BE2024C511I2 - - Google Patents

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Publication number
BE2024C511I2
BE2024C511I2 BE2024C511C BE2024C511C BE2024C511I2 BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2 BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2
Authority
BE
Belgium
Application number
BE2024C511C
Other languages
Dutch (nl)
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079161&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BE2024C511(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of BE2024C511I2 publication Critical patent/BE2024C511I2/nl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE2024C511C 2004-05-20 2024-03-15 BE2024C511I2 (enEXAMPLES)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004150979 2004-05-20

Publications (1)

Publication Number Publication Date
BE2024C511I2 true BE2024C511I2 (enEXAMPLES) 2024-10-08

Family

ID=35079161

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2024C511C BE2024C511I2 (enEXAMPLES) 2004-05-20 2024-03-15

Country Status (33)

Country Link
US (7) US7635704B2 (enEXAMPLES)
EP (4) EP3281939B1 (enEXAMPLES)
JP (1) JP3754064B2 (enEXAMPLES)
KR (1) KR20080064909A (enEXAMPLES)
CN (1) CN1956961B (enEXAMPLES)
AR (2) AR049280A1 (enEXAMPLES)
AU (1) AU2005245296B2 (enEXAMPLES)
BE (1) BE2024C511I2 (enEXAMPLES)
BR (1) BRPI0510114B8 (enEXAMPLES)
CA (1) CA2566922C (enEXAMPLES)
CY (4) CY1113010T1 (enEXAMPLES)
DK (2) DK1636190T3 (enEXAMPLES)
ES (2) ES2960824T3 (enEXAMPLES)
FI (2) FI3281939T3 (enEXAMPLES)
FR (1) FR23C1040I1 (enEXAMPLES)
HR (2) HRP20120681T1 (enEXAMPLES)
HU (2) HUE064615T2 (enEXAMPLES)
IL (1) IL179250A0 (enEXAMPLES)
LT (1) LT3281939T (enEXAMPLES)
LU (1) LUC00334I2 (enEXAMPLES)
MX (1) MXPA06013405A (enEXAMPLES)
MY (1) MY134672A (enEXAMPLES)
NO (8) NO339223B1 (enEXAMPLES)
NZ (1) NZ551839A (enEXAMPLES)
PE (2) PE20060358A1 (enEXAMPLES)
PL (2) PL3281939T3 (enEXAMPLES)
PT (2) PT1636190E (enEXAMPLES)
RS (2) RS52375B (enEXAMPLES)
RU (1) RU2330845C1 (enEXAMPLES)
SI (2) SI1636190T1 (enEXAMPLES)
TW (1) TWI329015B (enEXAMPLES)
WO (1) WO2005113508A1 (enEXAMPLES)
ZA (1) ZA200610647B (enEXAMPLES)

