BG64114B1 - Гранулат за получаване на бързо разпадащи се и бързо разтварящи се състави с високо съдържание на лекарствено средство - Google Patents

Гранулат за получаване на бързо разпадащи се и бързо разтварящи се състави с високо съдържание на лекарствено средство Download PDF

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Publication number
BG64114B1
BG64114B1 BG103047A BG10304798A BG64114B1 BG 64114 B1 BG64114 B1 BG 64114B1 BG 103047 A BG103047 A BG 103047A BG 10304798 A BG10304798 A BG 10304798A BG 64114 B1 BG64114 B1 BG 64114B1
Authority
BG
Bulgaria
Prior art keywords
weight
water
cellulose
granulate
tablets
Prior art date
Application number
BG103047A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG103047A (en
Inventor
Bernardus L.J. Dijkgraaf
Aart Muehlenbruch
Original Assignee
Yamanouchi Europe B.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8224133&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG64114(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Yamanouchi Europe B.V. filed Critical Yamanouchi Europe B.V.
Publication of BG103047A publication Critical patent/BG103047A/xx
Publication of BG64114B1 publication Critical patent/BG64114B1/bg

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • General Preparation And Processing Of Foods (AREA)
  • Jellies, Jams, And Syrups (AREA)
BG103047A 1996-07-03 1998-12-30 Гранулат за получаване на бързо разпадащи се и бързо разтварящи се състави с високо съдържание на лекарствено средство BG64114B1 (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP96201829 1996-07-03
US08/770,421 US5837292A (en) 1996-07-03 1996-12-20 Granulate for the preparation of fast-disintegrating and fast-dissolving compositions containing a high amount of drug
PCT/EP1997/003250 WO1998001114A1 (fr) 1996-07-03 1997-06-19 Granules destines a la preparation de compositions a haut pouvoir de desintegration et de dissolution, a teneur elevee en medicament

Publications (2)

Publication Number Publication Date
BG103047A BG103047A (en) 1999-07-30
BG64114B1 true BG64114B1 (bg) 2004-01-30

Family

ID=8224133

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103047A BG64114B1 (bg) 1996-07-03 1998-12-30 Гранулат за получаване на бързо разпадащи се и бързо разтварящи се състави с високо съдържание на лекарствено средство

Country Status (36)

Country Link
US (1) US5837292A (fr)
EP (1) EP0910344B1 (fr)
JP (1) JP4159607B2 (fr)
CN (1) CN1131025C (fr)
AR (1) AR008252A1 (fr)
AT (1) ATE237314T1 (fr)
AU (1) AU731276B2 (fr)
BG (1) BG64114B1 (fr)
BR (1) BR9710181B1 (fr)
CA (1) CA2258841C (fr)
CO (1) CO4890859A1 (fr)
CZ (1) CZ295893B6 (fr)
DE (1) DE69720995T2 (fr)
DK (1) DK0910344T3 (fr)
EA (1) EA001537B1 (fr)
EG (1) EG23814A (fr)
ES (1) ES2197351T3 (fr)
HK (1) HK1021511A1 (fr)
HU (1) HU225115B1 (fr)
ID (1) ID17128A (fr)
IL (1) IL127364A (fr)
JO (1) JO1969B1 (fr)
MY (1) MY116124A (fr)
NO (1) NO320767B1 (fr)
NZ (1) NZ333247A (fr)
PE (1) PE89798A1 (fr)
PL (1) PL188235B1 (fr)
PT (1) PT910344E (fr)
SI (1) SI0910344T1 (fr)
SK (1) SK284175B6 (fr)
TN (1) TNSN97114A1 (fr)
TR (1) TR199802762T2 (fr)
TW (1) TW473392B (fr)
UA (1) UA61917C2 (fr)
WO (1) WO1998001114A1 (fr)
ZA (1) ZA975848B (fr)

