BR0107036A - Grânulos à base de amido e de lactose - Google Patents

Grânulos à base de amido e de lactose

Info

Publication number
BR0107036A
BR0107036A BR0107036-3A BR0107036A BR0107036A BR 0107036 A BR0107036 A BR 0107036A BR 0107036 A BR0107036 A BR 0107036A BR 0107036 A BR0107036 A BR 0107036A
Authority
BR
Brazil
Prior art keywords
starch
granules
lactose
lactose granules
relates
Prior art date
Application number
BR0107036-3A
Other languages
English (en)
Inventor
Oliver Luhn
Original Assignee
Roquette Freres
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roquette Freres filed Critical Roquette Freres
Publication of BR0107036A publication Critical patent/BR0107036A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T428/00Stock material or miscellaneous articles
    • Y10T428/29Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
    • Y10T428/2982Particulate matter [e.g., sphere, flake, etc.]
    • Y10T428/2991Coated

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • General Preparation And Processing Of Foods (AREA)
  • Glanulating (AREA)
  • Grain Derivatives (AREA)
  • Jellies, Jams, And Syrups (AREA)
  • Formation And Processing Of Food Products (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)

Abstract

"GRâNULOS à BASE DE AMIDO E DE LACTOSE". A invenção refere-se a grânulos que consistem em lactose e amido caracterizados pelo fato de que os referidos apresentam uma friabilidade inferior ou igual a 80 % e de preferência a 60% de acordo com um teste A. A mesma também refere-se ao processo de preparação dos ditos grânulos assim como à utilização dos mesmos para a preparação de formas sólidas nos domínios farmacêuticos ou alimentares.
BR0107036-3A 2000-07-27 2001-07-25 Grânulos à base de amido e de lactose BR0107036A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00402159A EP1175899B1 (fr) 2000-07-27 2000-07-27 Granules à base d'amidon et de lactose
PCT/FR2001/002432 WO2002009673A1 (fr) 2000-07-27 2001-07-25 Granules a base d'amidon et de lactose

Publications (1)

Publication Number Publication Date
BR0107036A true BR0107036A (pt) 2002-06-04

Family

ID=8173789

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0107036-3A BR0107036A (pt) 2000-07-27 2001-07-25 Grânulos à base de amido e de lactose

Country Status (23)

Country Link
US (1) US6770368B2 (pt)
EP (1) EP1175899B1 (pt)
JP (1) JP4394313B2 (pt)
KR (1) KR100869171B1 (pt)
CN (1) CN1253148C (pt)
AT (1) ATE371439T1 (pt)
AU (1) AU785135B2 (pt)
BR (1) BR0107036A (pt)
CA (1) CA2353363C (pt)
CZ (1) CZ303682B6 (pt)
DE (1) DE60036205T2 (pt)
ES (1) ES2292414T3 (pt)
HU (1) HU229277B1 (pt)
IL (1) IL148752A0 (pt)
MX (1) MXPA01007666A (pt)
NO (1) NO333750B1 (pt)
NZ (1) NZ517931A (pt)
PL (1) PL203778B1 (pt)
RS (1) RS49931B (pt)
RU (1) RU2286142C2 (pt)
SK (1) SK286951B6 (pt)
WO (1) WO2002009673A1 (pt)
ZA (1) ZA200202178B (pt)

Families Citing this family (34)

