BE2024C511I2 - - Google Patents
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- Publication number
- BE2024C511I2 BE2024C511I2 BE2024C511C BE2024C511C BE2024C511I2 BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2 BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2
- Authority
- BE
- Belgium
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2004150979 | 2004-05-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE2024C511I2 true BE2024C511I2 (enEXAMPLES) | 2024-10-08 |
Family
ID=35079161
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE2024C511C BE2024C511I2 (enEXAMPLES) | 2004-05-20 | 2024-03-15 |
Country Status (33)
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
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US6891227B2 (en) | 2002-03-20 | 2005-05-10 | International Business Machines Corporation | Self-aligned nanotube field effect transistor and method of fabricating same |
AU2003302029B8 (en) * | 2002-11-20 | 2006-08-17 | Japan Tobacco Inc. | 4-oxoquinoline compound and utilization thereof as HIV integrase inhibitor |
MY134672A (en) * | 2004-05-20 | 2007-12-31 | Japan Tobacco Inc | Stable crystal of 4-oxoquinoline compound |
WO2007063869A1 (ja) * | 2005-11-30 | 2007-06-07 | Japan Tobacco Inc. | 高純度キノロン化合物の製造方法 |
US20090233964A1 (en) * | 2005-12-30 | 2009-09-17 | Gilead Sciences, Inc. | Methods for improving the pharmacokinetics of hiv integrase inhibitors |
AU2013203476C1 (en) * | 2005-12-30 | 2016-11-17 | Gilead Sciences, Inc. | Methods for improving the pharmacokinetics of hiv integrase inhibitors |
EA201201496A1 (ru) * | 2005-12-30 | 2013-07-30 | Джилид Сайэнс, Инк. | Способ ингибирования интегразы вич, способ улучшения фармакокинетики 6-(3-хлор-2-фторбензил)-1-[(2s)-1-гидрокси-3-метилбутан-2-ил]-7-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновой кислоты (варианты), набор, фармацевтическая композиция (варианты) и антиретровирусный агент (варианты) |
US20090018162A1 (en) * | 2006-02-01 | 2009-01-15 | Yuji Matsuzaki | Use of 6-(3-chloro-2-fluorobenzyl)-1-[(2s)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid or salt thereof for treating retrovirus infection |
WO2007092802A1 (en) * | 2006-02-09 | 2007-08-16 | Boehringer Ingelheim International Gmbh | Method for treating hiv infection through co-administration of tipranavir and gs 9137 |
EA017861B9 (ru) * | 2006-03-06 | 2014-05-30 | Джапан Тобакко Инк. | Способ получения 4-оксохинолинового соединения |
IN2014CN00532A (enEXAMPLES) | 2006-03-06 | 2015-04-03 | Japan Tobacco Inc | |
CN101490023B (zh) | 2006-07-07 | 2013-05-29 | 吉里德科学公司 | 治疗剂的药代动力学特性调节剂 |
EP2644587A3 (en) | 2006-09-12 | 2013-10-23 | Gilead Sciences, Inc. | Process and intermediates for preparing integrase inhibitors |
LT2487162T (lt) * | 2007-02-23 | 2016-11-10 | Gilead Sciences, Inc. | Terapinių agentų farmakokinetinių savybių moduliatoriai |
CA2692101A1 (en) * | 2007-06-29 | 2009-01-08 | Gilead Sciences, Inc. | Combination of 6-(3-chloro-2-fluorobenzyl)-1-[(2s)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid and a compound that inhibits a ugt pathway or ugt metabolism |
