BG108201A - Производни на n-(арилсулфонил)-бета-аминокиселини, съдържащи заместена аминоетилна група, метод за тяхното получаване и фармацевтични състави, които ги съдържат - Google Patents

Производни на n-(арилсулфонил)-бета-аминокиселини, съдържащи заместена аминоетилна група, метод за тяхното получаване и фармацевтични състави, които ги съдържат Download PDF

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BG108201A
BG108201A BG108201A BG10820103A BG108201A BG 108201 A BG108201 A BG 108201A BG 108201 A BG108201 A BG 108201A BG 10820103 A BG10820103 A BG 10820103A BG 108201 A BG108201 A BG 108201A
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Bulgaria
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compound
group
phenyl
formula
substituted
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BG108201A
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Bulgarian (bg)
English (en)
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Bernard Ferrari
Jean Gougat
Yvette Muneaux
Pierre Perreaut
Lionel Sarran
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Sanofi-Synthelabo
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Publication of BG108201A publication Critical patent/BG108201A/bg

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    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
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    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
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    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
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    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
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    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
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    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D495/04—Ortho-condensed systems
BG108201A 2001-03-28 2003-09-25 Производни на n-(арилсулфонил)-бета-аминокиселини, съдържащи заместена аминоетилна група, метод за тяхното получаване и фармацевтични състави, които ги съдържат BG108201A (bg)

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FR0104315A FR2822827B1 (fr) 2001-03-28 2001-03-28 Nouveaux derives de n-(arylsulfonyl) beta-aminoacides comportant un groupe aminomethyle substitue, leur procede de preparation et les compositions pharmaceutiques en contenant
PCT/FR2002/001059 WO2002076964A1 (fr) 2001-03-28 2002-03-27 Derives de n-(arylsulfonyl)beta-aminoacides comportant un groupe aminomethyle substitue, leur procede de preparation et les compositions pharmaceutiques en contenant

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