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FR2826549A1 (fr) * 2001-06-28 2003-01-03 Roquette Freres Procede de preparation d'un comprime edulcorant et comprime edulcorant ainsi obtenu.
FR2834889B1 (fr) * 2002-01-18 2004-04-02 Roquette Freres Forme pharmaceutique solide orodispersible
FR2834894B1 (fr) * 2002-01-21 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de piribedil
FR2834896B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible d'ivabradine
FR2834890B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible d'agomelatine
FR2834893B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de perindopril
FR2834897B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de testosterone
FR2834892B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de mitiglinide
FR2834891B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de 2-({2-methoxy-2-[3(trifluoromethyl)phenyl]ethyl}amino)ethyl4 -(2-(9h-fluoren-9-yl)acetyl]amino}ethyl)benzoate
US20030228370A1 (en) * 2002-06-11 2003-12-11 Michel Serpelloni Orodispersible solid pharmaceutical form
FR2857593B1 (fr) * 2003-07-18 2005-10-14 Servier Lab Composition pharmaceutique orodispersible d'un compose antithrombotique
GB0329208D0 (en) * 2003-12-17 2004-01-21 Ici Plc Particulate materials
GB0523810D0 (en) * 2005-11-23 2006-01-04 Astrazeneca Ab Pharmaceutical compositions
FR2894475B1 (fr) * 2005-12-14 2008-05-16 Servier Lab Composition pharmaceutique orodispersible pour administra- -tion oromucosale ou sublinguale d'agomelatine
CN101600431B (zh) * 2006-12-07 2011-09-07 第一三共株式会社 具有改进贮存稳定性的药物组合物
JP5274261B2 (ja) * 2006-12-07 2013-08-28 第一三共株式会社 低置換度ヒドロキシプロピルセルロースを含有する医薬組成物
KR101442862B1 (ko) * 2006-12-07 2014-09-22 다이이찌 산쿄 가부시키가이샤 만니톨 또는 유당을 함유하는 고형 제제
KR101665705B1 (ko) * 2006-12-07 2016-10-12 다이이찌 산쿄 가부시키가이샤 안정성이 개선된 필름 코팅 제제
FR2933299B1 (fr) 2008-07-04 2012-02-03 Roquette Freres Mannitol orodispersible
DE102008047910A1 (de) 2008-09-19 2010-03-25 Molkerei Meggle Wasserburg Gmbh & Co. Kg Tablettierhilfsstoff auf Laktose- und Cellulosebasis
ES2758624T3 (es) * 2009-02-12 2020-05-06 Fuji Chem Ind Co Ltd Composición de partículas desintegrantes y material de desintegración rápida moldeado por compresión que comprende la misma
FR2944971B1 (fr) * 2009-04-30 2012-09-07 Roquette Freres Coagglomerats de mannitol et d'amidon granulaire comprimables et a ecoulement libre
JP2013529633A (ja) * 2010-06-23 2013-07-22 コルゲート・パーモリブ・カンパニー 有効なカプセル化剤を形成させるためのラクトースマトリックス中への成分のカプセル化
FR2966828B1 (fr) * 2010-11-02 2012-12-28 Roquette Freres Poudre de polysaccharide et de polyol, comprimable et de haute viscosite
JP5483482B2 (ja) 2011-05-23 2014-05-07 三井製糖株式会社 糖液から固形物を製造する方法及び固形物
CN102516321A (zh) * 2011-12-08 2012-06-27 上海天伟生物制药有限公司 一种药用乳糖及其制备方法和用途
JP5276199B1 (ja) * 2012-03-23 2013-08-28 池田食研株式会社 多孔質顆粒の製造方法
US9522964B2 (en) * 2012-04-03 2016-12-20 Development, Inc. Micronized starch and methods for manufacturing same
CA2955845C (en) 2014-07-21 2022-08-16 Roquette Freres Sugar compositions for tableting by direct compression
EP3002005A1 (en) 2014-09-30 2016-04-06 Molkerei Meggle Wasserburg GmbH & Co. Kg Direct compression excipient based on lactose, cellulose and starch
EP3034070A1 (en) * 2014-12-18 2016-06-22 Omya International AG Method for the production of a pharmaceutical delivery system
JP6544564B2 (ja) * 2015-04-20 2019-07-17 清水建設株式会社 模擬粉体、及び粉体飛散状態評価方法
US10820608B1 (en) 2015-10-26 2020-11-03 The Hershey Company Hard candy confections with low hygroscopicity
EP3575285A4 (en) 2017-01-24 2020-08-12 Medshine Discovery Inc. LSD1 INHIBITOR AND MANUFACTURING METHOD AND APPLICATION OF IT

