ZA794627B - Novel tetrazolylalkoxycarbostyril derivatives and process for producing the same - Google Patents

Novel tetrazolylalkoxycarbostyril derivatives and process for producing the same

Info

Publication number
ZA794627B
ZA794627B ZA00794627A ZA794627A ZA794627B ZA 794627 B ZA794627 B ZA 794627B ZA 00794627 A ZA00794627 A ZA 00794627A ZA 794627 A ZA794627 A ZA 794627A ZA 794627 B ZA794627 B ZA 794627B
Authority
ZA
South Africa
Prior art keywords
novel
producing
same
tetrazolylalkoxycarbostyril
derivatives
Prior art date
Application number
ZA00794627A
Other languages
English (en)
Inventor
T Nishi
K Nakagawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=14470137&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA794627(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of ZA794627B publication Critical patent/ZA794627B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
ZA00794627A 1978-09-01 1979-08-31 Novel tetrazolylalkoxycarbostyril derivatives and process for producing the same ZA794627B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP10786978A JPS5535019A (en) 1978-09-01 1978-09-01 Carbostyryl derivative

Publications (1)

Publication Number Publication Date
ZA794627B true ZA794627B (en) 1980-08-27

Family

ID=14470137

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00794627A ZA794627B (en) 1978-09-01 1979-08-31 Novel tetrazolylalkoxycarbostyril derivatives and process for producing the same

Country Status (23)

Country Link
US (1) US4277479A (de)
JP (1) JPS5535019A (de)
AR (1) AR229342A1 (de)
AT (1) AT364363B (de)
AU (1) AU538410B2 (de)
BE (1) BE878548A (de)
CA (1) CA1139761A (de)
CH (1) CH641799A5 (de)
DE (1) DE2934747A1 (de)
DK (1) DK158788C (de)
ES (1) ES483792A1 (de)
FI (1) FI68398C (de)
FR (1) FR2434809A1 (de)
GB (1) GB2033893B (de)
IT (1) IT1119929B (de)
MX (1) MX6749E (de)
NL (1) NL183888C (de)
NO (1) NO153177C (de)
PH (1) PH18452A (de)
PT (1) PT70136A (de)
SE (1) SE432252B (de)
SU (1) SU1064868A3 (de)
ZA (1) ZA794627B (de)

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JP2753622B2 (ja) 1988-05-02 1998-05-20 大塚製薬株式会社 カルボスチリル誘導体
US5064837A (en) * 1989-11-13 1991-11-12 Schering Corporation 3-substituted-1-aryl-2(h)-quinolones and their pharmaceutical compositions
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US20030045547A1 (en) 2001-05-02 2003-03-06 Shinji Aki Process for producing carbostyril derivatives
JP4060523B2 (ja) * 1999-11-24 2008-03-12 大塚製薬株式会社 カルボスチリル誘導体の製造法
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US6458804B1 (en) 2001-01-26 2002-10-01 R.T. Alamo Venturesi, Llc Methods for the treatment of central nervous system disorders in certain patient groups
US6451813B1 (en) 2001-01-26 2002-09-17 R. T. Alamo Ventures I, Llc Treatment of gastroparesis in certain patient groups
US20050101631A1 (en) * 2002-08-01 2005-05-12 Otsuka Pharmaceuticals Company Process for producing carbostyril derivatives
US7399864B2 (en) * 2001-05-02 2008-07-15 Otsuka Pharmaceutical Co., Ltd. Process for producing carbostyril derivatives
JP2003063965A (ja) * 2001-06-13 2003-03-05 Otsuka Pharmaceut Factory Inc 注射用シロスタゾール水性製剤
US6573382B2 (en) * 2001-06-29 2003-06-03 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6596871B2 (en) * 2001-06-29 2003-07-22 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1h-tetraol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
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US6388080B1 (en) 2001-06-29 2002-05-14 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
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US20080206348A1 (en) * 2004-09-17 2008-08-28 Deepak Murpani Cilostazol-Containing Pharmaceutical Composition Based On Particles Of Less Than 50 Micrometers
CN100462360C (zh) * 2005-08-15 2009-02-18 上海立科药物化学有限公司 N-环己基-5-(4-氯丁基)-1h-四氮唑的合成方法
PL1942895T3 (pl) 2005-09-15 2012-07-31 Otsuka Pharma Co Ltd Lek złożony zawierający probukol i pochodną tetrazoliloalkoksydihydrokarbostyrylu o działaniu hamującym nadtlenek
US20070105898A1 (en) * 2005-11-09 2007-05-10 Apotex Pharmachem Inc. Process for the production of cilostazol
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Also Published As

Publication number Publication date
SE7907236L (sv) 1980-03-02
SU1064868A3 (ru) 1983-12-30
ES483792A1 (es) 1980-09-01
PT70136A (en) 1979-09-01
FI68398C (fi) 1985-09-10
MX6749E (es) 1986-06-25
NO153177B (no) 1985-10-21
NL183888C (nl) 1989-02-16
DK158788B (da) 1990-07-16
DE2934747C2 (de) 1988-01-28
AU538410B2 (en) 1984-08-16
AR229342A1 (es) 1983-07-29
DE2934747A1 (de) 1980-03-13
BE878548A (fr) 1979-12-17
AU5039779A (en) 1980-03-06
JPS5535019A (en) 1980-03-11
US4277479A (en) 1981-07-07
FR2434809B1 (de) 1982-09-17
FI68398B (fi) 1985-05-31
IT7968748A0 (it) 1979-08-31
AT364363B (de) 1981-10-12
JPS6155514B2 (de) 1986-11-28
CA1139761A (en) 1983-01-18
NO792829L (no) 1980-03-04
DK158788C (da) 1990-12-10
ATA584579A (de) 1981-03-15
DK363179A (da) 1980-03-02
GB2033893B (en) 1982-12-01
GB2033893A (en) 1980-05-29
NL7906523A (nl) 1980-03-04
SE432252B (sv) 1984-03-26
NO153177C (no) 1986-01-29
IT1119929B (it) 1986-03-19
FR2434809A1 (fr) 1980-03-28
CH641799A5 (de) 1984-03-15
FI792699A (fi) 1980-03-02
PH18452A (en) 1985-07-18

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