AU2002312933B2 - CDK inhibiting pyrimidines, production thereof and their use as medicaments - Google Patents

CDK inhibiting pyrimidines, production thereof and their use as medicaments Download PDF

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Publication number
AU2002312933B2
AU2002312933B2 AU2002312933A AU2002312933A AU2002312933B2 AU 2002312933 B2 AU2002312933 B2 AU 2002312933B2 AU 2002312933 A AU2002312933 A AU 2002312933A AU 2002312933 A AU2002312933 A AU 2002312933A AU 2002312933 B2 AU2002312933 B2 AU 2002312933B2
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Australia
Prior art keywords
pyrimidin
bromo
ylamino
methyl
benzenesulfonamide
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2002312933A
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English (en)
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AU2002312933A1 (en
Inventor
Thomas Brumby
Christoph Huwe
Rolf Jautelat
Ulrich Lucking
Olaf Prien
Martina Schafer
Gerhard Siemeister
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Bayer Pharma AG
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Schering AG
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Publication date
Priority claimed from DE10127581A external-priority patent/DE10127581A1/de
Priority claimed from DE10212098A external-priority patent/DE10212098A1/de
Application filed by Schering AG filed Critical Schering AG
Publication of AU2002312933A1 publication Critical patent/AU2002312933A1/en
Application granted granted Critical
Publication of AU2002312933B2 publication Critical patent/AU2002312933B2/en
Anticipated expiration legal-status Critical
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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AU2002312933A 2001-05-29 2002-05-23 CDK inhibiting pyrimidines, production thereof and their use as medicaments Ceased AU2002312933B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DEDE10127581.1 2001-05-29
DE10127581A DE10127581A1 (de) 2001-05-29 2001-05-29 CDK inhibitorische Pyrimidine, deren Herstellung und Verwendung als Arzneimittel
DEDE10212098.6 2002-03-11
DE10212098A DE10212098A1 (de) 2002-03-11 2002-03-11 CDK inhibitorische Pyrimidine, deren Herstellung und Verwendung als Arzneimittel
PCT/EP2002/005669 WO2002096888A1 (de) 2001-05-29 2002-05-23 Cdk inhibitorische pyrimidine, deren herstellung und verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
AU2002312933A1 AU2002312933A1 (en) 2003-05-08
AU2002312933B2 true AU2002312933B2 (en) 2007-12-06

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AU2002312933A Ceased AU2002312933B2 (en) 2001-05-29 2002-05-23 CDK inhibiting pyrimidines, production thereof and their use as medicaments

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EP (1) EP1392662B1 (enExample)
JP (1) JP4291135B2 (enExample)
KR (1) KR100874791B1 (enExample)
CN (1) CN100480242C (enExample)
AR (1) AR036035A1 (enExample)
AT (1) ATE420077T1 (enExample)
AU (1) AU2002312933B2 (enExample)
BR (1) BR0209774A (enExample)
CA (1) CA2449118A1 (enExample)
CO (1) CO5540316A2 (enExample)
DE (1) DE50213202D1 (enExample)
ES (1) ES2320204T3 (enExample)
HR (1) HRP20031081A2 (enExample)
IL (1) IL159120A0 (enExample)
ME (1) MEP13408A (enExample)
MX (1) MXPA03010810A (enExample)
NO (1) NO327129B1 (enExample)
NZ (1) NZ529654A (enExample)
PL (1) PL367130A1 (enExample)
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Families Citing this family (137)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1392662B1 (de) * 2001-05-29 2009-01-07 Bayer Schering Pharma Aktiengesellschaft Cdk inhibitorische pyrimidine, deren herstellung und verwendung als arzneimittel
EP1406875B1 (en) 2001-06-26 2013-07-31 Bristol-Myers Squibb Company N-heterocyclic inhibitors of tnf-alpha expression
DE50212771D1 (de) * 2001-10-17 2008-10-23 Boehringer Ingelheim Pharma Pyrimidinderivate, arzneimittel enthaltend diese verbindungen, deren verwendung und verfahren zu ihrer herstellung
WO2003032994A2 (de) * 2001-10-17 2003-04-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg 5-substituierte 4-amino-2-phenylamino-pyrimidinderivate und ihre verwendung als beta-amyloid modulatoren
AU2002367172A1 (en) * 2001-12-21 2003-07-15 Bayer Pharmaceuticals Corporation 2,4-diamino-pyrimidine derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
GB0205693D0 (en) 2002-03-09 2002-04-24 Astrazeneca Ab Chemical compounds
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