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BE575343A (pt) * 1955-09-09
AT376147B (de) * 1980-12-15 1984-10-10 Gergely Gerhard Verfahren und vorrichtung zum granulieren eines pulvergemisches
DE3505433A1 (de) * 1985-02-16 1986-08-21 Basf Ag, 6700 Ludwigshafen Direkttablettierhilfsmittel
US5043170A (en) * 1989-02-14 1991-08-27 Hoffmann-La Roche Inc. Animal feed composition containing a vitamin D metabolite
JPH0584054A (ja) * 1991-09-27 1993-04-06 Kunoole Shokuhin Kk スープまたはソース粉末もしくは顆粒の製造法
JP3349535B2 (ja) * 1993-01-12 2002-11-25 フロイント産業株式会社 球形顆粒の製造方法
JPH08298956A (ja) * 1995-05-10 1996-11-19 Ajinomoto Co Inc 顆粒状調味料の製造方法
JPH0937737A (ja) * 1995-05-25 1997-02-10 Tokiwa Kanpo Seiyaku:Kk 菊花含有健康食品
JP3611652B2 (ja) * 1995-10-30 2005-01-19 長谷川香料株式会社 コーティング粉末の製造方法
DE19603984A1 (de) * 1996-02-05 1997-08-07 Bayer Ag Granulate von Triazinen
JP3934179B2 (ja) * 1996-07-11 2007-06-20 不二製油株式会社 動物の体内へ摂取される物質からなる粉体を造粒する方法及び造粒物
JP3447042B2 (ja) * 1997-07-23 2003-09-16 フロイント産業株式会社 単一物質球形粒の製造方法

Also Published As

Publication number Publication date
AU785135B2 (en) 2006-10-05
HU229277B1 (en) 2013-10-28
AU7990901A (en) 2002-02-13
ES2292414T3 (es) 2008-03-16
RU2286142C2 (ru) 2006-10-27
CA2353363A1 (fr) 2002-01-27
CZ2002978A3 (cs) 2002-06-12
SK286951B6 (sk) 2009-08-06
RS49931B (sr) 2008-09-29
US6770368B2 (en) 2004-08-03
DE60036205T2 (de) 2008-05-21
PL353056A1 (en) 2003-10-06
US20020035248A1 (en) 2002-03-21
CA2353363C (fr) 2010-06-01
ATE371439T1 (de) 2007-09-15
CN1386064A (zh) 2002-12-18
YU22002A (sh) 2004-09-03
KR100869171B1 (ko) 2008-11-19
NZ517931A (en) 2003-11-28
WO2002009673A1 (fr) 2002-02-07
NO333750B1 (no) 2013-09-09
CZ303682B6 (cs) 2013-03-06
CN1253148C (zh) 2006-04-26
NO20021424D0 (no) 2002-03-21
SK3702002A3 (en) 2002-08-06
KR20020063868A (ko) 2002-08-05
DE60036205D1 (de) 2007-10-11
RU2002111360A (ru) 2004-01-10
NO20021424L (no) 2002-03-21
HUP0203064A2 (en) 2003-03-28
ZA200202178B (en) 2003-06-05
EP1175899A1 (fr) 2002-01-30
PL203778B1 (pl) 2009-11-30
IL148752A0 (en) 2002-09-12
EP1175899B1 (fr) 2007-08-29
JP4394313B2 (ja) 2010-01-06
MXPA01007666A (es) 2004-08-11
JP2002142690A (ja) 2002-05-21

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) DA LPI

B12B Appeal against refusal [chapter 12.2 patent gazette]
B08E Application fees: payment of additional fee required [chapter 8.5 patent gazette]

Free format text: COMPLEMENTAR A RETRIBUICAO DA 10A E 11A ANUIDADES DE ACORDO COM TABELA VIGENTE, REFERENTE AS GUIAS DE RECOLHIMENTO 221004887196 E 221106208131.

B08G Application fees: restoration [chapter 8.7 patent gazette]