AR028621A1 - Antagonistas receptores de adenosina a2a - Google Patents

Antagonistas receptores de adenosina a2a

Info

Publication number
AR028621A1
AR028621A1 ARP010102483A ARP010102483A AR028621A1 AR 028621 A1 AR028621 A1 AR 028621A1 AR P010102483 A ARP010102483 A AR P010102483A AR P010102483 A ARP010102483 A AR P010102483A AR 028621 A1 AR028621 A1 AR 028621A1
Authority
AR
Argentina
Prior art keywords
adenosine
antagonists
receiving
receiving antagonists
Prior art date
Application number
ARP010102483A
Other languages
English (en)
Spanish (es)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of AR028621A1 publication Critical patent/AR028621A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ARP010102483A 2000-05-26 2001-05-24 Antagonistas receptores de adenosina a2a AR028621A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US20714300P 2000-05-26 2000-05-26

Publications (1)

Publication Number Publication Date
AR028621A1 true AR028621A1 (es) 2003-05-14

Family

ID=22769372

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP010102483A AR028621A1 (es) 2000-05-26 2001-05-24 Antagonistas receptores de adenosina a2a

Country Status (31)

Country Link
US (4) US6630475B2 (enExample)
EP (1) EP1283839B1 (enExample)
JP (3) JP4574112B2 (enExample)
KR (1) KR100520907B1 (enExample)
CN (2) CN100384847C (enExample)
AR (1) AR028621A1 (enExample)
AT (1) ATE293627T1 (enExample)
AU (2) AU2001268089C1 (enExample)
BR (1) BRPI0111015B8 (enExample)
CA (1) CA2410237C (enExample)
CZ (1) CZ303790B6 (enExample)
DE (1) DE60110219T2 (enExample)
DK (1) DK1283839T3 (enExample)
EC (1) ECSP024364A (enExample)
ES (1) ES2237576T3 (enExample)
HK (1) HK1049007B (enExample)
HU (1) HU230420B1 (enExample)
IL (3) IL152726A0 (enExample)
MX (1) MXPA02011625A (enExample)
MY (1) MY132006A (enExample)
NO (1) NO325008B1 (enExample)
NZ (1) NZ522326A (enExample)
PE (1) PE20020062A1 (enExample)
PL (1) PL218764B1 (enExample)
PT (1) PT1283839E (enExample)
RU (1) RU2315053C2 (enExample)
SI (1) SI1283839T1 (enExample)
SK (1) SK287748B6 (enExample)
TW (1) TWI288137B (enExample)
WO (1) WO2001092264A1 (enExample)
ZA (1) ZA200208898B (enExample)

Families Citing this family (89)

* Cited by examiner, † Cited by third party
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KR20200140849A (ko) * 2018-04-08 2020-12-16 베이진 엘티디 A2a 수용체 길항제로서의 피라졸로트리아졸로피리미딘 유도체
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CN110742893B (zh) * 2018-07-23 2024-04-05 百济神州(北京)生物科技有限公司 A2a受体拮抗剂治疗癌症的方法
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TWI829857B (zh) 2019-01-29 2024-01-21 美商英塞特公司 作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶
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CN112592354B (zh) 2019-07-30 2022-05-27 厦门宝太生物科技股份有限公司 一种异噁唑并嘧啶类杂环化合物的制备方法
CN112608316B (zh) 2019-07-30 2022-10-21 厦门宝太生物科技股份有限公司 一种吡唑并三嗪类腺苷受体拮抗剂
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CN117946123B (zh) * 2024-01-26 2026-06-30 北京脑重大疾病研究院 放射性三氮唑并嘧啶基衍生物及其制备方法和应用
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CN118812539B (zh) * 2024-06-19 2025-11-28 苏州大学 一种5-氨基三唑并嘧啶衍生物及其制备方法

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Also Published As

Publication number Publication date
NZ522326A (en) 2006-03-31
US6897216B2 (en) 2005-05-24
HU230420B1 (hu) 2016-05-30
KR100520907B1 (ko) 2005-10-11
DE60110219D1 (de) 2005-05-25
BR0111015A (pt) 2005-01-11
TWI288137B (en) 2007-10-11
RU2315053C2 (ru) 2008-01-20
ES2237576T3 (es) 2005-08-01
NO325008B1 (no) 2008-01-14
ZA200208898B (en) 2004-03-01
HK1049007A1 (en) 2003-04-25
JP2003535094A (ja) 2003-11-25
CN1800186A (zh) 2006-07-12
US20050026932A1 (en) 2005-02-03
PT1283839E (pt) 2005-08-31
AU2001268089C1 (en) 2006-04-13
JP2007145875A (ja) 2007-06-14
IL152726A0 (en) 2003-06-24
MXPA02011625A (es) 2003-03-27
JP2006219497A (ja) 2006-08-24
IL220174A0 (en) 2012-07-31
EP1283839B1 (en) 2005-04-20
HUP0600239A2 (en) 2006-07-28
CA2410237C (en) 2008-01-08
IL152726A (en) 2012-07-31
SK287748B6 (sk) 2011-08-04
NO20025651L (no) 2003-01-23
US20040023997A1 (en) 2004-02-05
SK16712002A3 (sk) 2003-08-05
HK1049007B (en) 2005-09-16
US6630475B2 (en) 2003-10-07
NO20025651D0 (no) 2002-11-25
CN1247588C (zh) 2006-03-29
USRE44205E1 (en) 2013-05-07
WO2001092264A1 (en) 2001-12-06
BRPI0111015B8 (pt) 2021-05-25
KR20030003746A (ko) 2003-01-10
SI1283839T1 (enExample) 2005-08-31
AU2001268089B2 (en) 2005-04-28
EP1283839A1 (en) 2003-02-19
ECSP024364A (es) 2003-03-31
CA2410237A1 (en) 2001-12-06
MY132006A (en) 2007-09-28
CN1451007A (zh) 2003-10-22
JP4574112B2 (ja) 2010-11-04
US20020099061A1 (en) 2002-07-25
IL220174A (en) 2015-07-30
AU6808901A (en) 2001-12-11
DK1283839T3 (da) 2005-07-25
US7067655B2 (en) 2006-06-27
ATE293627T1 (de) 2005-05-15
PL218764B1 (pl) 2015-01-30
HUP0600239A3 (en) 2008-06-30
CN100384847C (zh) 2008-04-30
PE20020062A1 (es) 2002-02-02
BRPI0111015B1 (pt) 2017-11-07
DE60110219T2 (de) 2006-03-09
CZ20023886A3 (cs) 2003-02-12
CZ303790B6 (cs) 2013-05-09
PL360472A1 (en) 2004-09-06
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