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IT1305308B1 (it) * 1999-03-26 2001-05-04 Biosint S P A Granulato ad alto contenuto di l-carnitina o alcanoil-l-carnitina,particolarmente adatto alla produzione di compresse per compressione
AU4441899A (en) * 1999-05-14 2000-12-05 Eli Lilly And Company Process for preparing pharmaceutical bulk material having uniform dissolution
HU227070B1 (en) * 1999-08-11 2010-06-28 Egis Gyogyszergyar Nyilvanosan Immediate release pharmaceutical composition containing ciprofloxacin and process for its production
AR028253A1 (es) * 2000-03-16 2003-04-30 Pfizer Prod Inc Inhibidores de la glucogeno fosforilasa
FR2816507B1 (fr) * 2000-11-16 2003-02-28 Ethypharm Lab Prod Ethiques Microgranules a base de principe actif, procede de fabrication et compositons pharmaceutiques integrant lesdits microgranules
US6733781B2 (en) 2000-12-06 2004-05-11 Wyeth Fast dissolving tablet
US7799342B2 (en) * 2000-12-06 2010-09-21 Wyeth Llc Fast dissolving tablet
HUP0303178A3 (en) * 2001-02-05 2008-03-28 R P Scherer Technologies Methods and compositions for reducing the taste of pharmaceutically active agents
EP1285649A1 (fr) * 2001-08-23 2003-02-26 Cimex AG Comprimé dispersible à deux couches comprenant de l'amoxicilline et du clavulanate dans des couches séparées
RU2004123621A (ru) * 2002-02-01 2005-04-10 Пфайзер Продактс Инк. (Us) Лекарственные формы с немедленным высвобождением, содержащие твердые дисперсии лекарств
US20030229101A1 (en) * 2002-06-06 2003-12-11 Sherman Bernard Charles Tablets comprising ciprofloxacin hydrochloride
KR20050062514A (ko) * 2002-07-16 2005-06-23 랜박시 래보러터리스 리미티드 경구 투여용 분산성 정제
AU2003247023A1 (en) * 2002-08-02 2004-02-25 Ranbaxy Laboratories Limited A process for the preparation of dispersible tablet of cephalexin
JP4702763B2 (ja) * 2003-07-30 2011-06-15 塩野義製薬株式会社 結晶セルロースを含有する安定な錠剤
US7838029B1 (en) * 2003-07-31 2010-11-23 Watson Laboratories, Inc. Mirtazapine solid dosage forms
US7390503B1 (en) 2003-08-22 2008-06-24 Barr Laboratories, Inc. Ondansetron orally disintegrating tablets
PL3395338T3 (pl) * 2003-09-12 2019-10-31 Amgen Inc Szybko rozpuszczająca się formulacja zawierająca cynakalcet HCl
US20050089558A1 (en) * 2003-10-28 2005-04-28 Alamo Pharmaceuticals, Llc Compositions and methods for the co-formulation and administration of tramadol and propoxyphene
EP1681050A1 (fr) * 2005-01-13 2006-07-19 Strides Arcolab Limited Composition pharmaceutique dispersible avec libération prolongée
US7811604B1 (en) 2005-11-14 2010-10-12 Barr Laboratories, Inc. Non-effervescent, orally disintegrating solid pharmaceutical dosage forms comprising clozapine and methods of making and using the same
US8617597B2 (en) 2006-07-06 2013-12-31 Bayer Intellectual Property Gmbh Pharmaceutical composition containing a tetrahydrofolic acid
WO2008008120A1 (fr) * 2006-07-14 2008-01-17 Fmc Corporation Forme solide
JP5201819B2 (ja) * 2006-11-22 2013-06-05 エスエス製薬株式会社 固形組成物
US20080311162A1 (en) * 2007-05-16 2008-12-18 Olivia Darmuzey Solid form
JP5637624B2 (ja) * 2009-02-12 2014-12-10 富士化学工業株式会社 崩壊性粒子組成物及びそれを用いた速崩壊性圧縮成型物
WO2011152808A1 (fr) * 2010-06-03 2011-12-08 Mahmut Bilgic Formulation comprenant du cefpodoxime proxétil et de l'acide clavulanique
CN101912373B (zh) * 2010-08-24 2012-01-04 北京京丰制药有限公司 稳定的头孢克洛分散片及其制备方法
WO2013151517A1 (fr) * 2012-04-04 2013-10-10 Mahmut Bilgic Formulations en comprimés comprenant du cefpodoxime proxétil et de l'acide clavulanique
JP2015063521A (ja) * 2013-09-02 2015-04-09 科研製薬株式会社 高い薬物含有率を有する錠剤及びその製造方法
CN106255512B (zh) 2014-04-21 2021-01-01 株式会社大赛璐 含有微小纤维状纤维素的崩解性颗粒组合物
CN110051639B (zh) * 2019-03-15 2021-08-31 河北嘉迈医药科技有限公司 一种快速崩解型尼麦角林片及其制备方法
CN117683469A (zh) * 2023-10-24 2024-03-12 绍兴拓邦新能源股份有限公司 一种晶硅片背面碱抛光固态添加剂及其制备方法

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Also Published As

Publication number Publication date
CO4890859A1 (es) 2000-02-28
TR199802762T2 (xx) 1999-03-22
ES2197351T3 (es) 2004-01-01
PL330958A1 (en) 1999-06-21
HUP9903308A2 (hu) 2000-03-28
EA001537B1 (ru) 2001-04-23
DK0910344T3 (da) 2003-07-07
JO1969B1 (en) 1997-12-15
IL127364A (en) 2003-04-10
PL188235B1 (pl) 2004-12-31
CZ699A3 (cs) 1999-04-14
ZA975848B (en) 1999-04-12
MY116124A (en) 2003-11-28
CA2258841C (fr) 2006-05-30
BR9710181B1 (pt) 2009-08-11
JP2000513727A (ja) 2000-10-17
JP4159607B2 (ja) 2008-10-01
IL127364A0 (en) 1999-10-28
NO986157L (no) 1999-02-01
WO1998001114A1 (fr) 1998-01-15
BG103047A (en) 1999-07-30
EA199900075A1 (ru) 1999-06-24
PT910344E (pt) 2003-09-30
AU731276B2 (en) 2001-03-29
EP0910344A1 (fr) 1999-04-28
EG23814A (en) 2007-09-12
SI0910344T1 (en) 2003-08-31
ATE237314T1 (de) 2003-05-15
CA2258841A1 (fr) 1998-01-15
DE69720995T2 (de) 2003-11-13
NO320767B1 (no) 2006-01-23
AU3342197A (en) 1998-02-02
SK284175B6 (sk) 2004-10-05
CN1131025C (zh) 2003-12-17
AR008252A1 (es) 1999-12-29
CN1224348A (zh) 1999-07-28
TNSN97114A1 (fr) 2005-03-15
NO986157D0 (no) 1998-12-28
CZ295893B6 (cs) 2005-11-16
UA61917C2 (uk) 2003-12-15
TW473392B (en) 2002-01-21
NZ333247A (en) 2000-07-28
HU225115B1 (hu) 2006-06-28
DE69720995D1 (de) 2003-05-22
EP0910344B1 (fr) 2003-04-16
PE89798A1 (es) 1999-01-12
BR9710181A (pt) 1999-08-10
HK1021511A1 (en) 2000-06-16
HUP9903308A3 (en) 2001-03-28
US5837292A (en) 1998-11-17
SK176798A3 (en) 2000-04-10
ID17128A (id) 1997-12-04

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