AU2003268064A1 - Oxadiazoles as modulators of metabotropic glutamate receptor-5 - Google Patents

Oxadiazoles as modulators of metabotropic glutamate receptor-5 Download PDF

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Publication number
AU2003268064A1
AU2003268064A1 AU2003268064A AU2003268064A AU2003268064A1 AU 2003268064 A1 AU2003268064 A1 AU 2003268064A1 AU 2003268064 A AU2003268064 A AU 2003268064A AU 2003268064 A AU2003268064 A AU 2003268064A AU 2003268064 A1 AU2003268064 A1 AU 2003268064A1
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Australia
Prior art keywords
piperazine
phenyl
alkyl
carboxylic acid
methyl
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Abandoned
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AU2003268064A
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English (en)
Inventor
Louise Edwards
Methvin Isaac
Annika Kers
Johan Malmberg
Donald A. Mcleod
Karin Oscarsson
Abdelmalik Slassi
Thomas M. Stormann
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AstraZeneca AB
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AstraZeneca AB
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Publication of AU2003268064A1 publication Critical patent/AU2003268064A1/en
Assigned to ASTRAZENECA AB reassignment ASTRAZENECA AB Request for Assignment Assignors: ASTRAZENECA AB, NPS PHARMACEUTICALS, INC.
Abandoned legal-status Critical Current

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    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
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    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
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    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
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  • Organic Chemistry (AREA)
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  • Neurosurgery (AREA)
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  • Diabetes (AREA)
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  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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AU2003268064A 2002-08-09 2003-08-08 Oxadiazoles as modulators of metabotropic glutamate receptor-5 Abandoned AU2003268064A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40203902P 2002-08-09 2002-08-09
US60/402,039 2002-08-09
PCT/US2003/024912 WO2004014370A2 (en) 2002-08-09 2003-08-08 Oxadiazoles as modulators of metabotropic glutamate receptor-5

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AU2003268064A1 true AU2003268064A1 (en) 2004-02-25

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AU2003268064A Abandoned AU2003268064A1 (en) 2002-08-09 2003-08-08 Oxadiazoles as modulators of metabotropic glutamate receptor-5

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US (2) US20040132726A1 (enExample)
EP (1) EP1536790A2 (enExample)
JP (1) JP2006506340A (enExample)
KR (1) KR20050039846A (enExample)
CN (1) CN1691944A (enExample)
AR (1) AR041508A1 (enExample)
AU (1) AU2003268064A1 (enExample)
BR (1) BR0313266A (enExample)
CA (1) CA2495120A1 (enExample)
IL (1) IL166650A0 (enExample)
MX (1) MXPA05001592A (enExample)
NO (1) NO20051223L (enExample)
NZ (1) NZ538339A (enExample)
TW (2) TW200424183A (enExample)
WO (1) WO2004014370A2 (enExample)
ZA (1) ZA200501101B (enExample)

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