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WO2007063869A1 (ja) * 2005-11-30 2007-06-07 Japan Tobacco Inc. 高純度キノロン化合物の製造方法
US20090233964A1 (en) * 2005-12-30 2009-09-17 Gilead Sciences, Inc. Methods for improving the pharmacokinetics of hiv integrase inhibitors
AU2013203476C1 (en) * 2005-12-30 2016-11-17 Gilead Sciences, Inc. Methods for improving the pharmacokinetics of hiv integrase inhibitors
EA201201496A1 (ru) * 2005-12-30 2013-07-30 Джилид Сайэнс, Инк. Способ ингибирования интегразы вич, способ улучшения фармакокинетики 6-(3-хлор-2-фторбензил)-1-[(2s)-1-гидрокси-3-метилбутан-2-ил]-7-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновой кислоты (варианты), набор, фармацевтическая композиция (варианты) и антиретровирусный агент (варианты)
US20090018162A1 (en) * 2006-02-01 2009-01-15 Yuji Matsuzaki Use of 6-(3-chloro-2-fluorobenzyl)-1-[(2s)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid or salt thereof for treating retrovirus infection
WO2007092802A1 (en) * 2006-02-09 2007-08-16 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and gs 9137
EA017861B9 (ru) * 2006-03-06 2014-05-30 Джапан Тобакко Инк. Способ получения 4-оксохинолинового соединения
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CN101490023B (zh) 2006-07-07 2013-05-29 吉里德科学公司 治疗剂的药代动力学特性调节剂
EP2644587A3 (en) 2006-09-12 2013-10-23 Gilead Sciences, Inc. Process and intermediates for preparing integrase inhibitors
LT2487162T (lt) * 2007-02-23 2016-11-10 Gilead Sciences, Inc. Terapinių agentų farmakokinetinių savybių moduliatoriai
CA2692101A1 (en) * 2007-06-29 2009-01-08 Gilead Sciences, Inc. Combination of 6-(3-chloro-2-fluorobenzyl)-1-[(2s)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid and a compound that inhibits a ugt pathway or ugt metabolism
MX2009013828A (es) * 2007-06-29 2010-03-10 Gilead Sciences Inc Composiciones terapeuticas y su uso.
AR068403A1 (es) 2007-09-11 2009-11-18 Gilead Sciences Inc Proceso e intermediarios para la preparacion de inhibidores de integrasa
CN102123700A (zh) 2008-05-02 2011-07-13 吉里德科学公司 固体载体颗粒在改善药物制剂加工性中的应用
PT2393485E (pt) 2009-02-06 2015-10-23 Gilead Sciences Inc Comprimidos bicamada que compreendem elvitegravir, cobicistat, emtricitabina e tenofovir
WO2010137032A2 (en) * 2009-05-14 2010-12-02 Matrix Laboratories Ltd. Novel polymorphic forms of elvitegravir and its pharmaceutically acceptable salts
WO2011004389A2 (en) * 2009-06-18 2011-01-13 Matrix Laboratories Ltd An improved process for the preparation of elvitegravir
CN102212032B (zh) * 2011-04-20 2013-07-31 复旦大学 一种5-羟基喹诺酮类衍生物及其制备方法和用途
US10071957B2 (en) 2012-07-06 2018-09-11 Genentech, Inc. N-substituted benzamides and methods of use thereof
CN104520275B (zh) 2012-08-03 2016-11-02 吉利德科学公司 用于制备整合酶抑制剂的方法和中间产物
CN103819402B (zh) * 2012-11-17 2016-03-30 上海迪赛诺化学制药有限公司 埃替拉韦中间体及其制备方法和应用
CN103864682B (zh) * 2012-12-18 2016-12-28 上海迪赛诺化学制药有限公司 一种制备iii型埃替拉韦晶体的方法
SI3067358T1 (sl) 2012-12-21 2019-12-31 Gilead Sciences, Inc. Policiklične spojine karbamoilpiridona in njihova farmacevtska uporaba
NO2865735T3 (enEXAMPLES) 2013-07-12 2018-07-21
WO2015006731A1 (en) 2013-07-12 2015-01-15 Gilead Sciences, Inc. Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections
CN105315203A (zh) * 2014-06-06 2016-02-10 上海迪赛诺化学制药有限公司 一种v型埃替拉韦晶体及其制备方法
NO2717902T3 (enEXAMPLES) 2014-06-20 2018-06-23
TW201613936A (en) 2014-06-20 2016-04-16 Gilead Sciences Inc Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
TWI677489B (zh) 2014-06-20 2019-11-21 美商基利科學股份有限公司 多環型胺甲醯基吡啶酮化合物之合成
TWI738321B (zh) 2014-12-23 2021-09-01 美商基利科學股份有限公司 多環胺甲醯基吡啶酮化合物及其醫藥用途
NZ735575A (en) 2015-04-02 2018-11-30 Gilead Sciences Inc Polycyclic-carbamoylpyridone compounds and their pharmaceutical use
CN106008195B (zh) * 2016-05-19 2018-08-03 绍兴文理学院 一种2,4-二氟-5-碘苯甲酸的制备方法
EP3984536B1 (en) * 2020-10-19 2025-06-25 Centre national de la recherche scientifique Inhibition of the hiv-1 replication by compounds directed against a new target of the viral cycle

