TR201809072T4 - Antiinflamatuvar bileşikler olarak aromatik heterosiklik bileşikler. - Google Patents

Antiinflamatuvar bileşikler olarak aromatik heterosiklik bileşikler. Download PDF

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Publication number
TR201809072T4
TR201809072T4 TR2018/09072T TR201809072T TR201809072T4 TR 201809072 T4 TR201809072 T4 TR 201809072T4 TR 2018/09072 T TR2018/09072 T TR 2018/09072T TR 201809072 T TR201809072 T TR 201809072T TR 201809072 T4 TR201809072 T4 TR 201809072T4
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Prior art keywords
compound
formula
compounds
cells
mixture
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TR2018/09072T
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English (en)
Turkish (tr)
Inventor
Alistair Longshaw Ian
Alexander Euan Fordyce Fraser
Stuart Onions Thomas
King-Underwood John
Jennifer Venable Diane
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Respivert Ltd
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Publication of TR201809072T4 publication Critical patent/TR201809072T4/tr

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    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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TR2018/09072T 2014-02-14 2015-02-13 Antiinflamatuvar bileşikler olarak aromatik heterosiklik bileşikler. TR201809072T4 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201461940282P 2014-02-14 2014-02-14
US201461941064P 2014-02-18 2014-02-18

Publications (1)

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TR201809072T4 true TR201809072T4 (tr) 2018-07-23

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TR2018/09072T TR201809072T4 (tr) 2014-02-14 2015-02-13 Antiinflamatuvar bileşikler olarak aromatik heterosiklik bileşikler.

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US (8) US9447076B2 (enExample)
EP (4) EP3105223B1 (enExample)
JP (4) JP6586098B2 (enExample)
KR (1) KR102413704B1 (enExample)
CN (4) CN110522731B (enExample)
AU (3) AU2015216957B2 (enExample)
BR (1) BR112016015838B1 (enExample)
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PL (2) PL3357919T3 (enExample)
PT (2) PT3357919T (enExample)
SG (1) SG11201607058PA (enExample)
TR (1) TR201809072T4 (enExample)
TW (2) TWI664967B (enExample)
UY (1) UY35998A (enExample)
WO (2) WO2015121444A1 (enExample)

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CN102906090B (zh) 2010-02-01 2015-06-24 癌症研究技术有限公司 1-(5-叔丁基-2-苯基-2h-吡唑-3-基)-3-[2-氟-4-(1-甲基-2-氧代-2,3-二氢-1h-咪唑并[4,5-b]吡啶-7-基氧基)-苯基]-脲和相关化合物及它们在治疗中的应用
EP2578582A1 (en) 2011-10-03 2013-04-10 Respivert Limited 1-Pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl)oxy)napththalen-1-yl)ureas as p38 MAP kinase inhibitors
PT2763984T (pt) 2011-10-03 2016-07-25 Respivert Ltd 1-pirazolil-3-(4-((2-anilinopirimidin-4-il)oxi)naftalen-1-il) ureias como inibidores da map cinase p38
GB201214750D0 (en) 2012-08-17 2012-10-03 Respivert Ltd Compounds
WO2014033447A2 (en) 2012-08-29 2014-03-06 Respivert Limited Kinase inhibitors
US20150210722A1 (en) 2012-08-29 2015-07-30 Respivert Limited Kinase inhibitors
WO2014033449A1 (en) 2012-08-29 2014-03-06 Respivert Limited Kinase inhibitors
US9732063B2 (en) 2012-11-16 2017-08-15 Respivert Limited Kinase inhibitors
US20160016934A1 (en) 2013-03-14 2016-01-21 Respivert Limited Kinase inhibitors
EP2981534B1 (en) 2013-04-02 2017-07-19 Topivert Pharma Limited Kinase inhibitors based upon n-alkyl pyrazoles
KR102283883B1 (ko) 2013-04-02 2021-07-29 옥슬러 액퀴지션즈 리미티드 키나제 저해제
GB201320729D0 (en) 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Therapeutic compounds and their use
GB201320732D0 (en) 2013-11-25 2014-01-08 Cancer Rec Tech Ltd Methods of chemical synthesis
CA2934199A1 (en) 2013-12-20 2015-06-25 Respivert Limited Urea derivatives useful as kinase inhibitors
US9447076B2 (en) 2014-02-14 2016-09-20 Respivert Ltd. Inhibitor of p38 map kinase
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