EA199900282A2 - Способ получения феноксифенилсульфонилгалогенидов - Google Patents

Способ получения феноксифенилсульфонилгалогенидов

Info

Publication number
EA199900282A2
EA199900282A2 EA199900282A EA199900282A EA199900282A2 EA 199900282 A2 EA199900282 A2 EA 199900282A2 EA 199900282 A EA199900282 A EA 199900282A EA 199900282 A EA199900282 A EA 199900282A EA 199900282 A2 EA199900282 A2 EA 199900282A2
Authority
EA
Eurasian Patent Office
Prior art keywords
halides
phenoxyphenylsulfonyl halides
process foe
preparing phenoxyphenylsulfonyl
foe preparing
Prior art date
Application number
EA199900282A
Other languages
English (en)
Other versions
EA001756B1 (ru
EA199900282A3 (ru
Inventor
Джоел Майкл Хокинс
Original Assignee
Пфайзер Продактс Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Пфайзер Продактс Инк. filed Critical Пфайзер Продактс Инк.
Publication of EA199900282A2 publication Critical patent/EA199900282A2/ru
Publication of EA199900282A3 publication Critical patent/EA199900282A3/ru
Publication of EA001756B1 publication Critical patent/EA001756B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C301/00—Esters of sulfurous acid
    • C07C301/02—Esters of sulfurous acid having sulfite groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/32—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of salts of sulfonic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/02—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of sulfonic acids or halides thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/26—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids
    • C07C303/28—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids by reaction of hydroxy compounds with sulfonic acids or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/28—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/41—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton
    • C07C309/42—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton having the sulfo groups bound to carbon atoms of non-condensed six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/75—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing singly-bound oxygen atoms bound to the carbon skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Настоящее изобретение относится к способу получения феноксифенилсульфонилгалогенидов, которые полезны в качестве промежуточных соединений для получения ингибиторов матричных металлопротеиназ.
EA199900282A 1998-04-10 1999-04-09 Феноксифенилсульфонилгалогениды и способ их получения EA001756B1 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8139398P 1998-04-10 1998-04-10

Publications (3)

Publication Number Publication Date
EA199900282A2 true EA199900282A2 (ru) 1999-10-28
EA199900282A3 EA199900282A3 (ru) 2000-04-24
EA001756B1 EA001756B1 (ru) 2001-08-27

Family

ID=22163859

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199900282A EA001756B1 (ru) 1998-04-10 1999-04-09 Феноксифенилсульфонилгалогениды и способ их получения

Country Status (42)

Country Link
US (2) US6118016A (ru)
EP (1) EP0949246B1 (ru)
JP (1) JP3694419B2 (ru)
KR (1) KR100329901B1 (ru)
CN (1) CN1238329A (ru)
AP (1) AP1155A (ru)
AR (1) AR016205A1 (ru)
AT (1) ATE233729T1 (ru)
AU (1) AU758297B2 (ru)
BG (1) BG103321A (ru)
BR (1) BR9902041A (ru)
CA (1) CA2268679C (ru)
CO (1) CO4810300A1 (ru)
DE (1) DE69905633T2 (ru)
DK (1) DK0949246T3 (ru)
DZ (1) DZ2755A1 (ru)
EA (1) EA001756B1 (ru)
ES (1) ES2192021T3 (ru)
GT (1) GT199900044A (ru)
HR (1) HRP990107B1 (ru)
HU (1) HU221635B1 (ru)
ID (1) ID23645A (ru)
IL (1) IL129330A (ru)
IN (1) IN191233B (ru)
IS (1) IS5020A (ru)
MA (1) MA24834A1 (ru)
NO (1) NO991679L (ru)
NZ (1) NZ335106A (ru)
OA (1) OA11032A (ru)
PA (1) PA8469801A1 (ru)
PE (1) PE20000416A1 (ru)
PL (1) PL332452A1 (ru)
SG (1) SG75169A1 (ru)
SI (1) SI0949246T1 (ru)
SK (1) SK44999A3 (ru)
TN (1) TNSN99051A1 (ru)
TR (1) TR199900757A2 (ru)
TW (1) TW539664B (ru)
UA (1) UA59373C2 (ru)
UY (1) UY25472A1 (ru)
YU (1) YU18299A (ru)
ZA (1) ZA992628B (ru)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458822B2 (en) 2000-03-13 2002-10-01 Pfizer Inc. 2-oxo-imidazolidine-4-carboxylic acid hydroxamide compounds that inhibit matrix metalloproteinases
WO2003106381A2 (en) * 2002-06-12 2003-12-24 Exelixis, Inc. Human adam-10 inhibitors
AU2003300076C1 (en) 2002-12-30 2010-03-04 Angiotech International Ag Drug delivery from rapid gelling polymer composition
JP5830534B2 (ja) 2010-07-09 2015-12-09 ファイザー・リミテッドＰｆｉｚｅｒ Ｌｉｍｉｔｅｄ 化合物

