UY25472A1 - Procedimiento para la preparacion de fenoxifenilsulfonilo - Google Patents
Procedimiento para la preparacion de fenoxifenilsulfoniloInfo
- Publication number
- UY25472A1 UY25472A1 UY25472A UY25472A UY25472A1 UY 25472 A1 UY25472 A1 UY 25472A1 UY 25472 A UY25472 A UY 25472A UY 25472 A UY25472 A UY 25472A UY 25472 A1 UY25472 A1 UY 25472A1
- Authority
- UY
- Uruguay
- Prior art keywords
- procedure
- preparation
- compounds
- present
- phenoxifenylsulfonil
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C301/00—Esters of sulfurous acid
- C07C301/02—Esters of sulfurous acid having sulfite groups bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/26—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids
- C07C303/28—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids by reaction of hydroxy compounds with sulfonic acids or derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/28—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/41—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton
- C07C309/42—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton having the sulfo groups bound to carbon atoms of non-condensed six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/63—Esters of sulfonic acids
- C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/75—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton
Abstract
UN PROCEDIMIENTO PARA PREPARAR HALUROS DE FENOXIFENILSULFONILO, QUE SON INTERMEDIOS UTILES PARA LA PREPARACION DE INHIBIDORES DE LAS METALOPROTEINASAS DE LA MATRIZ. Son de utilidad para artritis, enfermedad inflamatoria del intedstino, enfermedad obstructiva crónica, asma, Alzheimer, cáncer, osteoporosis, aneurisma aortico, diabetes, etc. La presente invención se refiere a compuestos de fórmula (IIa) en la que R es H, Li, Naa, K, Mg, etc.El esquema (I) muestra la una de las preparaciones de los compuestos de la presente invención. Éster 4-fluorofenílico del ácido 4-(4-fluorofenoxi)bencenosulfónico
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8139398P | 1998-04-10 | 1998-04-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY25472A1 true UY25472A1 (es) | 1999-11-17 |
Family
ID=22163859
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY25472A UY25472A1 (es) | 1998-04-10 | 1999-04-12 | Procedimiento para la preparacion de fenoxifenilsulfonilo |
Country Status (42)
| Country | Link |
|---|---|
| US (2) | US6118016A (es) |
| EP (1) | EP0949246B1 (es) |
| JP (1) | JP3694419B2 (es) |
| KR (1) | KR100329901B1 (es) |
| CN (1) | CN1238329A (es) |
| AP (1) | AP1155A (es) |
| AR (1) | AR016205A1 (es) |
| AT (1) | ATE233729T1 (es) |
| AU (1) | AU758297B2 (es) |
| BG (1) | BG103321A (es) |
| BR (1) | BR9902041A (es) |
| CA (1) | CA2268679C (es) |
| CO (1) | CO4810300A1 (es) |
| DE (1) | DE69905633T2 (es) |
| DK (1) | DK0949246T3 (es) |
| DZ (1) | DZ2755A1 (es) |
| EA (1) | EA001756B1 (es) |
| ES (1) | ES2192021T3 (es) |
| GT (1) | GT199900044A (es) |
| HR (1) | HRP990107B1 (es) |
| HU (1) | HU221635B1 (es) |
| ID (1) | ID23645A (es) |
| IL (1) | IL129330A (es) |
| IN (1) | IN191233B (es) |
| IS (1) | IS5020A (es) |
| MA (1) | MA24834A1 (es) |
| NO (1) | NO991679L (es) |
| NZ (1) | NZ335106A (es) |
| OA (1) | OA11032A (es) |
| PA (1) | PA8469801A1 (es) |
| PE (1) | PE20000416A1 (es) |
| PL (1) | PL332452A1 (es) |
| SG (1) | SG75169A1 (es) |
| SI (1) | SI0949246T1 (es) |
| SK (1) | SK44999A3 (es) |
| TN (1) | TNSN99051A1 (es) |
| TR (1) | TR199900757A2 (es) |
| TW (1) | TW539664B (es) |
| UA (1) | UA59373C2 (es) |
| UY (1) | UY25472A1 (es) |
| YU (1) | YU18299A (es) |
| ZA (1) | ZA992628B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6458822B2 (en) | 2000-03-13 | 2002-10-01 | Pfizer Inc. | 2-oxo-imidazolidine-4-carboxylic acid hydroxamide compounds that inhibit matrix metalloproteinases |
| ES2425013T3 (es) * | 2002-06-12 | 2013-10-10 | Symphony Evolution, Inc. | Inhibidores de ADAM-10 humana |
| JP2006516548A (ja) | 2002-12-30 | 2006-07-06 | アンジオテック インターナショナル アクツィエン ゲゼルシャフト | 迅速ゲル化ポリマー組成物からの薬物送達法 |
| JP5830534B2 (ja) | 2010-07-09 | 2015-12-09 | ファイザー・リミテッドＰｆｉｚｅｒ Ｌｉｍｉｔｅｄ | 化合物 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE844004C (de) * | 1944-08-06 | 1952-07-14 | Cassella Farbwerke Mainkur Ag | Verfahren zur Herstellung von Sulfonsaeureestern |
