BG61767B1 - Кристали от антимикробно съединение - Google Patents

Кристали от антимикробно съединение Download PDF

Info

Publication number
BG61767B1
BG61767B1 BG99035A BG9903594A BG61767B1 BG 61767 B1 BG61767 B1 BG 61767B1 BG 99035 A BG99035 A BG 99035A BG 9903594 A BG9903594 A BG 9903594A BG 61767 B1 BG61767 B1 BG 61767B1
Authority
BG
Bulgaria
Prior art keywords
weak
fluoro
dihydroquinoline
hydrate
carboxylic acid
Prior art date
Application number
BG99035A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG99035A (bg
Inventor
Youichi Kimura
Katsuhiro Kawakami
Norimasa Mikata
Keiji Uchiyama
Tazuo Uemura
Yusuke Yukimoto
Original Assignee
Daiichi Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Pharmaceutical Co., Ltd. filed Critical Daiichi Pharmaceutical Co., Ltd.
Publication of BG99035A publication Critical patent/BG99035A/bg
Publication of BG61767B1 publication Critical patent/BG61767B1/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cephalosporin Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines Containing Plant Substances (AREA)
BG99035A 1993-09-10 1994-09-09 Кристали от антимикробно съединение BG61767B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP22538093 1993-09-10

Publications (2)

Publication Number Publication Date
BG99035A BG99035A (bg) 1995-05-31
BG61767B1 true BG61767B1 (bg) 1998-05-29

Family

ID=16828452

Family Applications (1)

Application Number Title Priority Date Filing Date
BG99035A BG61767B1 (bg) 1993-09-10 1994-09-09 Кристали от антимикробно съединение

Country Status (32)

Country Link
US (1) US5693814A (sk)
EP (1) EP0643058B1 (sk)
JP (1) JP3793583B2 (sk)
KR (1) KR100336247B1 (sk)
CN (1) CN1057297C (sk)
AT (1) ATE181069T1 (sk)
AU (1) AU679094B2 (sk)
BG (1) BG61767B1 (sk)
CA (1) CA2131761C (sk)
CZ (3) CZ284837B6 (sk)
DE (1) DE69418953T2 (sk)
DK (1) DK0643058T3 (sk)
ES (1) ES2136142T3 (sk)
FI (1) FI110777B (sk)
GE (1) GEP19981355B (sk)
GR (1) GR3031012T3 (sk)
HR (1) HRP940506B1 (sk)
HU (1) HU224970B1 (sk)
IL (2) IL123910A (sk)
LV (1) LV11322B (sk)
MY (1) MY112574A (sk)
NO (2) NO307419B1 (sk)
NZ (1) NZ264422A (sk)
PL (1) PL180163B1 (sk)
RU (1) RU2126402C1 (sk)
SG (1) SG50492A1 (sk)
SI (1) SI9400349B (sk)
SK (3) SK283190B6 (sk)
TW (1) TW393481B (sk)
UA (1) UA41312C2 (sk)
YU (1) YU49132B (sk)
ZA (1) ZA946853B (sk)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19546249A1 (de) * 1995-12-12 1997-06-19 Bayer Ag Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen
DE69802692D1 (de) * 1997-06-26 2002-01-10 Dong Wha Pharm Ind Co Ltd Derivate der chinoloncarbonsäure
JP2001300293A (ja) * 2000-04-25 2001-10-30 Nipro Corp 無機無水物または有機無水物の製造法
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
CN102718746B (zh) * 2012-06-18 2014-10-29 南京优科生物医药研究有限公司 西他沙星富马酸盐晶型a和其制药用途
CN103539776B (zh) * 2012-07-16 2016-06-08 深圳信立泰药业股份有限公司 一种西他沙星晶型及其制备方法
CN106749174B (zh) * 2016-12-06 2019-06-18 山东裕欣药业有限公司 一种西他沙星二水合物晶型、制备方法及其组合物片剂

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE203719C (sk) * 1907-11-02 1908-10-20
DK170473B1 (da) * 1985-06-20 1995-09-11 Daiichi Seiyaku Co S(-)-pyridobenzoxazinforbindelser
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co History of pyridonecarboxylic acid, their preparation and pharmaceutical preparations containing them
CA1332605C (en) * 1988-10-03 1994-10-18 Yasuhiro Nishitani Pyridonecarboxylic acids
TW208013B (sk) * 1990-03-01 1993-06-21 Daiichi Co Ltd
US4994809A (en) * 1990-03-07 1991-02-19 Hughes Aircraft Company Polystatic correlating radar
MY109714A (en) * 1990-10-18 1997-04-30 Daiichi Seiyaku Co Process for preparing 8-chloroquinolone derivatives
CN1065206A (zh) * 1991-04-01 1992-10-14 战永胜 天然中草药防治早泄、淋病双效药液制法
WO1993025545A1 (en) * 1992-06-09 1993-12-23 Korea Research Institute Of Chemical Technology Novel quinoline derivatives and processes for preparing the same

