AR103323A1 - Derivados de glucagón - Google Patents

Derivados de glucagón

Info

Publication number
AR103323A1
AR103323A1 ARP150104341A ARP150104341A AR103323A1 AR 103323 A1 AR103323 A1 AR 103323A1 AR P150104341 A ARP150104341 A AR P150104341A AR P150104341 A ARP150104341 A AR P150104341A AR 103323 A1 AR103323 A1 AR 103323A1
Authority
AR
Argentina
Prior art keywords
glucagon
peptide
treat obesity
receptors
glucagon derivatives
Prior art date
Application number
ARP150104341A
Other languages
English (en)
Inventor
Suk Lee Jong
Jin Park Young
Youb Jung Sung
Chang Kwon Se
Ki Lim Chang
Hyuk Choi Jae
Original Assignee
Hanmi Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hanmi Pharm Ind Co Ltd filed Critical Hanmi Pharm Ind Co Ltd
Publication of AR103323A1 publication Critical patent/AR103323A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/605Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/26Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente se refiere a un péptido de un derivado de glucagón y una composición para prevenir o tratar la obesidad que comprende el péptido como un ingrediente activo. El derivado de glucagón de acuerdo con la presente muestra un efecto activador más excelente con respecto a receptores de péptido 1 tipo glucagón y receptores de glucagón en comparación con glucagón nativo, y en consecuencia se pueden usar ampliamente como un agente efectivo para tratar obesidad.
ARP150104341A 2014-12-30 2015-12-30 Derivados de glucagón AR103323A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1020140193691A KR102418477B1 (ko) 2014-12-30 2014-12-30 글루카곤 유도체

Publications (1)

Publication Number Publication Date
AR103323A1 true AR103323A1 (es) 2017-05-03

Family

ID=56284668

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150104341A AR103323A1 (es) 2014-12-30 2015-12-30 Derivados de glucagón

Country Status (19)

Country Link
US (3) US10513550B2 (es)
EP (1) EP3240802B1 (es)
JP (1) JP6758297B2 (es)
KR (1) KR102418477B1 (es)
CN (1) CN107250155B (es)
AR (1) AR103323A1 (es)
AU (1) AU2015372767B2 (es)
BR (1) BR112017013845A2 (es)
CA (1) CA2972001A1 (es)
EA (1) EA036479B1 (es)
HK (1) HK1246323A1 (es)
IL (1) IL253001B (es)
MX (1) MX2017008715A (es)
PH (1) PH12017501205A1 (es)
SG (2) SG10201906912VA (es)
TW (1) TWI696631B (es)
UA (1) UA122967C2 (es)
WO (1) WO2016108617A1 (es)
ZA (1) ZA201704328B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
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SG11201705376SA (en) * 2014-12-30 2017-08-30 Hanmi Pharm Ind Co Ltd Glucagon derivative having improved stability
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TWI622596B (zh) 2015-10-26 2018-05-01 美國禮來大藥廠 升糖素受體促效劑
EP3398961B1 (en) 2015-12-31 2022-06-29 Hanmi Pharm. Co., Ltd. Triple activator activating glucagon, glp-1 and gip receptor
WO2024038067A1 (en) 2022-08-18 2024-02-22 Boehringer Ingelheim International Gmbh Combination therapy comprising long acting glp-1/glucagon and npy2 receptor agonists

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Also Published As

Publication number Publication date
UA122967C2 (uk) 2021-01-27
EP3240802A1 (en) 2017-11-08
EP3240802B1 (en) 2021-07-21
IL253001A0 (en) 2017-08-31
EP3240802A4 (en) 2018-10-10
SG11201705130XA (en) 2017-07-28
US10513550B2 (en) 2019-12-24
CN107250155A (zh) 2017-10-13
EA036479B1 (ru) 2020-11-16
AU2015372767A1 (en) 2017-07-13
US20200140515A1 (en) 2020-05-07
BR112017013845A2 (pt) 2018-01-02
CN107250155B (zh) 2021-08-10
IL253001B (en) 2022-04-01
EA201791498A1 (ru) 2017-10-31
AU2015372767B2 (en) 2020-07-16
TWI696631B (zh) 2020-06-21
US11254724B2 (en) 2022-02-22
ZA201704328B (en) 2021-01-27
CA2972001A1 (en) 2016-07-07
TW201632546A (zh) 2016-09-16
US20180002395A1 (en) 2018-01-04
WO2016108617A1 (en) 2016-07-07
KR20160082026A (ko) 2016-07-08
PH12017501205A1 (en) 2017-10-18
SG10201906912VA (en) 2019-09-27
JP2018505153A (ja) 2018-02-22
US20220025012A1 (en) 2022-01-27
MX2017008715A (es) 2017-11-17
JP6758297B2 (ja) 2020-09-23
KR102418477B1 (ko) 2022-07-08
HK1246323A1 (zh) 2018-09-07

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