DK363179A - Fremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater - Google Patents

Fremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater

Info

Publication number
DK363179A
DK363179A DK363179A DK363179A DK363179A DK 363179 A DK363179 A DK 363179A DK 363179 A DK363179 A DK 363179A DK 363179 A DK363179 A DK 363179A DK 363179 A DK363179 A DK 363179A
Authority
DK
Denmark
Prior art keywords
tetrazolylalcoxycarbostyric
derivatives
preparing
procedure
tetrazolylalcoxycarbostyric derivatives
Prior art date
Application number
DK363179A
Other languages
English (en)
Other versions
DK158788B (da
DK158788C (da
Inventor
T Nishi
K Nakagawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=14470137&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK363179(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of DK363179A publication Critical patent/DK363179A/da
Publication of DK158788B publication Critical patent/DK158788B/da
Application granted granted Critical
Publication of DK158788C publication Critical patent/DK158788C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
DK363179A 1978-09-01 1979-08-30 Analogifremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater DK158788C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10786978 1978-09-01
JP10786978A JPS5535019A (en) 1978-09-01 1978-09-01 Carbostyryl derivative

Publications (3)

Publication Number Publication Date
DK363179A true DK363179A (da) 1980-03-02
DK158788B DK158788B (da) 1990-07-16
DK158788C DK158788C (da) 1990-12-10

Family

ID=14470137

Family Applications (1)

Application Number Title Priority Date Filing Date
DK363179A DK158788C (da) 1978-09-01 1979-08-30 Analogifremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater

Country Status (23)

Country Link
US (1) US4277479A (da)
JP (1) JPS5535019A (da)
AR (1) AR229342A1 (da)
AT (1) AT364363B (da)
AU (1) AU538410B2 (da)
BE (1) BE878548A (da)
CA (1) CA1139761A (da)
CH (1) CH641799A5 (da)
DE (1) DE2934747A1 (da)
DK (1) DK158788C (da)
ES (1) ES483792A1 (da)
FI (1) FI68398C (da)
FR (1) FR2434809A1 (da)
GB (1) GB2033893B (da)
IT (1) IT1119929B (da)
MX (1) MX6749E (da)
NL (1) NL183888C (da)
NO (1) NO153177C (da)
PH (1) PH18452A (da)
PT (1) PT70136A (da)
SE (1) SE432252B (da)
SU (1) SU1064868A3 (da)
ZA (1) ZA794627B (da)

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JPH0681752B2 (ja) * 1986-04-02 1994-10-19 大塚製薬株式会社 カルボスチリル誘導体
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US6187790B1 (en) 1999-03-04 2001-02-13 Neal R. Cutler Use of cilostazol for treatment of sexual dysfunction
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US6458804B1 (en) * 2001-01-26 2002-10-01 R.T. Alamo Venturesi, Llc Methods for the treatment of central nervous system disorders in certain patient groups
US6451813B1 (en) 2001-01-26 2002-09-17 R. T. Alamo Ventures I, Llc Treatment of gastroparesis in certain patient groups
US20050101631A1 (en) * 2002-08-01 2005-05-12 Otsuka Pharmaceuticals Company Process for producing carbostyril derivatives
US7399864B2 (en) * 2001-05-02 2008-07-15 Otsuka Pharmaceutical Co., Ltd. Process for producing carbostyril derivatives
JP2003063965A (ja) * 2001-06-13 2003-03-05 Otsuka Pharmaceut Factory Inc 注射用シロスタゾール水性製剤
US6531603B1 (en) * 2001-06-29 2003-03-11 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6657061B2 (en) * 2001-06-29 2003-12-02 Grayson Walker Stowell Polymorphic forms of 6-[4-1(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
US6388080B1 (en) 2001-06-29 2002-05-14 Grayson Walker Stowell Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
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ITMI20031670A1 (it) * 2003-08-26 2005-02-27 Dinamite Dipharma S P A In Forma A Bbreviata Diph Processo per la preparazione di cilostazolo e di suoi intermedi.
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US20050255155A1 (en) * 2004-05-11 2005-11-17 Glenmark Pharmaceuticals Limited Modified release cilostazol compositions
WO2006030301A1 (en) * 2004-09-17 2006-03-23 Ranbaxy Laboratories Limited Cilostazol- containing pharmaceutical composition based on particles of less than 50 micrometers
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Also Published As

Publication number Publication date
PT70136A (en) 1979-09-01
BE878548A (fr) 1979-12-17
JPS5535019A (en) 1980-03-11
FI792699A (fi) 1980-03-02
FI68398C (fi) 1985-09-10
NO792829L (no) 1980-03-04
SU1064868A3 (ru) 1983-12-30
AT364363B (de) 1981-10-12
NO153177C (no) 1986-01-29
AR229342A1 (es) 1983-07-29
DK158788B (da) 1990-07-16
FI68398B (fi) 1985-05-31
FR2434809A1 (fr) 1980-03-28
GB2033893A (en) 1980-05-29
AU538410B2 (en) 1984-08-16
AU5039779A (en) 1980-03-06
MX6749E (es) 1986-06-25
NO153177B (no) 1985-10-21
DE2934747A1 (de) 1980-03-13
CA1139761A (en) 1983-01-18
JPS6155514B2 (da) 1986-11-28
PH18452A (en) 1985-07-18
NL183888C (nl) 1989-02-16
ATA584579A (de) 1981-03-15
GB2033893B (en) 1982-12-01
US4277479A (en) 1981-07-07
DE2934747C2 (da) 1988-01-28
SE432252B (sv) 1984-03-26
FR2434809B1 (da) 1982-09-17
IT1119929B (it) 1986-03-19
ES483792A1 (es) 1980-09-01
NL7906523A (nl) 1980-03-04
SE7907236L (sv) 1980-03-02
CH641799A5 (de) 1984-03-15
DK158788C (da) 1990-12-10
ZA794627B (en) 1980-08-27
IT7968748A0 (it) 1979-08-31

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