ATE112172T1 - Targetformer von antitumor-methyltrithioagenzien. - Google Patents

Targetformer von antitumor-methyltrithioagenzien.

Info

Publication number
ATE112172T1
ATE112172T1 AT88116338T AT88116338T ATE112172T1 AT E112172 T1 ATE112172 T1 AT E112172T1 AT 88116338 T AT88116338 T AT 88116338T AT 88116338 T AT88116338 T AT 88116338T AT E112172 T1 ATE112172 T1 AT E112172T1
Authority
AT
Austria
Prior art keywords
targetformers
methyltrithioagents
antitumoric
antitumoric methyltrithioagents
Prior art date
Application number
AT88116338T
Other languages
English (en)
Inventor
William James Mcgahren
Martin Leon Sassiver
George A Ellestad
Philip R Hamann
Lois M Hinman
Janis Upeslacis
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Application granted granted Critical
Publication of ATE112172T1 publication Critical patent/ATE112172T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/68Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an antibody, an immunoglobulin or a fragment thereof, e.g. an Fc-fragment
    • A61K47/6801Drug-antibody or immunoglobulin conjugates defined by the pharmacologically or therapeutically active agent
    • A61K47/6803Drugs conjugated to an antibody or immunoglobulin, e.g. cisplatin-antibody conjugates
    • A61K47/6807Drugs conjugated to an antibody or immunoglobulin, e.g. cisplatin-antibody conjugates the drug or compound being a sugar, nucleoside, nucleotide, nucleic acid, e.g. RNA antisense
    • A61K47/6809Antibiotics, e.g. antitumor antibiotics anthracyclins, adriamycin, doxorubicin or daunomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT88116338T 1987-10-30 1988-10-03 Targetformer von antitumor-methyltrithioagenzien. ATE112172T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11494087A 1987-10-30 1987-10-30

Publications (1)

Publication Number Publication Date
ATE112172T1 true ATE112172T1 (de) 1994-10-15

Family

ID=22358378

Family Applications (2)

Application Number Title Priority Date Filing Date
AT88116338T ATE112172T1 (de) 1987-10-30 1988-10-03 Targetformer von antitumor-methyltrithioagenzien.
AT88116339T ATE104309T1 (de) 1987-10-30 1988-10-03 Dischwefel-analoge von ll-e33288 antitumorverbindungen.

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT88116339T ATE104309T1 (de) 1987-10-30 1988-10-03 Dischwefel-analoge von ll-e33288 antitumorverbindungen.

Country Status (19)

Country Link
EP (2) EP0313873B1 (de)
JP (2) JP2720933B2 (de)
KR (2) KR0133130B1 (de)
AR (1) AR246083A1 (de)
AT (2) ATE112172T1 (de)
AU (2) AU618763B2 (de)
BR (1) BR1100939A (de)
CA (1) CA1321582C (de)
DE (2) DE3851682T2 (de)
DK (2) DK174739B1 (de)
ES (2) ES2061586T3 (de)
FI (2) FI91262C (de)
HK (2) HK131897A (de)
IE (2) IE65989B1 (de)
IL (2) IL87946A (de)
NO (2) NO176480C (de)
NZ (2) NZ226727A (de)
PT (2) PT88881B (de)
ZA (2) ZA888123B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5079233A (en) * 1987-01-30 1992-01-07 American Cyanamid Company N-acyl derivatives of the LL-E33288 antitumor antibiotics, composition and methods for using the same
US5606040A (en) * 1987-10-30 1997-02-25 American Cyanamid Company Antitumor and antibacterial substituted disulfide derivatives prepared from compounds possessing a methyl-trithio group
IL115770A (en) * 1989-04-14 1999-03-12 American Cyanamid Co Substituted disulfides of formula q-sp-ss-w their preparation and use for inhibiting the growth of tumours and for treating bacterial infections
GB9007384D0 (en) * 1990-04-02 1990-05-30 Duncan Ruth Coupling between polymers and other organic molecular entities utilising thiol-specific reactive groups
US5714586A (en) * 1995-06-07 1998-02-03 American Cyanamid Company Methods for the preparation of monomeric calicheamicin derivative/carrier conjugates
US5712374A (en) * 1995-06-07 1998-01-27 American Cyanamid Company Method for the preparation of substantiallly monomeric calicheamicin derivative/carrier conjugates
US6395511B1 (en) 1998-11-27 2002-05-28 Darwin Discovery, Ltd. Nucleic acids encoding a novel family of TGF-β binding proteins from humans
US20040009535A1 (en) 1998-11-27 2004-01-15 Celltech R&D, Inc. Compositions and methods for increasing bone mineralization
NZ511705A (en) * 2001-05-14 2004-03-26 Horticulture & Food Res Inst Methods and rapid immunoassay device for detecting progesterone and other steroids
EP1636270B1 (de) 2003-06-16 2016-07-20 UCB Pharma S.A. Spezifische antikörper für sclerostin und verfahren zur erhöhung der knochenmineralisierung
WO2008028050A2 (en) * 2006-08-30 2008-03-06 Wisconsin Alumni Research Foundation Reversible natural product glycosyltransferase-catalyzed reactions, compounds and related methods
KR100979928B1 (ko) * 2008-07-16 2010-09-03 한주학 수직축형 부력풍차
US9902691B2 (en) * 2013-11-04 2018-02-27 Pfizer Inc. Intermediates and methods for synthesizing calicheamicin derivatives
KR20190111086A (ko) * 2017-01-24 2019-10-01 화이자 인코포레이티드 칼리키아마이신 유도체 및 이의 항체 약물 접합체
WO2020168298A2 (en) * 2019-02-15 2020-08-20 University Of Southern California Lym-1 and lym-2 antibody compositions and improved car constructs
JP7750853B2 (ja) * 2020-10-22 2025-10-07 富士フイルム株式会社 皮膚感作性測定試薬、化合物、及び皮膚感作性の測定方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2430943A1 (fr) * 1978-07-13 1980-02-08 Toyo Jozo Kk Nouveaux derives disulfures
DE3175151D1 (en) * 1980-05-21 1986-09-25 Teijin Ltd Reactive polymer and process for the preparation thereof
US4530835A (en) * 1983-07-08 1985-07-23 Warner-Lambert Company CL-1577 Antibiotic compounds and their production
CA1314245C (en) * 1984-05-23 1993-03-09 Franz Jansen Process for the preparation of conjugates in which a monovalent carboxylic ionophore is associated by means of a covalent bond with a macromolecule, which are useful as immunotoxin potentiators
EP0182152B1 (de) * 1984-11-16 1999-05-26 American Cyanamid Company Antitumorale Antibiotika (Komplex LL-E-33288)
EP0330874A3 (de) * 1988-02-29 1989-10-18 American Cyanamid Company Antibakterielle und Antitumor-Mittel LL-E33288 epsilon-I und LL-E33288-epsilon-Br, deren Herstellungen und Zwischenprodukte
EP0342341A3 (de) * 1988-05-17 1991-07-24 American Cyanamid Company Verfahren zur Herstellung von Antitumor-Antibiotika LL-E33288 Gamma 2

