AU2015216705B2 - Pyrazolyl-ureas as kinase inhibitors - Google Patents

Pyrazolyl-ureas as kinase inhibitors Download PDF

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Publication number
AU2015216705B2
AU2015216705B2 AU2015216705A AU2015216705A AU2015216705B2 AU 2015216705 B2 AU2015216705 B2 AU 2015216705B2 AU 2015216705 A AU2015216705 A AU 2015216705A AU 2015216705 A AU2015216705 A AU 2015216705A AU 2015216705 B2 AU2015216705 B2 AU 2015216705B2
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butyl
naphthalen
pyrazol
pyridin
amino
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AU2015216705A1 (en
Inventor
Euan Alexander Fraser Fordyce
John King-Underwood
Alistair Ian Longshaw
Stuart Thomas Onions
Jennifer Diane Venable
Iain Walters
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Respivert Ltd
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Respivert Ltd
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    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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AU2015216705A 2014-02-14 2015-02-13 Pyrazolyl-ureas as kinase inhibitors Active AU2015216705B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201461940282P 2014-02-14 2014-02-14
US61/940,282 2014-02-14
US201461941064P 2014-02-18 2014-02-18
US61/941,064 2014-02-18
PCT/GB2015/050401 WO2015121660A1 (en) 2014-02-14 2015-02-13 Pyrazolyl-ureas as kinase inhibitors

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AU2015216705A1 AU2015216705A1 (en) 2016-08-18
AU2015216705B2 true AU2015216705B2 (en) 2019-03-28

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AU2015216705A Active AU2015216705B2 (en) 2014-02-14 2015-02-13 Pyrazolyl-ureas as kinase inhibitors
AU2015216957A Active AU2015216957B2 (en) 2014-02-14 2015-02-13 Aromatic heterocyclic compounds as antiinflammatory compounds
AU2019204525A Active AU2019204525B2 (en) 2014-02-14 2019-06-26 Aromatic heterocyclic compounds as antiinflammatory compounds

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AU2019204525A Active AU2019204525B2 (en) 2014-02-14 2019-06-26 Aromatic heterocyclic compounds as antiinflammatory compounds

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US (8) US9447076B2 (enExample)
EP (4) EP3105223B1 (enExample)
JP (4) JP6586098B2 (enExample)
KR (1) KR102413704B1 (enExample)
CN (4) CN106164067B (enExample)
AU (3) AU2015216705B2 (enExample)
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WO2009077766A1 (en) 2007-12-19 2009-06-25 Cancer Research Technology Limited Pyrido[2,3-b]pyrazine-8-substituted compounds and their use
JP5760010B2 (ja) 2010-02-01 2015-08-05 キャンサー・リサーチ・テクノロジー・リミテッド 1−(5−tert−ブチル−2−フェニル−2H−ピラゾール−3−イル)−3−[2−フルオロ−4−(1−メチル−2−オキソ−2,3−ジヒドロ−1H−イミダゾ[4,5−B]ピリジン−7−イルオキシ)−フェニル]−尿素および関連化合物ならびに治療におけるそれらの使用
KR102057058B1 (ko) 2011-10-03 2019-12-18 레스피버트 리미티드 P38 map 키나제 저해제인 1-피라졸릴-3-(4-((2-아닐리노피리미딘-4-일)옥시)나프탈렌-1-일) 우레아
EP2578582A1 (en) 2011-10-03 2013-04-10 Respivert Limited 1-Pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl)oxy)napththalen-1-yl)ureas as p38 MAP kinase inhibitors
GB201214750D0 (en) 2012-08-17 2012-10-03 Respivert Ltd Compounds
US20150225373A1 (en) 2012-08-29 2015-08-13 Respivert Limited Kinase inhibitors
US9783556B2 (en) 2012-08-29 2017-10-10 Respivert Limited Kinase inhibitors
US20150210722A1 (en) 2012-08-29 2015-07-30 Respivert Limited Kinase inhibitors
EP2925742B1 (en) 2012-11-16 2016-10-26 Respivert Limited Kinase inhibitors
US20160016934A1 (en) 2013-03-14 2016-01-21 Respivert Limited Kinase inhibitors
TWI641592B (zh) 2013-04-02 2018-11-21 英商瑞斯比維特有限公司 激酶抑制劑
US9771353B2 (en) 2013-04-02 2017-09-26 Topivert Pharma Limited Kinase inhibitors based upon N-alkyl pyrazoles
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