ITMI20032259A1 - Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione - Google Patents

Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione

Info

Publication number
ITMI20032259A1
ITMI20032259A1 IT002259A ITMI20032259A ITMI20032259A1 IT MI20032259 A1 ITMI20032259 A1 IT MI20032259A1 IT 002259 A IT002259 A IT 002259A IT MI20032259 A ITMI20032259 A IT MI20032259A IT MI20032259 A1 ITMI20032259 A1 IT MI20032259A1
Authority
IT
Italy
Prior art keywords
metossi
carbosxyl
diidro
diazabiclo
chloridrate
Prior art date
Application number
IT002259A
Other languages
English (en)
Inventor
Valentina Aromatario
Pietro Massario
Stefano Turchetta
Original Assignee
Chemi Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemi Spa filed Critical Chemi Spa
Priority to IT002259A priority Critical patent/ITMI20032259A1/it
Priority to US10/580,173 priority patent/US8236817B2/en
Priority to DE602004018370T priority patent/DE602004018370D1/de
Priority to JP2006540424A priority patent/JP4732361B2/ja
Priority to EP04791330A priority patent/EP1685130B1/en
Priority to PCT/EP2004/052699 priority patent/WO2005054240A1/en
Priority to ES04791330T priority patent/ES2319125T3/es
Publication of ITMI20032259A1 publication Critical patent/ITMI20032259A1/it
Priority to US13/538,249 priority patent/US20120277263A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT002259A 2003-11-20 2003-11-20 Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione ITMI20032259A1 (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT002259A ITMI20032259A1 (it) 2003-11-20 2003-11-20 Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
US10/580,173 US8236817B2 (en) 2003-11-20 2004-10-28 Polymorphs of 1-cyclopropy1-7-([s,s])-2,8-diazadicyclo[4.3.0]non-8-yl)-6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
DE602004018370T DE602004018370D1 (de) 2003-11-20 2004-10-28 Polymorphe von 1-cyclopropyl-7-(äs,sü - 2,8-diazadicyclo ä4.3.0ü non-8-yl) -6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäurehydrochlorid und verfahren zu deren herstellung
JP2006540424A JP4732361B2 (ja) 2003-11-20 2004-10-28 塩酸1−シクロプロピル−7−((s,s)−2,8−ジアザジシクロ(4.3.0)ノン−8−イル)−6−フルオロ−1,4−ジヒドロ−8−メトキシ−4−オキソ−3−キノリンカルボン酸の多形およびその調製方法
EP04791330A EP1685130B1 (en) 2003-11-20 2004-10-28 Polymorphs of 1-cyclopropyl-7-([s,s] - 2,8-diazadicyclo [4.3.0] non-8-yl) -6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
PCT/EP2004/052699 WO2005054240A1 (en) 2003-11-20 2004-10-28 Polymorphs of 1-cyclopropyl-7-([s,s]-2,8-diazadicyclo[4.3.0]non-8-yl)-6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
ES04791330T ES2319125T3 (es) 2003-11-20 2004-10-28 Polimorfos del clorhidrato del acido 1-ciclopropil-7-((s,s)-2,8-diazadiciclo(4.3.0)-non-8-il)-6-fluoro-1,4-dihidro-8-metoxi-4-oxo-3-quinolina carboxilico y metodos para la preparacion de los mismos.
US13/538,249 US20120277263A1 (en) 2003-11-20 2012-06-29 Polymorphs of 1-cyclopropyl-7-([s,s])-2,8-diazadicyclo[4.3.0]non-8-yl)-6-fluoro-1,4-dihydro -8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT002259A ITMI20032259A1 (it) 2003-11-20 2003-11-20 Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione

Publications (1)

Publication Number Publication Date
ITMI20032259A1 true ITMI20032259A1 (it) 2005-05-21

Family

ID=43721882

Family Applications (1)

Application Number Title Priority Date Filing Date
IT002259A ITMI20032259A1 (it) 2003-11-20 2003-11-20 Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione

Country Status (3)

Country Link
US (2) US8236817B2 (it)
JP (1) JP4732361B2 (it)
IT (1) ITMI20032259A1 (it)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060264635A1 (en) * 2003-08-05 2006-11-23 Chava Satyanarayana Process for the preparation of moxifloxacin hydrochloride