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE844004C (de) * 1944-08-06 1952-07-14 Cassella Farbwerke Mainkur Ag Verfahren zur Herstellung von Sulfonsaeureestern
US4032506A (en) * 1973-12-28 1977-06-28 General Electric Company Flame retardant polycarbonate composition
ZA794723B (en) * 1978-09-11 1980-08-27 Univ Miami Anti-hypertensive agents
GB9000725D0 (en) * 1990-01-12 1990-03-14 Pfizer Ltd Therapeutic agents
US5340489A (en) * 1992-06-05 1994-08-23 The Dow Chemical Company Aryl arenesulfonates and a method of lubrication using the aryl arenesulfonates
US5863949A (en) * 1995-03-08 1999-01-26 Pfizer Inc Arylsulfonylamino hydroxamic acid derivatives
TR199900387T2 (xx) * 1996-08-23 1999-04-21 Pfizer Inc. Arils�lfonilamino hidroksamik asit t�revleri.
EA002594B1 (ru) * 1997-02-03 2002-06-27 Пфайзер Продактс Инк. Производные арилсульфониламиногидроксамовой кислоты
AU7294098A (en) * 1997-05-09 1998-11-27 Agouron Pharmaceuticals, Inc. Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
ATE217863T1 (de) * 1997-08-08 2002-06-15 Pfizer Prod Inc Arylsulfonylaminohydroxamsäurederivate
PT1003720E (pt) * 1997-08-08 2004-07-30 Pfizer Prod Inc Derivados de acido ariloxiarilsulfonilamino hidroxamico
PA8469401A1 (es) * 1998-04-10 2000-05-24 Pfizer Prod Inc Derivados biciclicos del acido hidroxamico

Also Published As

Publication number Publication date
KR19990082980A (ko) 1999-11-25
US6118016A (en) 2000-09-12
HU9901042D0 (en) 1999-06-28
PL332452A1 (en) 1999-10-11
IS5020A (is) 1999-10-11
DE69905633T2 (de) 2003-11-06
CA2268679C (en) 2004-07-27
TNSN99051A1 (fr) 2005-11-10
HRP990107B1 (en) 2003-10-31
GT199900044A (es) 2000-09-14
EP0949246A1 (en) 1999-10-13
IL129330A (en) 2003-12-10
ES2192021T3 (es) 2003-09-16
AP9901509A0 (en) 1999-06-30
JP3694419B2 (ja) 2005-09-14
SI0949246T1 (en) 2003-06-30
UY25472A1 (es) 1999-11-17
ID23645A (id) 2000-05-04
PA8469801A1 (es) 2000-09-29
KR100329901B1 (ko) 2002-03-22
MA24834A1 (fr) 1999-12-31
US20010011143A1 (en) 2001-08-02
EA001756B1 (ru) 2001-08-27
AP1155A (en) 2003-06-30
YU18299A (sh) 2002-11-15
UA59373C2 (ru) 2003-09-15
IN191233B (ru) 2003-10-11
CN1238329A (zh) 1999-12-15
SG75169A1 (en) 2000-09-19
HUP9901042A3 (en) 2000-06-28
ATE233729T1 (de) 2003-03-15
HU221635B1 (hu) 2002-12-28
EA199900282A3 (ru) 2000-04-24
TR199900757A3 (tr) 1999-11-22
NO991679D0 (no) 1999-04-09
PE20000416A1 (es) 2000-05-24
AR016205A1 (es) 2001-06-20
IL129330A0 (en) 2000-02-17
TR199900757A2 (xx) 1999-11-22
HRP990107A2 (en) 2000-02-29
EP0949246B1 (en) 2003-03-05
AU2369299A (en) 1999-10-21
NZ335106A (en) 2000-09-29
HUP9901042A2 (hu) 1999-12-28
CA2268679A1 (en) 1999-10-10
DZ2755A1 (fr) 2003-09-15
SK44999A3 (en) 2000-09-12
OA11032A (en) 2002-02-06
TW539664B (en) 2003-07-01
AU758297B2 (en) 2003-03-20
CO4810300A1 (es) 1999-06-30
JPH11322704A (ja) 1999-11-24
BR9902041A (pt) 2000-05-02
BG103321A (en) 2001-08-31
ZA992628B (en) 2000-10-09
NO991679L (no) 1999-10-11
DK0949246T3 (da) 2003-04-07
DE69905633D1 (de) 2003-04-10

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU