BR0107036A - Grânulos à base de amido e de lactose - Google Patents
Grânulos à base de amido e de lactoseInfo
- Publication number
- BR0107036A BR0107036A BR0107036-3A BR0107036A BR0107036A BR 0107036 A BR0107036 A BR 0107036A BR 0107036 A BR0107036 A BR 0107036A BR 0107036 A BR0107036 A BR 0107036A
- Authority
- BR
- Brazil
- Prior art keywords
- starch
- granules
- lactose
- lactose granules
- relates
- Prior art date
Links
- 239000008187 granular material Substances 0.000 title abstract 4
- GUBGYTABKSRVRQ-QKKXKWKRSA-N Lactose Natural products OC[C@H]1O[C@@H](O[C@H]2[C@H](O)[C@@H](O)C(O)O[C@@H]2CO)[C@H](O)[C@@H](O)[C@H]1O GUBGYTABKSRVRQ-QKKXKWKRSA-N 0.000 title abstract 3
- 229920002472 Starch Polymers 0.000 title abstract 3
- 239000008101 lactose Substances 0.000 title abstract 3
- 239000008107 starch Substances 0.000 title abstract 3
- 235000019698 starch Nutrition 0.000 title abstract 3
- 235000013305 food Nutrition 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000007787 solid Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T428/00—Stock material or miscellaneous articles
- Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
- Y10T428/2991—Coated
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Saccharide Compounds (AREA)
- General Preparation And Processing Of Foods (AREA)
- Glanulating (AREA)
- Grain Derivatives (AREA)
- Jellies, Jams, And Syrups (AREA)
- Formation And Processing Of Food Products (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
Abstract
"GRâNULOS à BASE DE AMIDO E DE LACTOSE". A invenção refere-se a grânulos que consistem em lactose e amido caracterizados pelo fato de que os referidos apresentam uma friabilidade inferior ou igual a 80 % e de preferência a 60% de acordo com um teste A. A mesma também refere-se ao processo de preparação dos ditos grânulos assim como à utilização dos mesmos para a preparação de formas sólidas nos domínios farmacêuticos ou alimentares.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP00402159A EP1175899B1 (fr) | 2000-07-27 | 2000-07-27 | Granules à base d'amidon et de lactose |
PCT/FR2001/002432 WO2002009673A1 (fr) | 2000-07-27 | 2001-07-25 | Granules a base d'amidon et de lactose |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0107036A true BR0107036A (pt) | 2002-06-04 |
Family
ID=8173789
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0107036-3A BR0107036A (pt) | 2000-07-27 | 2001-07-25 | Grânulos à base de amido e de lactose |
Country Status (23)
Country | Link |
---|---|
US (1) | US6770368B2 (pt) |
EP (1) | EP1175899B1 (pt) |
JP (1) | JP4394313B2 (pt) |
KR (1) | KR100869171B1 (pt) |
CN (1) | CN1253148C (pt) |
AT (1) | ATE371439T1 (pt) |
AU (1) | AU785135B2 (pt) |
BR (1) | BR0107036A (pt) |
CA (1) | CA2353363C (pt) |
CZ (1) | CZ303682B6 (pt) |
DE (1) | DE60036205T2 (pt) |
ES (1) | ES2292414T3 (pt) |
HU (1) | HU229277B1 (pt) |
IL (1) | IL148752A0 (pt) |
MX (1) | MXPA01007666A (pt) |
NO (1) | NO333750B1 (pt) |
NZ (1) | NZ517931A (pt) |
PL (1) | PL203778B1 (pt) |
RS (1) | RS49931B (pt) |
RU (1) | RU2286142C2 (pt) |
SK (1) | SK286951B6 (pt) |
WO (1) | WO2002009673A1 (pt) |
ZA (1) | ZA200202178B (pt) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2826549A1 (fr) * | 2001-06-28 | 2003-01-03 | Roquette Freres | Procede de preparation d'un comprime edulcorant et comprime edulcorant ainsi obtenu. |