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
TW209865B (it) 1992-01-10 1993-07-21 Bayer Ag
ZA946853B (en) 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
DE19546249A1 (de) 1995-12-12 1997-06-19 Bayer Ag Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen
DE19751948A1 (de) * 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
KR100817425B1 (ko) * 2000-02-09 2008-03-27 다이이찌 세이야꾸 가부시기가이샤 피리돈카복실산류를 유효성분으로 하는 항항산균제
US6627646B2 (en) * 2001-07-17 2003-09-30 Sepracor Inc. Norastemizole polymorphs
AU2002351255A1 (en) 2001-12-10 2003-06-23 Bristol-Myers Squibb Company Bis hydrochloride monohydrate salt of rsv fusion inhibitor
EP1615645B2 (en) * 2003-04-09 2013-08-21 Dr. Reddy's Laboratories Ltd. A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for the preparation thereof
US20060264635A1 (en) 2003-08-05 2006-11-23 Chava Satyanarayana Process for the preparation of moxifloxacin hydrochloride

Also Published As

Publication number Publication date
US20120277263A1 (en) 2012-11-01
US20070072895A1 (en) 2007-03-29
JP4732361B2 (ja) 2011-07-27
JP2007511580A (ja) 2007-05-10
US8236817B2 (en) 2012-08-07

Similar Documents

Publication Publication Date Title
IS2722B (is) 1, 2, 3, 4- Tetrasetin indól til meðhöndlunar á öndunarfærasjúkdómum
DE602004006169D1 (de) Substituierte 8'-pyri(mi)dinyl-dihydrospiro-äcycloalkylaminü-pyrimidoä1,2aüpyrimidin-6-onderivate
DE60039643D1 (de) Herzfrequenz-Überwachungsgerät
DE60225561D1 (de) Indanessigsäure-derivate und ihre verwendung als pharmazeutische mittel, zwischenprodukten und verfahren zur herstellung
FI20022225A0 (fi) Sykerajan asettaminen sykemittarissa
ITRM20040317A1 (it) Apparecchio per la stimolazione dei muscoli dell'apparato locomotorio.
ITMI20010077A1 (it) Procedimento per la produzione dell'imipenem
PT1603550E (pt) Composição farmacêutica que compreende ácido 5-metil-2-2¿- (cloro-6¿-fluoroanilino)fenilacético
ITMI20032259A1 (it) Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
ITMI20011132A0 (it) Procedimento per la preparazione dell'acido 1-amminometil-1-cicloesanacetico
ITMI20021168A0 (it) Procedimento per la preparazione dell'acido (s)-tetraidro-a-(1-metiletil)-2-osso-1(2h)-piridinacetico
ITMI20020974A1 (it) Procedimento per la preparazione dell'acido 4-fluoro-antranilico
ITMI20032390A1 (it) Metodo per la determinazione dell'attivita' di beta-galattosidasi.
ITFI20030256A1 (it) Dispositivo per l'eliminazione dell'anidride carbonica
FR2843683B1 (fr) Dispositif de collecte, retournement, nettoyage, redistribution de poches d'huitres d'elevage
ITMI20031471A1 (it) Processo per la racemizzazione dell'acido etodolico
ITRM20030440A0 (it) Sistema d'indicazione temporale, in particolare dell'orario.
ITMI20020132A0 (it) Processo per l'ottenimento dell'acido (6s)-5,6,7,8-tetraidrofolico
ITMI20030822A1 (it) Processo per la preparazione dell'acido ursodesossicolico
IT1318703B1 (it) Procedimento per la preparazione dell'acido 13-cis-retinoico.
ITMI20051387A1 (it) Nuovo procedimento per sintetizzare ammidi dell'acido retinoico e nuovo intermedio utilizzato in tale procedimento
DK1173092T3 (da) Pulssensor
ITMI20042402A1 (it) Processo per la preparazione di n,n-dimetil-n'-feniluree
ITNA20030016A1 (it) Sistema alternativo per la raccolta dell'acqua piovana.
ITMI20032068A1 (it) Derivati dell'acido 1-fenilcicloalcancarbossilico per il trattamento delle malattie neurodegenerative.