Also Published As

Publication number Publication date
NO992513L (no) 1995-03-13
FI110777B (fi) 2003-03-31
IL123910A (en) 1999-06-20
SK283189B6 (sk) 2003-03-04
BG99035A (bg) 1995-05-31
SI9400349B (sl) 2000-08-31
IL110909A0 (en) 1994-11-28
TW393481B (en) 2000-06-11
CZ21598A3 (cs) 1999-02-17
DE69418953D1 (de) 1999-07-15
HUT68541A (en) 1995-06-28
NO943313D0 (no) 1994-09-08
CN1106006A (zh) 1995-08-02
AU7286294A (en) 1995-03-23
JP3793583B2 (ja) 2006-07-05
SK283188B6 (sk) 2003-03-04
NO943313L (no) 1995-03-13
HU9402597D0 (en) 1994-11-28
NO307419B1 (no) 2000-04-03
KR100336247B1 (ko) 2005-08-11
CZ284837B6 (cs) 1999-03-17
MY112574A (en) 2001-07-31
NO992513D0 (no) 1999-05-25
JPH07126266A (ja) 1995-05-16
CZ217694A3 (en) 1995-03-15
YU49132B (sh) 2004-03-12
SK107694A3 (en) 1995-05-10
CZ284737B6 (cs) 1999-02-17
EP0643058A1 (en) 1995-03-15
RU94032286A (ru) 1996-08-10
ATE181069T1 (de) 1999-06-15
CA2131761C (en) 2002-04-30
FI944174A (fi) 1995-03-11
US5693814A (en) 1997-12-02
EP0643058B1 (en) 1999-06-09
GR3031012T3 (en) 1999-12-31
NZ264422A (en) 1995-07-26
IL110909A (en) 1998-12-06
KR950008506A (ko) 1995-04-17
FI944174A0 (fi) 1994-09-09
CA2131761A1 (en) 1995-03-11
CZ284738B6 (cs) 1999-02-17
HU224970B1 (en) 2006-04-28
GEP19981355B (en) 1998-08-25
ZA946853B (en) 1995-04-24
SK283190B6 (sk) 2003-03-04
SI9400349A (en) 1995-04-30
HRP940506B1 (en) 2000-10-31
AU679094B2 (en) 1997-06-19
RU2126402C1 (ru) 1999-02-20
SG50492A1 (en) 1998-07-20
PL180163B1 (pl) 2000-12-29
ES2136142T3 (es) 1999-11-16
DK0643058T3 (da) 1999-11-15
HRP940506A2 (en) 1997-04-30
PL304989A1 (en) 1995-03-20
LV11322B (en) 1996-10-20
DE69418953T2 (de) 2000-01-13
CN1057297C (zh) 2000-10-11
NO307753B1 (no) 2000-05-22
CZ21498A3 (cs) 1999-02-17
UA41312C2 (uk) 2001-09-17
LV11322A (lv) 1996-06-20
YU53694A (sh) 1997-03-07

Similar Documents

Publication Publication Date Title
KR100525146B1 (ko) Cdch의신규결정성변형체,그의제조방법및이변형체를함유하는 항균 조성물
KR100245938B1 (ko) 트리아졸릴티오메틸티오 세팔로스포린 염산염, 그의 결정성 수화물 및 이들의 제조방법
RU2125571C1 (ru) СОЛЬ 7-([1α,5α,6α]-6-АМИНО-3-АЗАБИЦИКЛО [3.1.0] ГЕКС-3-ИЛ)-6-ФТОР-1-(2,4-ДИФТОРФЕНИЛ)-1,4- ДИГИДРО-4-ОКСО-1,8-НАФТИРИДИН-3-КАРБОНОВОЙ И МЕТАНСУЛЬФОНОВОЙ КИСЛОТ И СПОСОБ ЕЕ ПОЛУЧЕНИЯ
JPS6145626B2 (sk)
BG61767B1 (bg) Кристали от антимикробно съединение
EP0547646A2 (en) Crystalline form of a cephalosporin antibiotic
EP2946781B1 (en) Crystalline levofolinic acid and process for its preparation
US4607046A (en) 4-(1-imidazolylmethyl)cinnamic acid hydrochloride monohydrate and pharmaceutical compositions
EP0101170B1 (en) Process for the manufacture of sodium cefoperazone
US20030191296A1 (en) Erythromycin derivative having novel crystal structures and processes for their production
US5302588A (en) Crystalline (5R,6S)-2-carbamoyloxymethyl-6-[(1R)-hydroxyethyl]-2-penem-carboxylic acid and its pharmaceutical formulation
WO2002060441A1 (en) Novel forms of 2,3-dimethyl-8-(2-ethyl-6-methylbenzylamino)-imidazo (1,2-a)pyridine-6-carboxamide
AP788A (en) Novel crystal form of anhydrous 7-(1a, 5a, 6a)-6-Amino-3-Azabicyclo(3.1.0) hex-3-YI)-6-Fluoro-1-(2,4- Difluorophenyl)-1,4-Dihydro-4-Oxo-1, 8-Naphthyridine-3-Carboxylic Acid, Methanesulfonic acid salt.
CS209950B2 (en) Method of making the new 4- amino-6,7-dialcoxy-2-piperazinochinazoline derivatives