FR2834889B1 (fr) * | 2002-01-18 | 2004-04-02 | Roquette Freres | Forme pharmaceutique solide orodispersible |
FR2834894B1 (fr) * | 2002-01-21 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de piribedil |
FR2834896B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible d'ivabradine |
FR2834890B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible d'agomelatine |
FR2834893B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de perindopril |
FR2834897B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de testosterone |
FR2834892B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de mitiglinide |
FR2834891B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de 2-({2-methoxy-2-[3(trifluoromethyl)phenyl]ethyl}amino)ethyl4 -(2-(9h-fluoren-9-yl)acetyl]amino}ethyl)benzoate |
US20030228370A1 (en) * | 2002-06-11 | 2003-12-11 | Michel Serpelloni | Orodispersible solid pharmaceutical form |
FR2857593B1 (fr) * | 2003-07-18 | 2005-10-14 | Servier Lab | Composition pharmaceutique orodispersible d'un compose antithrombotique |
GB0329208D0 (en) * | 2003-12-17 | 2004-01-21 | Ici Plc | Particulate materials |
GB0523810D0 (en) * | 2005-11-23 | 2006-01-04 | Astrazeneca Ab | Pharmaceutical compositions |
FR2894475B1 (fr) * | 2005-12-14 | 2008-05-16 | Servier Lab | Composition pharmaceutique orodispersible pour administra- -tion oromucosale ou sublinguale d'agomelatine |
CN101600431B (zh) * | 2006-12-07 | 2011-09-07 | 第一三共株式会社 | 具有改进贮存稳定性的药物组合物 |
JP5274261B2 (ja) * | 2006-12-07 | 2013-08-28 | 第一三共株式会社 | 低置換度ヒドロキシプロピルセルロースを含有する医薬組成物 |
KR101442862B1 (ko) * | 2006-12-07 | 2014-09-22 | 다이이찌 산쿄 가부시키가이샤 | 만니톨 또는 유당을 함유하는 고형 제제 |
KR101665705B1 (ko) * | 2006-12-07 | 2016-10-12 | 다이이찌 산쿄 가부시키가이샤 | 안정성이 개선된 필름 코팅 제제 |
FR2933299B1 (fr) | 2008-07-04 | 2012-02-03 | Roquette Freres | Mannitol orodispersible |
DE102008047910A1 (de) | 2008-09-19 | 2010-03-25 | Molkerei Meggle Wasserburg Gmbh & Co. Kg | Tablettierhilfsstoff auf Laktose- und Cellulosebasis |
ES2758624T3 (es) * | 2009-02-12 | 2020-05-06 | Fuji Chem Ind Co Ltd | Composición de partículas desintegrantes y material de desintegración rápida moldeado por compresión que comprende la misma |
FR2944971B1 (fr) * | 2009-04-30 | 2012-09-07 | Roquette Freres | Coagglomerats de mannitol et d'amidon granulaire comprimables et a ecoulement libre |
JP2013529633A (ja) * | 2010-06-23 | 2013-07-22 | コルゲート・パーモリブ・カンパニー | 有効なカプセル化剤を形成させるためのラクトースマトリックス中への成分のカプセル化 |
FR2966828B1 (fr) * | 2010-11-02 | 2012-12-28 | Roquette Freres | Poudre de polysaccharide et de polyol, comprimable et de haute viscosite |
JP5483482B2 (ja) | 2011-05-23 | 2014-05-07 | 三井製糖株式会社 | 糖液から固形物を製造する方法及び固形物 |
CN102516321A (zh) * | 2011-12-08 | 2012-06-27 | 上海天伟生物制药有限公司 | 一种药用乳糖及其制备方法和用途 |
JP5276199B1 (ja) * | 2012-03-23 | 2013-08-28 | 池田食研株式会社 | 多孔質顆粒の製造方法 |
US9522964B2 (en) * | 2012-04-03 | 2016-12-20 | Development, Inc. | Micronized starch and methods for manufacturing same |
CA2955845C (en) | 2014-07-21 | 2022-08-16 | Roquette Freres | Sugar compositions for tableting by direct compression |
EP3002005A1 (en) | 2014-09-30 | 2016-04-06 | Molkerei Meggle Wasserburg GmbH & Co. Kg | Direct compression excipient based on lactose, cellulose and starch |
EP3034070A1 (en) * | 2014-12-18 | 2016-06-22 | Omya International AG | Method for the production of a pharmaceutical delivery system |
JP6544564B2 (ja) * | 2015-04-20 | 2019-07-17 | 清水建設株式会社 | 模擬粉体、及び粉体飛散状態評価方法 |