Also Published As

Publication number Publication date
IL87947A0 (en) 1989-03-31
EP0313874B1 (de) 1994-04-13
FI884984A0 (fi) 1988-10-28
FI95204C (fi) 1996-01-10
NZ226726A (en) 1991-08-27
FI884983L (fi) 1989-05-01
NO176480B (no) 1995-01-02
CA1321582C (en) 1993-08-24
NO884834D0 (no) 1988-10-28
EP0313873A1 (de) 1989-05-03
BR1100939A (pt) 1999-08-31
KR890006245A (ko) 1989-06-12
NO176480C (no) 1995-04-12
DE3851682D1 (de) 1994-11-03
KR970011385B1 (ko) 1997-07-10
DK602488A (da) 1989-05-01
FI95204B (fi) 1995-09-29
AU2449488A (en) 1989-05-04
AU2448988A (en) 1989-05-04
FI91262B (fi) 1994-02-28
ZA888127B (en) 1989-07-26
PT88882B (pt) 1993-01-29
JP2820256B2 (ja) 1998-11-05
DE3889063T2 (de) 1994-12-01
KR890006244A (ko) 1989-06-12
IE883262L (en) 1989-04-30
AU612714B2 (en) 1991-07-18
JPH0296599A (ja) 1990-04-09
DK602588D0 (da) 1988-10-28
NO884834L (no) 1989-05-02
EP0313874A2 (de) 1989-05-03
NZ226727A (en) 1991-12-23
IE883261L (en) 1989-04-30
KR0133130B1 (ko) 1998-04-17
HK131897A (en) 1997-10-03
FI884984A7 (fi) 1989-05-01
ES2059464T3 (es) 1994-11-16
IE65989B1 (en) 1995-11-29
EP0313874A3 (en) 1990-05-09
JPH01193282A (ja) 1989-08-03
ATE104309T1 (de) 1994-04-15
NO884833L (no) 1989-05-02
NO173506B (no) 1993-09-13
AR246083A1 (es) 1994-03-30
DE3851682T2 (de) 1995-05-04
IL87947A (en) 1995-05-26
DK602488D0 (da) 1988-10-28
IL87946A (en) 1995-06-29
DK174739B1 (da) 2003-10-13
JP2720933B2 (ja) 1998-03-04
AU618763B2 (en) 1992-01-09
FI884983A0 (fi) 1988-10-28
ES2061586T3 (es) 1994-12-16
NO884833D0 (no) 1988-10-28
IL87946A0 (en) 1989-03-31
ZA888123B (en) 1989-07-26
NO173506C (no) 1993-12-22
DE3889063D1 (de) 1994-05-19
HK131997A (en) 1997-10-03
IE65053B1 (en) 1995-10-04
EP0313873B1 (de) 1994-09-28
FI91262C (fi) 1994-06-10
PT88881B (pt) 1993-01-29
DK602588A (da) 1989-05-01

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Legal Events

Date Code Title Description
EELA Cancelled due to lapse of time