| US4032506A (en) * | 1973-12-28 | 1977-06-28 | General Electric Company | Flame retardant polycarbonate composition |
| ZA794723B (en) * | 1978-09-11 | 1980-08-27 | Univ Miami | Anti-hypertensive agents |
| GB9000725D0 (en) * | 1990-01-12 | 1990-03-14 | Pfizer Ltd | Therapeutic agents |
| US5340489A (en) * | 1992-06-05 | 1994-08-23 | The Dow Chemical Company | Aryl arenesulfonates and a method of lubrication using the aryl arenesulfonates |
| US5863949A (en) * | 1995-03-08 | 1999-01-26 | Pfizer Inc | Arylsulfonylamino hydroxamic acid derivatives |
| US6153609A (en) * | 1996-08-23 | 2000-11-28 | Pfizer Inc | Arylsulfonylamino hydroxamic acid derivatives |
| TR199901849T2 (xx) * | 1997-02-03 | 2000-02-21 | Pfizer Products Inc. | Arils�lfonilamino hidroksamik asit t�revleri. |
| WO1998050348A1 (en) * | 1997-05-09 | 1998-11-12 | Agouron Pharmaceuticals, Inc. | Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses |
| ATE217863T1 (de) * | 1997-08-08 | 2002-06-15 | Pfizer Prod Inc | Arylsulfonylaminohydroxamsäurederivate |
| ATE263147T1 (de) * | 1997-08-08 | 2004-04-15 | Pfizer Prod Inc | Derivate von aryloxyarylsulfonylamino hydroxyaminsäuren |
| PA8469401A1 (es) * | 1998-04-10 | 2000-05-24 | Pfizer Prod Inc | Derivados biciclicos del acido hidroxamico |
-
1999
- 1999-03-24 GT GT199900044A patent/GT199900044A/es unknown
- 1999-03-26 PA PA19998469801A patent/PA8469801A1/es unknown
- 1999-04-01 OA OA9900075A patent/OA11032A/en unknown
- 1999-04-05 IL IL12933099A patent/IL129330A/xx not_active IP Right Cessation
- 1999-04-06 IS IS5020A patent/IS5020A/is unknown
- 1999-04-06 SK SK449-99A patent/SK44999A3/sk unknown
- 1999-04-06 PE PE1999000276A patent/PE20000416A1/es not_active Application Discontinuation
- 1999-04-06 TW TW088105444A patent/TW539664B/zh not_active IP Right Cessation
- 1999-04-06 IN IN511DE1999 patent/IN191233B/en unknown
- 1999-04-07 MA MA25531A patent/MA24834A1/fr unknown
- 1999-04-07 TN TNTNSN99051A patent/TNSN99051A1/fr unknown
- 1999-04-07 JP JP10000199A patent/JP3694419B2/ja not_active Expired - Fee Related
- 1999-04-07 KR KR1019990011940A patent/KR100329901B1/ko not_active IP Right Cessation
- 1999-04-07 US US09/287,930 patent/US6118016A/en not_active Expired - Fee Related
- 1999-04-07 DZ DZ990056A patent/DZ2755A1/xx active
- 1999-04-08 SI SI9930219T patent/SI0949246T1/xx unknown
- 1999-04-08 YU YU18299A patent/YU18299A/sh unknown
- 1999-04-08 SG SG1999001821A patent/SG75169A1/en unknown
- 1999-04-08 UA UA99042000A patent/UA59373C2/uk unknown
- 1999-04-08 ES ES99302744T patent/ES2192021T3/es not_active Expired - Lifetime
- 1999-04-08 DE DE69905633T patent/DE69905633T2/de not_active Expired - Fee Related
- 1999-04-08 AT AT99302744T patent/ATE233729T1/de not_active IP Right Cessation
- 1999-04-08 EP EP99302744A patent/EP0949246B1/en not_active Expired - Lifetime
- 1999-04-08 DK DK99302744T patent/DK0949246T3/da active
- 1999-04-08 TR TR1999/00757A patent/TR199900757A2/xx unknown
- 1999-04-08 CA CA002268679A patent/CA2268679C/en not_active Expired - Fee Related
- 1999-04-08 AR ARP990101602A patent/AR016205A1/es unknown
- 1999-04-08 ID IDP990311D patent/ID23645A/id unknown
- 1999-04-08 AP APAP/P/1999/001509A patent/AP1155A/en active
- 1999-04-09 HU HU9901042A patent/HU221635B1/hu not_active IP Right Cessation
- 1999-04-09 PL PL99332452A patent/PL332452A1/xx unknown
- 1999-04-09 EA EA199900282A patent/EA001756B1/ru not_active IP Right Cessation
- 1999-04-09 NZ NZ335106A patent/NZ335106A/xx unknown
- 1999-04-09 BG BG103321A patent/BG103321A/xx unknown
- 1999-04-09 AU AU23692/99A patent/AU758297B2/en not_active Ceased
- 1999-04-09 CN CN99104929A patent/CN1238329A/zh active Pending
- 1999-04-09 HR HR990107A patent/HRP990107B1/xx not_active IP Right Cessation
- 1999-04-09 ZA ZA9902628A patent/ZA992628B/xx unknown
- 1999-04-09 NO NO991679A patent/NO991679L/no not_active Application Discontinuation
- 1999-04-12 CO CO99021410A patent/CO4810300A1/es unknown
- 1999-04-12 BR BR9902041-6A patent/BR9902041A/pt not_active IP Right Cessation
- 1999-04-12 UY UY25472A patent/UY25472A1/es unknown
-
2000
- 2000-12-19 US US09/740,398 patent/US20010011143A1/en not_active Abandoned
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| DESI | Application deemed to be withdrawn |
Effective date: 20071105 |