US10820608B1 (en) | 2015-10-26 | 2020-11-03 | The Hershey Company | Hard candy confections with low hygroscopicity |
EP3575285A4 (en) | 2017-01-24 | 2020-08-12 | Medshine Discovery Inc. | LSD1 INHIBITOR AND MANUFACTURING METHOD AND APPLICATION OF IT |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE575343A (pt) * | 1955-09-09 | |||
AT376147B (de) * | 1980-12-15 | 1984-10-10 | Gergely Gerhard | Verfahren und vorrichtung zum granulieren eines pulvergemisches |
DE3505433A1 (de) * | 1985-02-16 | 1986-08-21 | Basf Ag, 6700 Ludwigshafen | Direkttablettierhilfsmittel |
US5043170A (en) * | 1989-02-14 | 1991-08-27 | Hoffmann-La Roche Inc. | Animal feed composition containing a vitamin D metabolite |
JPH0584054A (ja) * | 1991-09-27 | 1993-04-06 | Kunoole Shokuhin Kk | スープまたはソース粉末もしくは顆粒の製造法 |
JP3349535B2 (ja) * | 1993-01-12 | 2002-11-25 | フロイント産業株式会社 | 球形顆粒の製造方法 |
JPH08298956A (ja) * | 1995-05-10 | 1996-11-19 | Ajinomoto Co Inc | 顆粒状調味料の製造方法 |
JPH0937737A (ja) * | 1995-05-25 | 1997-02-10 | Tokiwa Kanpo Seiyaku:Kk | 菊花含有健康食品 |
JP3611652B2 (ja) * | 1995-10-30 | 2005-01-19 | 長谷川香料株式会社 | コーティング粉末の製造方法 |
DE19603984A1 (de) * | 1996-02-05 | 1997-08-07 | Bayer Ag | Granulate von Triazinen |
JP3934179B2 (ja) * | 1996-07-11 | 2007-06-20 | 不二製油株式会社 | 動物の体内へ摂取される物質からなる粉体を造粒する方法及び造粒物 |
JP3447042B2 (ja) * | 1997-07-23 | 2003-09-16 | フロイント産業株式会社 | 単一物質球形粒の製造方法 |
-
2000
- 2000-07-27 ES ES00402159T patent/ES2292414T3/es not_active Expired - Lifetime
- 2000-07-27 AT AT00402159T patent/ATE371439T1/de not_active IP Right Cessation
- 2000-07-27 EP EP00402159A patent/EP1175899B1/fr not_active Expired - Lifetime
- 2000-07-27 DE DE60036205T patent/DE60036205T2/de not_active Expired - Lifetime
-
2001
- 2001-07-13 US US09/905,569 patent/US6770368B2/en not_active Expired - Lifetime
- 2001-07-23 CA CA2353363A patent/CA2353363C/fr not_active Expired - Lifetime
- 2001-07-25 SK SK370-2002A patent/SK286951B6/sk not_active IP Right Cessation
- 2001-07-25 WO PCT/FR2001/002432 patent/WO2002009673A1/fr active IP Right Grant
- 2001-07-25 HU HU0203064A patent/HU229277B1/hu unknown
- 2001-07-25 CN CNB01802176XA patent/CN1253148C/zh not_active Expired - Lifetime
- 2001-07-25 RU RU2002111360/15A patent/RU2286142C2/ru active
- 2001-07-25 NZ NZ517931A patent/NZ517931A/en not_active IP Right Cessation
- 2001-07-25 KR KR1020027003970A patent/KR100869171B1/ko active IP Right Grant
- 2001-07-25 BR BR0107036-3A patent/BR0107036A/pt not_active Application Discontinuation
- 2001-07-25 RS YUP-220/02A patent/RS49931B/sr unknown
- 2001-07-25 IL IL14875201A patent/IL148752A0/xx unknown
- 2001-07-25 CZ CZ20020978A patent/CZ303682B6/cs not_active IP Right Cessation
- 2001-07-25 AU AU79909/01A patent/AU785135B2/en not_active Expired
- 2001-07-25 PL PL353056A patent/PL203778B1/pl unknown
- 2001-07-26 JP JP2001226631A patent/JP4394313B2/ja not_active Expired - Lifetime
- 2001-07-27 MX MXPA01007666A patent/MXPA01007666A/es active IP Right Grant
-
2002
- 2002-03-18 ZA ZA200202178A patent/ZA200202178B/xx unknown
- 2002-03-21 NO NO20021424A patent/NO333750B1/no not_active IP Right Cessation
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B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) DA LPI |
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B12B | Appeal against refusal [chapter 12.2 patent gazette] | ||
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