AU2010260058B2 - GIP receptor-active glucagon compounds - Google Patents

GIP receptor-active glucagon compounds Download PDF

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Publication number
AU2010260058B2
AU2010260058B2 AU2010260058A AU2010260058A AU2010260058B2 AU 2010260058 B2 AU2010260058 B2 AU 2010260058B2 AU 2010260058 A AU2010260058 A AU 2010260058A AU 2010260058 A AU2010260058 A AU 2010260058A AU 2010260058 B2 AU2010260058 B2 AU 2010260058B2
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AU
Australia
Prior art keywords
amino acid
glucagon
seq
peptide
analog
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Ceased
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AU2010260058A
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AU2010260058A1 (en
Inventor
Joseph Chabenne
Jonathan Day
Maria Dimarchi
Richard D. Dimarchi
Tao MA
James Patterson
David L. Smiley
Brian P. Ward
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Indiana University Research and Technology Corp
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Indiana University Research and Technology Corp
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Publication of AU2010260058A1 publication Critical patent/AU2010260058A1/en
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Publication of AU2010260058B2 publication Critical patent/AU2010260058B2/en
Ceased legal-status Critical Current
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
AU2010260058A 2009-06-16 2010-06-16 GIP receptor-active glucagon compounds Ceased AU2010260058B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18757809P 2009-06-16 2009-06-16
US61/187,578 2009-06-16
PCT/US2010/038825 WO2010148089A1 (en) 2009-06-16 2010-06-16 Gip receptor-active glucagon compounds

Publications (2)

Publication Number Publication Date
AU2010260058A1 AU2010260058A1 (en) 2012-02-02
AU2010260058B2 true AU2010260058B2 (en) 2015-09-24

Family

ID=43356738

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2010260058A Ceased AU2010260058B2 (en) 2009-06-16 2010-06-16 GIP receptor-active glucagon compounds

Country Status (17)

Country Link
US (2) US9150632B2 (forum.php)
EP (1) EP2443146B1 (forum.php)
JP (1) JP5887265B2 (forum.php)
KR (1) KR20120087875A (forum.php)
CN (1) CN102459325B (forum.php)
AU (1) AU2010260058B2 (forum.php)
BR (1) BRPI1014508A2 (forum.php)
CA (1) CA2765026A1 (forum.php)
CL (1) CL2011003173A1 (forum.php)
IL (1) IL216881A (forum.php)
IN (1) IN2012DN00377A (forum.php)
MX (1) MX2011013625A (forum.php)
PE (1) PE20120914A1 (forum.php)
RU (1) RU2012101274A (forum.php)
SG (1) SG176858A1 (forum.php)
TW (1) TWI549687B (forum.php)
WO (1) WO2010148089A1 (forum.php)

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* Cited by examiner, † Cited by third party
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