2004-06-22 |
US20030013663A1 (en) | 2003-01-16 |
CN1543472A (zh) | 2004-11-03 |
WO2002046204A1 (en) | 2002-06-13 |
CA2431032A1 (en) | 2002-06-13 |
AU2002230708A1 (en) | 2002-06-18 |
EP1343798A1 (en) | 2003-09-17 |
CN1310934C (zh) | 2007-04-18 |
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