MX2009013828A (es) * | 2007-06-29 | 2010-03-10 | Gilead Sciences Inc | Composiciones terapeuticas y su uso. |
AR068403A1 (es) | 2007-09-11 | 2009-11-18 | Gilead Sciences Inc | Proceso e intermediarios para la preparacion de inhibidores de integrasa |
CN102123700A (zh) | 2008-05-02 | 2011-07-13 | 吉里德科学公司 | 固体载体颗粒在改善药物制剂加工性中的应用 |
PT2393485E (pt) | 2009-02-06 | 2015-10-23 | Gilead Sciences Inc | Comprimidos bicamada que compreendem elvitegravir, cobicistat, emtricitabina e tenofovir |
WO2010137032A2 (en) * | 2009-05-14 | 2010-12-02 | Matrix Laboratories Ltd. | Novel polymorphic forms of elvitegravir and its pharmaceutically acceptable salts |
WO2011004389A2 (en) * | 2009-06-18 | 2011-01-13 | Matrix Laboratories Ltd | An improved process for the preparation of elvitegravir |
CN102212032B (zh) * | 2011-04-20 | 2013-07-31 | 复旦大学 | 一种5-羟基喹诺酮类衍生物及其制备方法和用途 |
US10071957B2 (en) | 2012-07-06 | 2018-09-11 | Genentech, Inc. | N-substituted benzamides and methods of use thereof |
CN104520275B (zh) | 2012-08-03 | 2016-11-02 | 吉利德科学公司 | 用于制备整合酶抑制剂的方法和中间产物 |
CN103819402B (zh) * | 2012-11-17 | 2016-03-30 | 上海迪赛诺化学制药有限公司 | 埃替拉韦中间体及其制备方法和应用 |
CN103864682B (zh) * | 2012-12-18 | 2016-12-28 | 上海迪赛诺化学制药有限公司 | 一种制备iii型埃替拉韦晶体的方法 |
SI3067358T1 (sl) | 2012-12-21 | 2019-12-31 | Gilead Sciences, Inc. | Policiklične spojine karbamoilpiridona in njihova farmacevtska uporaba |
NO2865735T3 (enEXAMPLES) | 2013-07-12 | 2018-07-21 | ||
WO2015006731A1 (en) | 2013-07-12 | 2015-01-15 | Gilead Sciences, Inc. | Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections |
CN105315203A (zh) * | 2014-06-06 | 2016-02-10 | 上海迪赛诺化学制药有限公司 | 一种v型埃替拉韦晶体及其制备方法 |
NO2717902T3 (enEXAMPLES) | 2014-06-20 | 2018-06-23 | ||
TW201613936A (en) | 2014-06-20 | 2016-04-16 | Gilead Sciences Inc | Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide |
TWI677489B (zh) | 2014-06-20 | 2019-11-21 | 美商基利科學股份有限公司 | 多環型胺甲醯基吡啶酮化合物之合成 |
TWI738321B (zh) | 2014-12-23 | 2021-09-01 | 美商基利科學股份有限公司 | 多環胺甲醯基吡啶酮化合物及其醫藥用途 |
NZ735575A (en) | 2015-04-02 | 2018-11-30 | Gilead Sciences Inc | Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
CN106008195B (zh) * | 2016-05-19 | 2018-08-03 | 绍兴文理学院 | 一种2,4-二氟-5-碘苯甲酸的制备方法 |
EP3984536B1 (en) * | 2020-10-19 | 2025-06-25 | Centre national de la recherche scientifique | Inhibition of the hiv-1 replication by compounds directed against a new target of the viral cycle |
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JPH0651229B2 (ja) | 1989-07-31 | 1994-07-06 | 新日本製鐵株式会社 | プラズマアーク溶接方法および装置 |
IL100555A (en) | 1991-02-07 | 2000-08-31 | Hoechst Marion Roussel Inc | N-substituted quinoline derivatives their preparation their use for the preparation of medicaments and the pharmaceutical compositions containing them |
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JPH06199835A (ja) | 1993-01-08 | 1994-07-19 | Hokuriku Seiyaku Co Ltd | 8−ジフルオロメトキシキノリン−3−カルボン酸誘導体 |
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JPH0826772A (ja) | 1994-07-22 | 1996-01-30 | Sony Corp | 融着用ガラス、その製造方法及び製造装置、並びに磁気ヘッドの製造方法 |
PT892801E (pt) | 1996-04-12 | 2002-06-28 | Us Gov Health & Human Serv | Compostos derivados de acridona uteis como agentes antineoplasicos e antiretrovirais |