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Also Published As

Publication number Publication date
NO20190051A1 (no) 2007-02-07
WO2005113508A1 (en) 2005-12-01
IL179250A0 (en) 2007-03-08
JP2006001927A (ja) 2006-01-05
US20100204271A1 (en) 2010-08-12
PL1636190T3 (pl) 2012-10-31
SI1636190T1 (sl) 2012-09-28
HUS2400006I1 (hu) 2024-04-28
EP4299563A3 (en) 2024-02-28
EP1636190B1 (en) 2012-06-27
NO20161297A1 (no) 2007-02-07
EP4299563A2 (en) 2024-01-03
PE20060358A1 (es) 2006-05-12
CN1956961A (zh) 2007-05-02
US8981103B2 (en) 2015-03-17
MY134672A (en) 2007-12-31
HRP20231588T3 (hr) 2024-03-15
RU2330845C1 (ru) 2008-08-10
FIC20240008I1 (fi) 2024-03-20
EP3281939A1 (en) 2018-02-14
NO2024034I1 (no) 2024-07-15
CY2015009I2 (el) 2024-09-20
LT3281939T (lt) 2023-11-27
ES2388441T3 (es) 2012-10-15
EP3281939B1 (en) 2023-10-18
CY2024008I1 (el) 2024-09-20
CA2566922A1 (en) 2005-12-01
US20190185433A1 (en) 2019-06-20
US20180029989A1 (en) 2018-02-01
BRPI0510114A (pt) 2007-09-25
KR20080064909A (ko) 2008-07-09
CY1113010T1 (el) 2016-04-13
HUE064615T2 (hu) 2024-04-28
NO20230913A1 (no) 2007-02-07
TW200600097A (en) 2006-01-01
RS52375B (en) 2012-12-31
BRPI0510114B8 (pt) 2021-05-25
AR049280A1 (es) 2006-07-12
PT1636190E (pt) 2012-08-20
DK1636190T3 (da) 2012-09-24
AU2005245296B2 (en) 2010-08-12
AU2005245296A1 (en) 2005-12-01
NZ551839A (en) 2009-11-27
ES2960824T3 (es) 2024-03-06
CY1126560T1 (el) 2024-09-20
CY2024008I2 (el) 2024-09-20
AR096100A2 (es) 2015-12-09
NO20220690A1 (no) 2007-02-07
NO339223B1 (no) 2016-11-21
US20060030710A1 (en) 2006-02-09
NO347902B1 (no) 2024-05-06
PE20120361A1 (es) 2012-05-03
NO20200873A1 (no) 2007-02-07
EP1636190A1 (en) 2006-03-22
PT3281939T (pt) 2023-11-22
CN1956961B (zh) 2010-05-26
NO20065790L (no) 2007-02-07
FI3281939T3 (fi) 2023-10-23
HRP20120681T1 (hr) 2012-09-30
RS64845B1 (sr) 2023-12-29
PL3281939T3 (pl) 2024-03-18
US20250091995A1 (en) 2025-03-20
TWI329015B (en) 2010-08-21
MXPA06013405A (es) 2007-03-01
FR23C1040I1 (fr) 2023-12-29
CY2015009I1 (el) 2024-09-20
JP3754064B2 (ja) 2006-03-08
ZA200610647B (en) 2008-06-25
US7635704B2 (en) 2009-12-22
NO20240384A1 (no) 2007-02-07
EP2514746A1 (en) 2012-10-24
CA2566922C (en) 2011-01-11
US20150361044A1 (en) 2015-12-17
BRPI0510114B1 (pt) 2020-09-15
DK3281939T3 (da) 2024-01-22
US20220235009A1 (en) 2022-07-28
SI3281939T1 (sl) 2024-02-29
HK1083341A1 (en) 2006-06-30
LUC00334I2 (enEXAMPLES) 2024-07-01

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