FR2761687B1 (fr) * | 1997-04-08 | 2000-09-15 | Centre Nat Rech Scient | Derives de quinoleines, possedant notamment des proprietes antivirales, leurs preparations et leurs applications biologiques |
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RU2206564C1 (ru) * | 2002-03-07 | 2003-06-20 | Общество с ограниченной ответственностью "Поливит" | Способ получения этилового эфира 6-фтор-7-хлор-1,4-дигидро-4-оксо-3-хинолинкарбоновой кислоты |
JP4035765B2 (ja) | 2002-10-31 | 2008-01-23 | 横河電機株式会社 | フーリエ変換型赤外線分光計 |
JP3567162B1 (ja) | 2002-11-20 | 2004-09-22 | 日本たばこ産業株式会社 | 4−オキソキノリン化合物及びそのhivインテグラーゼ阻害剤としての利用 |
AU2003302029B8 (en) * | 2002-11-20 | 2006-08-17 | Japan Tobacco Inc. | 4-oxoquinoline compound and utilization thereof as HIV integrase inhibitor |
MY134672A (en) * | 2004-05-20 | 2007-12-31 | Japan Tobacco Inc | Stable crystal of 4-oxoquinoline compound |
US7531554B2 (en) * | 2004-05-20 | 2009-05-12 | Japan Tobacco Inc. | 4-oxoquinoline compound and use thereof as HIV integrase inhibitor |
JP4629104B2 (ja) | 2004-05-21 | 2011-02-09 | 日本たばこ産業株式会社 | 4−オキソキノリン誘導体および抗hiv剤を含む併用剤 |
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2005
- 2005-05-18 MY MYPI20052258A patent/MY134672A/en unknown
- 2005-05-19 PT PT05726243T patent/PT1636190E/pt unknown
- 2005-05-19 DK DK05726243.8T patent/DK1636190T3/da active
- 2005-05-19 TW TW094116234A patent/TWI329015B/zh not_active IP Right Cessation
- 2005-05-19 BR BRPI0510114A patent/BRPI0510114B8/pt active IP Right Grant
- 2005-05-19 HR HRP20120681TT patent/HRP20120681T1/hr unknown
- 2005-05-19 CA CA2566922A patent/CA2566922C/en not_active Expired - Lifetime
- 2005-05-19 HR HRP20231588TT patent/HRP20231588T3/hr unknown
- 2005-05-19 HU HUE17186674A patent/HUE064615T2/hu unknown
- 2005-05-19 LT LTEP17186674.2T patent/LT3281939T/lt unknown
- 2005-05-19 CN CN2005800161426A patent/CN1956961B/zh not_active Expired - Lifetime
- 2005-05-19 RU RU2006145302/04A patent/RU2330845C1/ru active
- 2005-05-19 PL PL17186674.2T patent/PL3281939T3/pl unknown
- 2005-05-19 RS RS20120306A patent/RS52375B/en unknown
- 2005-05-19 PT PT171866742T patent/PT3281939T/pt unknown
- 2005-05-19 RS RS20231092A patent/RS64845B1/sr unknown
- 2005-05-19 SI SI200531572T patent/SI1636190T1/sl unknown
- 2005-05-19 KR KR1020087014768A patent/KR20080064909A/ko not_active Withdrawn
- 2005-05-19 WO PCT/JP2005/009604 patent/WO2005113508A1/en active Application Filing
- 2005-05-19 ES ES17186674T patent/ES2960824T3/es not_active Expired - Lifetime
- 2005-05-19 FI FIEP17186674.2T patent/FI3281939T3/fi active
- 2005-05-19 NZ NZ551839A patent/NZ551839A/en not_active IP Right Cessation
- 2005-05-19 AR ARP050102058A patent/AR049280A1/es not_active Application Discontinuation
- 2005-05-19 JP JP2005147219A patent/JP3754064B2/ja not_active Expired - Lifetime
- 2005-05-19 EP EP17186674.2A patent/EP3281939B1/en not_active Expired - Lifetime
- 2005-05-19 EP EP12173572A patent/EP2514746A1/en not_active Withdrawn
- 2005-05-19 SI SI200532315T patent/SI3281939T1/sl unknown
- 2005-05-19 EP EP05726243A patent/EP1636190B1/en not_active Expired - Lifetime
- 2005-05-19 MX MXPA06013405A patent/MXPA06013405A/es active IP Right Grant
- 2005-05-19 ZA ZA200610647A patent/ZA200610647B/en unknown
- 2005-05-19 ES ES05726243T patent/ES2388441T3/es not_active Expired - Lifetime
- 2005-05-19 AU AU2005245296A patent/AU2005245296B2/en active Active
- 2005-05-19 PL PL05726243T patent/PL1636190T3/pl unknown
- 2005-05-19 DK DK17186674.2T patent/DK3281939T3/da active
- 2005-05-19 EP EP23203885.1A patent/EP4299563A3/en active Pending
- 2005-05-20 PE PE2005000561A patent/PE20060358A1/es active IP Right Grant
- 2005-05-20 US US11/133,471 patent/US7635704B2/en active Active
- 2005-05-20 PE PE2011002129A patent/PE20120361A1/es active IP Right Grant
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2006
- 2006-11-14 IL IL179250A patent/IL179250A0/en active IP Right Grant
- 2006-12-14 NO NO20065790A patent/NO339223B1/no unknown
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2009
- 2009-08-10 US US12/538,694 patent/US8981103B2/en active Active
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2012
- 2012-07-11 CY CY20121100621T patent/CY1113010T1/el unknown
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2014
- 2014-04-25 AR ARP140101722A patent/AR096100A2/es active IP Right Grant
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2015
- 2015-01-09 US US14/593,946 patent/US20150361044A1/en not_active Abandoned
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2016
- 2016-08-12 NO NO20161297A patent/NO20161297A1/no not_active Application Discontinuation
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2017
- 2017-03-01 US US15/447,007 patent/US20180029989A1/en not_active Abandoned
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2018
- 2018-07-20 US US16/041,458 patent/US20190185433A1/en not_active Abandoned
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2019
- 2019-01-15 NO NO20190051A patent/NO20190051A1/no not_active Application Discontinuation
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2020
- 2020-08-04 NO NO20200873A patent/NO20200873A1/no not_active Application Discontinuation
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2021
- 2021-08-24 US US17/445,817 patent/US20220235009A1/en not_active Abandoned
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2022
- 2022-06-17 NO NO20220690A patent/NO20220690A1/no not_active Application Discontinuation
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2023
- 2023-08-25 NO NO20230913A patent/NO347902B1/no unknown
- 2023-09-28 CY CY2015009C patent/CY2015009I1/el unknown
- 2023-11-02 FR FR23C1040C patent/FR23C1040I1/fr active Active
- 2023-12-05 CY CY20231100714T patent/CY1126560T1/el unknown
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2024
- 2024-03-14 LU LU00334C patent/LUC00334I2/fr unknown
- 2024-03-15 BE BE2024C511C patent/BE2024C511I2/nl unknown
- 2024-03-19 CY CY2024008C patent/CY2024008I2/el unknown
- 2024-03-20 HU HUS2400006C patent/HUS2400006I1/hu unknown
- 2024-03-20 FI FIC20240008C patent/FIC20240008I1/fi unknown
- 2024-04-12 US US18/634,451 patent/US20250091995A1/en active Pending
- 2024-04-22 NO NO20240384A patent/NO20240384A1/no unknown
- 2024-07-15 NO NO2024034C patent/NO2024034I1/no unknown